Collect. Czech. Chem. Commun.
1983, 48, 1212-1223
https://doi.org/10.1135/cccc19831212
Oxidative transformations of some pyrimidine derivatives into oxazolidine derivatives
Jiří Křepelka, Vladimír Pouzar, Jiří Schlanger, Jiří Holubek, Jiří Körbl, Fedir Jančik and Rudolf Kotva
Research Institute for Pharmacy and Biochemistry, 130 60 Prague 3
Individual author index pages
Other CCCC articles of these authors
- Eva Šťastná, Hana Chodounská*, Vladimír Pouzar, Jiřina Borovská and Ladislav Vyklický, Jr.
Synthesis of pregnane 3-carboxylic acids via Pd-catalyzed alkoxycarbonylation and their effect on NMDA receptor activity
2011, Vol. 76, Issue 9, pp. 1141–1161 [Abstract] - Vojtěch Kapras, Eva Šťastná, Hana Chodounská*, Vladimír Pouzar and Zdena Krištofíková
Preparation of steroid sulfamates and their interaction with GABAA receptor
2009, Vol. 74, Issue 4, pp. 643–650 [Abstract] - Pavel Herrmann, Jaroslav Kvíčala, Vladimír Pouzar and Hana Chodounská*
Synthesis of Fluorinated Steroids Using a Novel Fluorinating Reagent Tetrabutylammonium Difluorodimethylphenylsilicate (TAMPS)
2008, Vol. 73, Issue 12, pp. 1825–1834 [Abstract] - Ivan Černý, Helena Havlíková, Martin Hill, Richard Hampl and Vladimír Pouzar*
Synthetic Approach to 5α-Pregnanolone 19-[O-(Carboxymethyl)oxime] Derivatives
2004, Vol. 69, Issue 9, pp. 1805–1817 [Abstract] - Miroslav Reschel, Miloš Buděšínský, Ivan Černý, Vladimír Pouzar and Pavel Drašar*
Synthesis of Linear Steroid Oligoesters Based on Etienic Acid
2002, Vol. 67, Issue 11, pp. 1709–1718 [Abstract] - Martin Hill*, Helena Havlíková, Jan Klak, Marie Bičíková, Vladimír Pouzar, Richard Hampl and Luboslav Stárka
Rapid Immunoassay for Pregnenolone Sulfate and Its Applications in Endocrinology
2002, Vol. 67, Issue 1, pp. 140–162 [Abstract] - Ivan Černý*, Miloš Buděšínský, Vladimír Pouzar and Pavel Drašar
Linear Chaining of Etienic Acid Derivatives with the Amide Bond. Synthesis of Oligomeric Steroids
2001, Vol. 66, Issue 6, pp. 933–946 [Abstract] - Ivan Černý*, Vladimír Pouzar, Miloš Buděšínský and Pavel Drašar
Synthesis of Symmetrical Bis-Steroid Pyrazines Connected via D-Rings
2000, Vol. 65, Issue 10, pp. 1597–1608 [Abstract] - Vladimír Pouzar*, Ivan Černý and Pavel Drašar
Coupling of Steroid O-(Carboxymethyl)oxime Derivatives with Single-Protected α,ω-Diaminoalkanes
1999, Vol. 64, Issue 12, pp. 2035–2043 [Abstract] - Vladimír Pouzar, Tereza Slavíková and Ivan Černý
Lengthening of the Alkyl Chain in Steroid O-(ω-Carboxyalkyl)oximes by Wittig Reaction
1998, Vol. 63, Issue 10, pp. 1623–1634 [Abstract] - Tereza Slavíková, Vladimír Pouzar and Ivan Černý
Synthesis of Steroid O-(ω-Hydroxyalkyl)oximes by Reduction of Corresponding O-(ω-Carboxyalkyl)oxime Derivatives
1998, Vol. 63, Issue 4, pp. 557–576 [Abstract] - Ivan Černý, Vladimír Pouzar, Oldřich Lapčík and Richard Hampl
Addition of Azoimide to Unsaturated Ketones in the Steroid Series. Synthesis of N-(17β-Hydroxy-3-oxo-5α-androstan-15β-yl)succinamoic Acid and Its Evaluation as Hapten for Dihydrotestosterone Immunoanalysis
1997, Vol. 62, Issue 12, pp. 1931–1939 [Abstract] - Ivan Černý, Tereza Slavíková and Vladimír Pouzar
Synthesis of (15E)-17β-hydroxy-5α-androstane-3,15-dione 15-[O-(Carboxymethyl)]oxime, New Hapten for Dihydrotestosterone (17β-hydroxy-5α-androstan-3-one)
1997, Vol. 62, Issue 10, pp. 1642–1649 [Abstract] - Tereza Slavíková, Vladimír Pouzar and Ivan Černý
Syntheses of Steroid O-(3-Carboxypropyl)oximes
1997, Vol. 62, Issue 3, pp. 457–470 [Abstract] - Vladimír Pouzar, Tereza Slavíková and Ivan Černý
Synthesis of (19E)-3β,7β-Dihydroxy-17-oxoandrost-5-en-19-al 19-(O-Carboxymethyl)oxime, New Hapten for 7β-Hydroxydehydroepiandrosterone (3β,7β-Dihydroxyandrost-5-en-17-one)
1997, Vol. 62, Issue 1, pp. 109–123 [Abstract] - Jan Fajkoš, Vladimír Pouzar and Ivan Černý
Synthesis of (15E)-3β-Hydroxyandrost-5-ene-15,17-dione 15-(O-Carboxymethyl)oxime; The New Hapten for 3β-Hydroxyandrost-5-en-17-one (Dehydroepiandrosterone, DHEA)
1996, Vol. 61, Issue 11, pp. 1647–1654 [Abstract] - Oldřich Lapčík, Richard Hampl, Martin Hill, Luboslav Stárka, Alexander Kasal, Vladimír Pouzar and Zdeněk Putz
Radioimmunological and Chromatographic Properties of Tyrosine Methyl Ester Conjugates with Stereoisomeric Steroid Carboxy Derivatives
1996, Vol. 61, Issue 5, pp. 799–807 [Abstract] - Vladimír Pouzar, Tereza Slavíková and Ivan Černý
Preparation of 7-[O-(Carboxymethyl)oxime] Derivatives of Dehydroepiandrosterone and Pregnenolone
1996, Vol. 61, Issue 3, pp. 404–412 [Abstract] - Vladimír Pouzar and Ivan Černý
Coupling of Steroid O-(Carboxymethyl)oxime Derivatives with Amino Alcohols
1996, Vol. 61, Issue 2, pp. 288–297 [Abstract] - Jasmina Novakovic, Eva Tvrzická, Václav Všetečka, Vladimír Pouzar and Ladislav Feltl
Capillary Gas-Chromatographic Retention Behavior and Physico-Chemical Properties of Underivatized Equine Estrogens
1995, Vol. 60, Issue 5, pp. 813–819 [Abstract] - Vladimír Pouzar and Ivan Černý
Preparation of (20E)-21-Ethoxycarbonyl-14β,17α-pregna-5,20-dien-3β-yl Hydrogen Butanedioate
1995, Vol. 60, Issue 4, pp. 715–718 [Abstract] - Vladimír Pouzar and Ivan Černý
17-(O-(2-Carboxyethyl)oxime) Derivatives of Androstanes of 3-Hydroxy-5α-, -5β-, -5-ene and 3-Oxo-4-ene Series
1995, Vol. 60, Issue 1, pp. 137–149 [Abstract] - Ivan Černý, Miloš Buděšínský, Pavel Drašar and Vladimír Pouzar
Construction of the Side-Chain in 14β-Androst-5-ene Derivatives. Preparation of 14β-Pregnenolone
1994, Vol. 59, Issue 12, pp. 2691–2704 [Abstract] - Vladimír Pouzar and Ivan Černý
Preparation of (17E)-3β-Hydroxyandrost-5-en-17-one (O-Carboxymethyl)oxime Derivatives with Short Peptide Chain
1994, Vol. 59, Issue 9, pp. 2042–2056 [Abstract] - Rudolf Kotva, Jindřich Pytela and František Rypáček
Synthesis of N2-[N5-(2-Hydroxyethyl)-L-glutaminyl]-N5-(2-hydroxyethyl)-L-glutamine
1994, Vol. 59, Issue 8, pp. 1897–1900 [Abstract] - Hana Chodounská and Vladimír Pouzar
Preparation of 3-(6-Deoxy-β-D-glucopyranosyloxy) and 3-(6-Deoxy-α-L-mannopyranosyloxy)androstane Derivatives with Unsaturated Side Chain in Position 17β
1993, Vol. 58, Issue 12, pp. 3000–3008 [Abstract] - Vladimír Pouzar, Ivan Černý and Pavel Drašar
Acrylate Side Chain Derivatives of 5β-Steroids
1993, Vol. 58, Issue 12, pp. 2963–2976 [Abstract] - Libuše Arnoštová, Ivan Černý, Vladimír Pouzar and Pavel Drašar
Synthesis of 5α-Cholestane Type Glycoside Sulfates
1993, Vol. 58, Issue 5, pp. 1180–1190 [Abstract] - Alexander Kasal, Květa Fuksová and Vladimír Pouzar
Preparation of Unlabelled and [3H]-Labelled Epitestosterone and Its Metabolites
1993, Vol. 58, Issue 3, pp. 600–611 [Abstract] - Vladimír Pouzar, Ivan Černý and Pavel Drašar
Z-Isomers of Steroid 17β-Side Chain Methyl Acrylates
1992, Vol. 57, Issue 9, pp. 1928–1936 [Abstract] - Lenka Schneiderová, Oldřich Štrouf, Bohumír Grüner, Vladimír Pouzar, Pavel Drašar, Richard Hampl and Irena Kimlová
Synthesis of o-Carboranylmethyl Ethers of Steroids as Potential Target Substrates for Boron Neutron Capture Therapy
1992, Vol. 57, Issue 3, pp. 463–471 [Abstract] - Ivan Černý, Vladimír Pouzar, Pavel Drašar and Miroslav Havel
Glucosylation of Some Steroidal 17-Hydroxy Derivatives
1992, Vol. 57, Issue 2, pp. 362–374 [Abstract] - Vladimír Pouzar, Hana Chodounská, Ivan Černý and Pavel Drašar
Derivatives of 5α-androstan-3α- and 3β-ol with acrylonitrile side chain
1991, Vol. 56, Issue 12, pp. 2906–2916 [Abstract] - Jan Fajkoš and Vladimír Pouzar
Synthesis of (19E)-17β-hydroxy-3-oxo-5α-androstan-19-al 19-(O-carboxymethyl)oxime
1991, Vol. 56, Issue 12, pp. 2884–2891 [Abstract] - Jan Fajkoš, Vladimír Pouzar and Karel Vereš
Synthesis of (19E)-3,20-dioxopregn-4-en-19-al 19-(O-carboxymethyl)oxime
1991, Vol. 56, Issue 5, pp. 1087–1092 [Abstract] - Karel Šindelář, Josef Pomykáček, Jiří Holubek, Emil Svátek, Martin Valchář, Karel Dobrovský, Jiřina Metyšová and Zdeněk Polívka
Potential antidepressants and selective inhibitors of 5-hydroxytryptamine re-uptake in the brain: Synthesis of several potential metabolites of moxifetin and of two A-ring fluorinated analogues
1991, Vol. 56, Issue 2, pp. 459–477 [Abstract] - Vladimír Valenta, Jiří Holubek, Emil Svátek, Martin Valchář, Ivan Krejčí and Miroslav Protiva
Potential nootropic agents: Synthesis of some (2-oxo-1-pyrrolidinyl)acetamides and some related compounds
1990, Vol. 55, Issue 11, pp. 2756–2764 [Abstract] - Ivan Černý, Vladimír Pouzar, Miloš Buděšínský, Pavel Drašar and Miroslav Havel
Epimeric 17-hydroxy derivatives of 14β-androst-5-en-3β-yl acetate
1990, Vol. 55, Issue 10, pp. 2510–2520 [Abstract] - Vladimír Valenta, Jiří Holubek, Emil Svátek and Miroslav Protiva
Potential cholinergic and anticholinergic compounds: Synthesis of 2,8-substituted 2,8-diazaspiro[4,5]decane-1,3-diones
1990, Vol. 55, Issue 9, pp. 2304–2316 [Abstract] - Karel Šindelář, Jiří Jílek, Josef Pomykáček, Vladimír Valenta, Marta Hrubantová, Marie Vlková, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiřina Metyšová and Miroslav Protiva
Tricyclic neuroleptics: Synthesis of metabolites of isofloxythepin and some related compounds
1990, Vol. 55, Issue 9, pp. 2282–2303 [Abstract] - Jan Fajkoš, Vladimír Pouzar and Karel Vereš
Synthesis of (19E)-17β-hydroxy-3-oxoandrost-4-en-19-al 19-(O-carboxymethyl)oxime
1990, Vol. 55, Issue 8, pp. 2086–2094 [Abstract] - Jiří Jílek, Miroslav Rajšner, Vladimír Valenta, Miloš Borovička, Jiří Holubek, Miroslav Ryska, Emil Svátek, Jan Metyš and Miroslav Protiva
Synthesis of piperidine derivatives as potential analgetic agents
1990, Vol. 55, Issue 7, pp. 1828–1853 [Abstract] - Vojtěch Kmoníček, Emil Svátek, Jiří Holubek, Miroslav Ryska, Martin Valchář and Miroslav Protiva
Synthesis of 1-acyl- and 1-(thioacyl)-4-benzylpiperazines as potential antidepressants
1990, Vol. 55, Issue 7, pp. 1817–1827 [Abstract] - Hana Chodounská and Vladimír Pouzar
Preparation of 3-(β-D-galactopyranosyloxy)androstane derivatives with unsaturated side chain in position 17β
1990, Vol. 55, Issue 6, pp. 1639–1646 [Abstract] - Vladimír Pouzar, Ivan Černý, Pavel Drašar and Miroslav Havel
Preparation of (20E)-21-ethoxycarbonyl-5β-pregn-20-en-3β-yl hydrogen butanedioate
1990, Vol. 55, Issue 6, pp. 1635–1638 [Abstract] - Vladimír Valenta, Karel Šindelář, Jiří Holubek, Miroslav Ryska, Ivan Krejčí, Antonín Dlabač and Miroslav Protiva
Potential nootropic agents: Synthesis of a series of (2-oxo-1-pyrrolidinyl)acetic acid piperazides
1990, Vol. 55, Issue 6, pp. 1613–1629 [Abstract] - Karel Šindelář, Jiří Holubek, Ivan Koruna, Marta Hrubantová and Miroslav Protiva
Modified syntheses of 2-(methylthio)-10-(2-(1-methyl-2-piperidinyl)ethyl)phenothiazine (thioridazine) and 1-(3-(2-(methylsulfonyl)-10-phenothiazinyl)propyl)-piperidine-4-carboxamide (metopimazine)
1990, Vol. 55, Issue 6, pp. 1586–1601 [Abstract] - Vladimír Valenta, Jiří Holubek, Emil Svátek, Oluše Matoušová, Jiřina Metyšová and Miroslav Protiva
Potential neuroleptics of the orthopramide series; synthesis of heterocyclic 5-amino-2-methoxybenzamides and of some related compounds
1990, Vol. 55, Issue 5, pp. 1297–1310 [Abstract] - Miroslav Protiva, Vladimír Valenta, Zdeňka Kopicová, Juraj Lukáč, Jiří Holubek and Ivan Krejčí
Potential cerebral stimulants: Esters of 2-dimethylaminoethanol with some lipophilic carboxylic acids
1990, Vol. 55, Issue 5, pp. 1278–1289 [Abstract] - Jiří Jílek, Karel Šindelář, Jaroslava Grimová, Eva Maturová, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Jan Metyš, Marta Hrubantová and Miroslav Protiva
Potential antidepressant and anti-inflammatory agents: 4-(2-Propylthio)acetophenone oximes and 4-(2-propylthio)phenylalkanoic acids
1990, Vol. 55, Issue 5, pp. 1266–1277 [Abstract] - Vladimír Pouzar, Hana Chodounská, Dalibor Sameš, Pavel Drašar and Miroslav Havel
Derivatives of 5α-androstan-3α- and 3β-ol with acrylate side chain
1990, Vol. 55, Issue 5, pp. 1243–1256 [Abstract] - Jiří Urban, Zdeněk Šedivý, Jiří Holubek, Emil Svátek, Miroslav Ryska, Ivan Koruna, Antonín Dlabač, Martin Valchář, Jiřina Metyšová, Zdeněk Polívka, Karel Šindelář, Josef Pomykáček, Marta Hrubantová and Miroslav Protiva
Potential antidepressants: 1-(2-(Methoxy- and hydroxyphenylthio)phenyl)-2-propylamines
1990, Vol. 55, Issue 4, pp. 1077–1098 [Abstract] - Miloš Beran, Antonín Černý, Miroslav Kuchař, Hana Adamírová, Jiří Holubek, Jan Taimr, Jaroslav Vachek, Maria Frühaufová, Karel Řežábek, Martin Valchář and Ivan Krejčí
9,10-Dihydroergopeptines modified in position 6
1990, Vol. 55, Issue 3, pp. 819–832 [Abstract] - Vladimír Valenta, Marie Vlková, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
Potential neuroleptics of the orthopramide series; Synthesis of N-(3-(tert.amino)propyl)-5-sulfamoyl-2-methoxybenzamides
1990, Vol. 55, Issue 3, pp. 797–808 [Abstract] - Karel Šindelář, Jiří Holubek, Emil Svátek, Jiří Schlanger, Antonín Dlabač, Martin Valchář, Marta Hrubantová and Miroslav Protiva
Open-ring models of hetero-cannabinoids: Synthesis of 2-(alkylthio)-5-(2-aminoethyl)hydroquinone derivatives
1990, Vol. 55, Issue 3, pp. 782–796 [Abstract] - Vladimír Pouzar, Dalibor Sameš and Miroslav Havel
Preparation of selectively protected derivatives of 21-nor-5-pregnene-3β,20-diol
1990, Vol. 55, Issue 2, pp. 499–511 [Abstract] - Miroslav Kuchař, Jaroslava Grimová, Václav Rejholec, Hana Tomková, Magda Jelínková and Jiří Holubek
Use of QSAR in design of antiinflammatory fluorinated arylalkanoic acids
1990, Vol. 55, Issue 1, pp. 296–306 [Abstract] - Karel Šindelář, Vladimír Valenta, Jiří Holubek, Oluše Matoušová and Miroslav Protiva
Potential antidepressants. Synthesis of 6,11-dihydrodibenzo[b,e]thiepin-11-yl (dimethylaminomethyl)phenyl ethers, sulfides, amines and some related compounds
1990, Vol. 55, Issue 1, pp. 282–295 [Abstract] - Pavel Drašar, Vladimír Pouzar, Ivan Černý, George R. Pettit and Miroslav Havel
Synthesis and in vitro antimetabolic evaluation of some steroidal thiazoles
1989, Vol. 54, Issue 12, pp. 3339–3347 [Abstract] - Jiří Jílek, Karel Šindelář, Josef Pomykáček, Vojtěch Kmoníček, Zdeněk Šedivý, Marta Hrubantová, Jiří Holubek, Emil Svátek, Miroslav Ryska, Ivan Koruna, Martin Valchář, Antonín Dlabač, Jiřina Metyšová, Nataša Dlohožková and Miroslav Protiva
Potential antidepressants: 2-(Methoxy- and hydroxyphenylthio)benzylamines as selective inhibitors of 5-hydroxytryptamine re-uptake in the brain
1989, Vol. 54, Issue 12, pp. 3294–3338 [Abstract] - Zdeněk Polívka, Miloš Buděšínský, Jiří Holubek, Bohdan Schneider, Zdeněk Šedivý, Emil Svátek, Oluše Matoušová, Jan Metyš, Martin Valchář, Radomír Souček and Miroslav Protiva
4H-Benzo[4,5]cyclohepta[1,2-b]thiophenes and 9,10-dihydro derivatives - Sulfonium analogues of pizotifen and ketotifen; Chirality of ketotifen; Synthesis of the 2-bromo derivative of ketotifen
1989, Vol. 54, Issue 9, pp. 2443–2469 [Abstract] - Jiří Jílek, Jiří Urban, Vojtěch Kmoníček, Josef Pomykáček, Jiří Holubek, Emil Svátek, Oluše Matoušová, Jan Metyš, Martin Valchář, Stanislav Wildt and Miroslav Protiva
Potential anticonvulsants: 3-Chlorobenzophenone derivatives
1989, Vol. 54, Issue 8, pp. 2248–2260 [Abstract] - Jiří Jílek, Jiří Urban, Petr Taufmann, Jiří Holubek, Antonín Dlabač, Martin Valchář and Miroslav Protiva
Potential antidepressants: 2-(Phenylthio)aralkylamines
1989, Vol. 54, Issue 7, pp. 1995–2008 [Abstract] - Vladimír Valenta, Marie Vlková, Jiří Holubek, Jiřina Metyšová and Miroslav Protiva
Potential antidepressants: 10-Amino-2-chloro-10,11-dihydrodibenzo[b,f]thiepins
1989, Vol. 54, Issue 7, pp. 1979–1994 [Abstract] - Irena Červená, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
Potential antidepressants: 2-(Aminoalkoxy)biphenyls and some related ω-substituted 2-alkoxybiphenyls
1989, Vol. 54, Issue 7, pp. 1966–1978 [Abstract] - Irena Červená, Jiří Holubek, Emil Svátek, Miroslav Ryska and Miroslav Protiva
Potential antidepressants: 6-(Aminoalkoxy)dibenzo[b,f]thiepin-10(11H)-ones and 6-(aminoalkoxy)-10,11-dihydrodibenzo[b,f]thiepin-10-ols
1989, Vol. 54, Issue 7, pp. 1955–1965 [Abstract] - Vladimír Pouzar, Lenka Schneiderová, Pavel Drašar, Oldřich Štrouf and Miroslav Havel
Synthesis of 2-propynyl ethers of steroid alcohols
1989, Vol. 54, Issue 7, pp. 1888–1902 [Abstract] - Martin Mandel, Ludvík Novák, Miroslav Rajšner, Jiří Holubek and Vladislava Holá
New synthesis of oxime-type beta-lactam antibiotics
1989, Vol. 54, Issue 6, pp. 1734–1745 [Abstract] - Vojtěch Kmoníček, Zdeněk Vejdělek, Jiří Holubek, Martin Valchář and Miroslav Protiva
Potential antidepressants: 1-(4-Aminoalkoxy)phenyl)-2-propylamines
1989, Vol. 54, Issue 6, pp. 1721–1733 [Abstract] - Hana Hulinská, Miroslav Ryska, Ivan Koruna, Jiří Holubek, Jan Taimr, Emil Svátek and Miroslav Protiva
Some further 2-(4-substituted 1-piperazinyl)acetamides derived from 6,11-dihydrodibenzo[b,e]thiepin. Transformations of 6,11-dihydrodibenzo[b,e]thiepin derivatives into anthraquinones, anthrones and anthracenes
1989, Vol. 54, Issue 5, pp. 1388–1402 [Abstract] - Hana Hulinská, Miloš Buděšínský, Jiří Holubek, Oluše Matoušová, Hana Frycová and Miroslav Protiva
Reactions of N-substituted 2-aminopyridines with chloroacetyl chloride; Formation of a new series of heterocyclic betaines: 1-Substituted 4-chloromethyl-2-oxopyrido[1,2-a]pyrimidin-5-ium-3-olates
1989, Vol. 54, Issue 5, pp. 1376–1387 [Abstract] - Zdeněk Polívka, Vladimír Valenta, Karel Šindelář, Jiří Holubek, Miloš Buděšínský, Miroslav Ryska, Ivan Koruna, Jitka Kohoutová, Jan Metyš, Jiřina Metyšová, Martin Valchář and Miroslav Protiva
Potential antidepressants: Saturated side chain amines derived from 6,11-dihydrodibenzo[b,e]thiepin and 4,9-dihydrothieno[2,3-c]-2-benzothiepin
1989, Vol. 54, Issue 1, pp. 235–247 [Abstract] - Irena Červená, Jiří Holubek, Emil Svátek, Jan Metyš, Martin Valchář and Miroslav Protiva
Potential antidepressants: Synthesis of two 4-(aminoalkoxy)dibenzo[b,e]thiepin-11(6H)-ones
1989, Vol. 54, Issue 1, pp. 225–228 [Abstract] - Jiří Jílek, Martin Valchář, Jiří Holubek, Nataša Dlohožková, Josef Pomykáček, Oluše Matoušová, Jiřina Metyšová and Miroslav Protiva
Noncataleptic neuroleptic agents: 2-(4-(2-(2-Chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yloxy)ethyl)piperazine-1-yl)ethanol and some related compounds
1988, Vol. 53, Issue 11, pp. 2731–2741 [Abstract] - Zdena Koblicová, Jiří Holubek and Jan Trojánek
Synthesis of stereoisomeric vincamines
1988, Vol. 53, Issue 11, pp. 2722–2730 [Abstract] - Miroslav Kuchař, Eva Maturová, Bohumila Brunová, Jaroslava Grimová, Hana Tomková and Jiří Holubek
Quantitative relations between structure and antiinflammatory activity of aryloxoalkanoic acids
1988, Vol. 53, Issue 8, pp. 1862–1872 [Abstract] - Hana Hulinská, Zdeněk Polívka, Jiří Jílek, Karel Šindelář, Jiří Holubek, Emil Svátek, Oluše Matoušová, Miloš Buděšínský, Hana Frycová and Miroslav Protiva
Experimental antiulcer agents: N-substituted 2-(4-methyl-1-piperazinyl)acetamides as pirenzepine models and some related compounds
1988, Vol. 53, Issue 8, pp. 1820–1844 [Abstract] - Irena Červená, Jiří Holubek, Emil Svátek and Miroslav Protiva
Potential antidepressants: 4-(Aminoalkoxy)thioxanthones
1988, Vol. 53, Issue 6, pp. 1307–1316 [Abstract] - Jiří Jílek, Jiří Holubek, Emil Svátek, Jan Metyš, Hana Frycová, Josef Pomykáček and Miroslav Protiva
Tricyclic analogues of the antiallergic agent oxatomide: 1-(3-(4-(10,11-Dihydro-5H-dibenzo[a,d]cycloheptene-5-yl)-1-piperazinyl)propyl)-1,3-dihydro-2H-benzimidazol-2-one and the related 6,11-dihydrodibenzo[b,e]thiepin, 4,9-dihydrothieno[2,3-c]-2-benzothiepin, and 10,11-dihydrodibenzo[b,f]thiepin derivatives
1988, Vol. 53, Issue 4, pp. 870–883 [Abstract] - Vladimír Valenta, Hana Hulinská, Jiří Holubek, Antonín Dlabač, Jan Metyš, Hana Frycová and Miroslav Protiva
N-substituted derivatives of 6,11-dihydrodibenzo[b,e]thiepin-11-amine and related compounds; Synthesis and pharmacological screening
1988, Vol. 53, Issue 4, pp. 860–869 [Abstract] - Zdeněk Vejdělek, Jiří Holubek, Miloš Buděšínský, Miroslav Ryska, Emil Svátek and Miroslav Protiva
Reactions of 4-chloro-1-nitrobenzene with (3-chloro-4-methoxyphenyl)acetonitrile and (3,4-dimethoxyphenyl)acetonitrile; Synthesis of 8-chloro-1-methyl (and methylthiomethyl-6-(3,4-disubstituted phenyl)-4H-s-triazolo[4,3-a]-1,4-benzodiazepines
1988, Vol. 53, Issue 2, pp. 361–372 [Abstract] - Karel Šindelář, Jiří Holubek, Oluše Matoušová, Emil Svátek, Martin Valchář, Antonín Dlabač, Nataša Dlohožková, Marta Hrubantová and Miroslav Protiva
Aminoalkylidene and aminoalkyl derivatives of 6,11-dihydrodibenzo[b,e]thiepin-2- and -9-carbonitrile and 4,10-dihydrothieno[2,3-c]-1-benzothiepin-6-carbonitrile; Antidepressants with a new activity profile
1988, Vol. 53, Issue 2, pp. 340–360 [Abstract] - Zdeněk Vejdělek, Jan Metyš, Jiří Holubek, Miloš Buděšínský, Emil Svátek, Oluše Matoušová and Miroslav Protiva
Potentional anxiolytics and hypnotics: 1-(Alkanesulfonamidoalkyl)-6-aryl-8-halogeno-s-triazolo[4,3-a]-1,4-benzodiazepines and related compounds
1988, Vol. 53, Issue 1, pp. 132–144 [Abstract] - Vladimír Valenta, Jiří Holubek, Emil Svátek and Miroslav Protiva
Synthesis of 4-methoxyphenoxyacetic and 3,4,5-trimethoxyphenoxyacetic acid amides and hydrazides as potential neurotropic and cardiovascular agents
1987, Vol. 52, Issue 12, pp. 3013–3023 [Abstract] - Antonín Černý, Jiří Křepelka, Karel Řežábek, Maria Frühaufová, Václav Plaisner and Jiří Holda
Some dopaminergically active esters of N-[(5R,8S,10R)-6-propyl-8-ergolinyl]carbamic acid with cancerogenicity manifestations
1987, Vol. 52, Issue 12, pp. 2983–2990 [Abstract] - Zdeněk Polívka, Jiří Holubek, Miloš Buděšínský, Oluše Matoušová, Emil Svátek, Jan Metyš and Miroslav Protiva
Potential antihistamine agents: 4-(6,11-Dihydrodibenzo[b,e]thiepin-11-ylidene)-1-methyltetrahydrothiopyranium iodide and similar sulfonium salts derived from related tricyclic systems
1987, Vol. 52, Issue 11, pp. 2758–2774 [Abstract] - Vladimír Pouzar, Lenka Kárászová and Miroslav Havel
Preparation of 21-methoxycarbonyl-21-methylene-5-pregnen-3β-ol derivatives
1987, Vol. 52, Issue 11, pp. 2735–2743 [Abstract] - Irena Červená, Jiří Holubek, Emil Svátek, Martin Valchář and Miroslav Protiva
Potential antidepressants: 3-Methyl-6-dimethylamino-1,2-diphenylhexan-3-ol and related compounds
1987, Vol. 52, Issue 10, pp. 2564–2571 [Abstract] - Zdeněk Vejdělek, Jiří Holubek, Miroslav Ryska, Ivan Koruna, Emil Svátek, Miloš Buděšínský and Miroslav Protiva
Reactions of 4-chloro-1-nitrobenzene with o-substituted phenylacetonitriles; Synthesis of 8-chloro-1-methyl(and methylthiomethyl)-6-(2-substituted phenyl)-4H-s-triazolo[4,3-a]-1,4-benzodiazepines
1987, Vol. 52, Issue 10, pp. 2545–2563 [Abstract] - Vladimír Valenta, Jiří Holubek, Emil Svátek, Vladimír Miller, Marie Vlková and Miroslav Protiva
2-Diethylaminoethyl esters of 1,3-disubstituted propane-2-carboxylic acids
1987, Vol. 52, Issue 10, pp. 2534–2544 [Abstract] - Ivan Černý, Vladimír Pouzar, Pavel Drašar and Miroslav Havel
β-Glucosides of steroidal unsaturated nitriles
1987, Vol. 52, Issue 10, pp. 2521–2533 [Abstract] - Karel Šindelář, Miloš Buděšínský, Tomáš Vaněk, Jiří Holubek, Emil Svátek, Oluše Matoušová, Charles Wayne Rees and Miroslav Protiva
Reaction of 6,11-dihydrodibenzo[b,e]thiepin-11-carbonitrile with 1,2-dibromoethane, a reinvestigation. Formation of 11,12-dihydro-6H-6,12-methanodibenzo[b,f]thiocin-12-carbonitrile
1987, Vol. 52, Issue 9, pp. 2281–2294 [Abstract] - Miroslav Protiva, Jiří Jílek, Miroslav Rajšner, Karel Šindelář, Václav Bártl, Miroslav Ryska, Ivan Koruna, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Antonín Dlabač, Josef Pomykáček and František Mikšík
Fluorinated tricyclic neuroleptics with prolonged action: derivatives and analogues of 2-(4-(7-fluoro-2-isopropyl-10,11-dihydrodibenzo[b,f]thiepin-11-yl)-piperazine-1-yl)ethanol
1987, Vol. 52, Issue 7, pp. 1811–1833 [Abstract] - Vladimír Pouzar, Ivan Černý, Pavel Drašar and Miroslav Havel
Preparation of (20E)-21-methoxycarbonyl-5,14,20-pregnatrien-3β-ol derivatives
1987, Vol. 52, Issue 7, pp. 1803–1810 [Abstract] - Zdeněk Polívka, Irena Lichá, Petr Taufmann, Emil Svátek, Jiří Holubek and Miroslav Protiva
Synthesis of 3-(6,11-dihydrodibenzo[b,e]thiepin-11-ylidene)propanoic acid and related compounds
1987, Vol. 52, Issue 6, pp. 1566–1582 [Abstract] - Vladimír Valenta, Jiří Holubek and Miroslav Protiva
4-Substituted 1-(1-(2-(arylthio)-5-halogenophenyl)ethyl)piperazines; Synthesis and biological screening
1987, Vol. 52, Issue 4, pp. 1062–1072 [Abstract] - Vladimír Pouzar, Ivan Černý, Pavel Drašar, Soňa Vašíčková and Miroslav Havel
Preparation of 3β-hydroxy-21,26,27-trinorcholesta-5,23-dien-25→22-olide and 3β-hydroxy-20-(2-furyl)-21-nor-5-pregnene derivatives
1987, Vol. 52, Issue 4, pp. 1043–1051 [Abstract] - Vojtěch Kmoníček, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
2-(tert.amino)-11-(4-methylpiperazino)dibenzo[b,f]thiepins and their 10,11-dihydro derivatives; Synthesis and neuroleptic activity
1987, Vol. 52, Issue 3, pp. 793–803 [Abstract] - Vladimír Pouzar, Ivan Černý, Pavel Drašar and Miroslav Havel
New approach to steroidal hemisuccinates and glycosides
1987, Vol. 52, Issue 3, pp. 775–787 [Abstract] - Zdeněk Veselý, Jiří Holubek and Jan Trojánek
Reactions in the series of substituted isoindolo[1,2-b][3]-benzazepin-5-ones
1987, Vol. 52, Issue 1, pp. 233–241 [Abstract] - Martin Černý, Evžen Kasafírek, Jozef Rovenský and Jiří Křepelka
Synthesis of blood serum thymic factor and its analogs
1986, Vol. 51, Issue 12, pp. 2909–2918 [Abstract] - Miroslav Kuchař, Bohumila Brunová, Jaroslava Grimová, Stanislav Vaněček and Jiří Holubek
Synthesis of cyclohexylaliphatic acids and their pharmacological properties
1986, Vol. 51, Issue 12, pp. 2896–2908 [Abstract] - Karel Šindelář, Jiří Holubek, Miroslav Ryska, Ivan Koruna and Miroslav Protiva
5-Substituted and 5,7-disubstituted 5,7-dihydrodibenzo[c,e]thiepins and the corresponding S-oxygenated compounds: Alkylamines, carboxylic acids, and carboxamides; synthesis and pharmacological screening
1986, Vol. 51, Issue 12, pp. 2848–2868 [Abstract] - Miroslav Protiva, Jiří Jílek, Irena Červená, Josef Pomykáček, Václav Bártl, Antonín Dlabač, Martin Valchář, Jiřina Metyšová, Jiří Holubek and Emil Svátek
Noncataleptic neuroleptic agents: 4-Substituted 1-(2-chloro-7-fluoro-10,11-dihydrodibenzo[b,f]thiepin-10-yl)piperazines and related compounds
1986, Vol. 51, Issue 11, pp. 2598–2616 [Abstract] - Vladimír Pouzar, Ivan Černý, Pavel Drašar and Miroslav Havel
New method of preparation of cardioglycoside hemisuccinates
1986, Vol. 51, Issue 9, pp. 2019–2028 [Abstract] - Jiří Křepelka, Antonín Černý, Rudolf Kotva, Jaroslav Vachek and Milan Mělka
Some derivatives of 5-(2-amino-6-hydroxy-4-oxo-3,4-dihydro-5-pyrimidinyl)pentanoic acid
1986, Vol. 51, Issue 5, pp. 1140–1149 [Abstract] - Vojtěch Kmoníček, Emil Svátek, Jiří Holubek and Miroslav Protiva
Synthesis of potential neuroleptics and tranquillizers: 2-(tert.Amino)-9-(3-dimethylaminopropylidene)thioxanthenes
1986, Vol. 51, Issue 4, pp. 937–947 [Abstract] - Miroslav Protiva, Jiří Jílek, Miroslav Rajšner, Josef Pomykáček, Miroslav Ryska, Jiří Holubek, Emil Svátek and Jiřina Metyšová
Fluorinated tricyclic neuroleptics with prolonged action: 7-Fluoro-11-[4-(2-hydroxyethyl)piperazino]-2-isopropyl-10,11-dihydrodibenzo[b,f]thiepin
1986, Vol. 51, Issue 3, pp. 698–722 [Abstract] - Michal P. Nemeryuk, Andrej L. Sedov, Tamara S. Safonova, Antonín Černý and Jiří Křepelka
Transformations of substituted 5-aminopyrimidines under conditions of the diazotization
1986, Vol. 51, Issue 1, pp. 215–233 [Abstract] - Irena Červená, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Martin Valchář, Antonín Dlabač, Stanislav Wildt and Miroslav Protiva
6-Substituted and 2-chloro-6-substituted 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins as potential antidepressants; Synthesis and pharmacology
1986, Vol. 51, Issue 1, pp. 141–155 [Abstract] - Ivan Černý, Vladimír Pouzar, Pavel Drašar, František Tureček and Miroslav Havel
Steroids with the β-crotonate (2-butenoate) side chain
1986, Vol. 51, Issue 1, pp. 128–140 [Abstract] - Soňa Vašíčková, Vladimír Pouzar, Ivan Černý, Pavel Drašar and Miroslav Havel
Infrared spectra of compounds with the methoxymethyl protecting group
1986, Vol. 51, Issue 1, pp. 90–100 [Abstract] - Pavel Drašar, Vladimír Pouzar, Ivan Černý, Miroslav Havel, František Tureček, Daniela Schmiedová and Karel Vereš
Preparation of 3-carboxypropanoates of digitoxin and digoxin and their conjugates with L-tyrosine
1985, Vol. 50, Issue 12, pp. 2760–2774 [Abstract] - Jiří Jílek, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Josef Pomykáček, Zdeněk Šedivý and Miroslav Protiva
Potential metabolites of the neuroleptic agents belonging to the 8-methylthio-10-piperazino-10,11-dihydrodibenzo[b,f]thiepin series; Synthesis of 2-hydroxy and 3-hydroxy derivatives
1985, Vol. 50, Issue 10, pp. 2179–2190 [Abstract] - Miroslav Protiva, Zdeněk Šedivý, Jiří Holubek, Emil Svátek and Jiří Němec
Cyclic amidines derived from benz[c,d]indole and 4,5-dihydro-3H-1-benzazepine including some related compounds: Synthesis and pharmacological screening
1985, Vol. 50, Issue 8, pp. 1888–1898 [Abstract] - Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Martin Valchář and Miroslav Protiva
Butaclamol-like neuroleptic agents: Synthesis of 1-(11H-dibenz[b,f]-1,4-oxathiepin-11-yl)methyl-4-isobutylpiperidin-4-ol and of some related compounds
1985, Vol. 50, Issue 7, pp. 1484–1497 [Abstract] - Zdeněk Polívka, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
Synthesis of the semi-rigid analogues of prothiadene and dithiadene as potential antidepressant and antihistamine agents: 11-[2-(Dimethylaminomethyl)cyclohexylidene]-6,11-dihydrodibenzo[b,e]thiepins and 4-[2-(dimethylaminomethyl)cyclohexylidene]-4,9-dihydrothieno-[2,3-c]-2-benzothiepins
1985, Vol. 50, Issue 5, pp. 1078–1088 [Abstract] - Jan Šmidrkal, Jiří Holubek and Jan Trojánek
The synthesis of 2,3,7,8-bismethylenedioxy-11-methoxy-5-methylbenzo[c]phenanthridinium chloride
1985, Vol. 50, Issue 4, pp. 984–990 [Abstract] - Vladimír Pouzar, Pavel Drašar, Ivan Černý and Miroslav Havel
Preparation and absolute configuration at C(22) of 21,26,27-trinor-5α-cholestan-25→22-olide derivatives
1985, Vol. 50, Issue 4, pp. 869–877 [Abstract] - Jan Šmidrkal, Jiří Holubek, Jiří Šlanger and Jan Trojánek
Attempts at the synthesis of 11-methoxysubstituted benzo[c]phenantridines
1985, Vol. 50, Issue 4, pp. 861–868 [Abstract] - Jiří Jílek, Jiří Holubek, Emil Svátek, Jiří Schlanger, Josef Pomykáček and Miroslav Protiva
Highly polar potential metabolites of the neuroleptic agent oxyprothepin: Synthesis of 2-hydroxy-8-methylsulfonyl and 3-hydroxy-8-methylsulfonyl derivatives of 10-[4-(3-hydroxypropyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
1985, Vol. 50, Issue 2, pp. 519–537 [Abstract] - Karel Šindelář, Jiří Holubek, Jiří Schlanger, Antonín Dlabač, Martin Valchář and Miroslav Protiva
Synthesis of spiro(piperidine-4,6'-dibenz[b,e]-1,4-oxathiepin) and its 1-methyl derivative as potential antidepressant agents
1985, Vol. 50, Issue 2, pp. 503–509 [Abstract] - Antonín Černý, Jiří Křepelka, Viktor Zikán, Drahuše Vlčková, Jaroslav Vachek, Jiří Holubek, Karel Řežábek, Maria Frühaufová, Miroslav Šeda, Jana Chlebounová and Otakar Marhan
Some 6-substituted 1-[(5R,8S,10R)-8-ergolinyl]-3,3-diethylureas
1984, Vol. 49, Issue 12, pp. 2828–2836 [Abstract] - Zdeněk Vejdělek, Jan Metyš, Jiří Holubek, Emil Svátek and Miroslav Protiva
Potential antiparkinsonic agents: Synthesis and pharmacology of some 4-fluoro-4'-halogen'benzhydryl 2-(N,N-disubstituted amino)ethyl ethers
1984, Vol. 49, Issue 11, pp. 2649–2660 [Abstract] - Karel Šindelář, Jiří Holubek, Miroslav Ryska, Antonín Dlabač, Martin Valchář, Jiřina Metyšová and Miroslav Protiva
Tricyclic compounds containing two chalcogen atoms in the central seven-membered rings as potential drugs: Synthesis of 3-chloro-6-(1-methyl-4-piperidyl)-6H-dibenz[b,e]-1,4-oxathiepin and 6-oxodibenz[b,e]-1,4-oxathiepin-2-acetic acid
1984, Vol. 49, Issue 11, pp. 2531–2540 [Abstract] - Václav Bártl, Karel Šindelář, Vladimír Valenta, Jiří Holubek, Emil Svátek, Jiří Schlanger, Antonín Dlabač, Jiřina Metyšová and Miroslav Protiva
Potential antipsychotic agents: 2-Chloro- and 2-methyl-11-(2-piperazinoethoxy)-6,11-dihydrodibenzo[b,e]thiepins and some related compounds; Synthesis and pharmacology
1984, Vol. 49, Issue 11, pp. 2520–2530 [Abstract] - Pavel Drašar, Vladimír Pouzar, Ivan Černý and Miroslav Havel
Synthesis of 4-(21-nor-5-pregnen-20-yl)-1,3-thiazole derivatives
1984, Vol. 49, Issue 4, pp. 1051–1059 [Abstract] - Pavel Drašar, Vladimír Pouzar, Ivan Černý, Jorga Smolíková and Miroslav Havel
Synthesis of 17β-[4-(1,3-thiazolyl)]androstane 3β-hemisuccinate and glycoside
1984, Vol. 49, Issue 4, pp. 1039–1050 [Abstract] - Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Antonín Dlabač, Martin Valchář and Miroslav Protiva
Analogues of the neuroleptic agent isobutaclamol: Stereoisomeric 3b,4,5,6,7,9,9a,10-octahydro-[1]benzothiepino[2,3,4-ed]pyrido[2,1-a]isoquinolin-5-ols and some related compounds
1984, Vol. 49, Issue 4, pp. 1021–1038 [Abstract] - Ivan Černý, Vladimír Pouzar, Pavel Drašar, Miloš Buděšínský and Miroslav Havel
Glucosylation of 5-androsten-3β-ol derivatives containing butenolide, furan or unsaturated ester moieties in the side chain
1984, Vol. 49, Issue 4, pp. 881–891 [Abstract] - Vladimír Pouzar, Pavel Drašar, Ivan Černý and Miroslav Havel
Preparation of 21,26,27-trinor-5α-cholest-23-en-25→20-olide from a propargyl synthone
1984, Vol. 49, Issue 4, pp. 871–880 [Abstract] - Zdeněk Polívka, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
Potential hypnotics and anxiolytics: Synthesis of 2-bromo-4-(2-chlorophenyl)-9-[4-(2-methoxyethyl)piperazino]-6H-thieno[3,2,4-triazolo[4,3-a]-1,4-diazepine and of some related compounds
1984, Vol. 49, Issue 3, pp. 621–636 [Abstract] - Jiří Jílek, Josef Pomykáček, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiří Protiva and Miroslav Protiva
Reactions of 4,4'-disubstituted diphenyl sulfides with chloroacetyl chloride and aluminium chloride
1984, Vol. 49, Issue 3, pp. 603–620 [Abstract] - Pavel Drašar, Ivan Černý, Vladimír Pouzar and Miroslav Havel
New preparation of steroidal 3-hemisuccinates
1984, Vol. 49, Issue 1, pp. 306–312 [Abstract] - Miroslav Kuchař, Bohumila Brunová, Václav Rejholc, Magda Jelínková, Jiří Holubek and Oldřich Němeček
Quantitative relations between structure and activation of fibrinolysis in selected series of arylaliphatic acids
1984, Vol. 49, Issue 1, pp. 122–136 [Abstract] - Jiří Křepelka, Drahuše Vlčková and Milan Mělka
Some 1-substitution derivatives of 4-aryl-2,3-dihalogeno-1-naphthols
1984, Vol. 49, Issue 1, pp. 110–121 [Abstract] - Zdeněk Polívka, Jiří Jílek, Jiří Holubek, Emil Svátek, Antonín Dlabač, Martin Valchář and Miroslav Protiva
Noncataleptic neuroleptic agents: 2-Halogeno-8-isopropyl-10-piperazino-10,11-dihydrodibenzo[b,f,]thiepins
1984, Vol. 49, Issue 1, pp. 86–109 [Abstract] - Zdeněk Polívka, Jiří Holubek, Jan Metyš, Zdeněk Šedivý and Miroslav Protiva
Potential hypnotics and anxiolytics: 8-Chloro-6-(2-chlorophenyl)-1-[4-(2-methoxyethyl)piperazino]-methyl-4H-s-triazolo[4,3-a]-1,4-benzodiazepine and related compounds
1983, Vol. 48, Issue 12, pp. 3433–3443 [Abstract] - Vladimír Pouzar, Soňa Vašíčková, Pavel Drašar, Ivan Černý and Miroslav Havel
Preparation and absolute configuration at C(22) of 21,26,27-trinor-5α-cholestane-22,25-diol derivatives
1983, Vol. 48, Issue 8, pp. 2423–2435 [Abstract] - Zdeněk Polívka, Miroslav Ryska, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
Potential hypnotics and anxiolytics in the 4H-s-triazolo[4,3-a]-1,4-benzodiazepine series: 8-Chloro-6-(2-chlorophenyl)-1-[4-(2-methoxyethyl)piperazino]-4H-s-triazolo[4,3-a]-1,4-benzodiazepine and some related compounds
1983, Vol. 48, Issue 8, pp. 2395–2410 [Abstract] - Ivan Černý, Vladimír Pouzar, Pavel Drašar and Miroslav Havel
Synthesis of 17β-steroidal 4-(2-butenolides)
1983, Vol. 48, Issue 7, pp. 2064–2071 [Abstract] - Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Jiří Urban and Miroslav Protiva
11-(Dimethylaminoalkyl)-6,11-dihydrodibenzo[b,e]thiepin-11-carbonitriles and some related compounds
1983, Vol. 48, Issue 7, pp. 1898–1909 [Abstract] - Antonín Černý, Viktor Zikán, Drahuše Vlčková, Jan Beneš, Jiří Holubek, Karel Řežábek, Marie Aušková and Jiří Křepelka
(5R,8S,10R)-6-Alkyl-8-ergolinecarboxylic acids and some of their derivatives
1983, Vol. 48, Issue 5, pp. 1483–1488 [Abstract] - Zdeněk Polívka, Jiří Holubek, Emil Svátek, Antonín Dlabač, Dušan Půček, Zdeněk Šedivý and Miroslav Protiva
3-(4-Methylpiperazino)dibenzo[b,f]-1,2,4-triazolo[4,3-d]-1,4-thiazepine and its 6-chloro and 12-chloro derivatives; Synthesis and pharmacology
1983, Vol. 48, Issue 5, pp. 1465–1476 [Abstract] - Vladimír Valenta, Jiří Holubek, Emil Svátek, Antonín Dlabač, Marie Bartošová and Miroslav Protiva
α-(4-Tolyl)dopamine, derivatives and analogues; Synthesis and pharmacological screening
1983, Vol. 48, Issue 5, pp. 1447–1464 [Abstract] - Pavel Drašar, Vladimír Pouzar, Ivan Černý and Miroslav Havel
Alternative syntheses of steroidal maleimides
1983, Vol. 48, Issue 4, pp. 1224–1232 [Abstract] - Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Jiří Urban, Jaroslava Grimová, Irena Červená, Marta Hrubantová and Miroslav Protiva
Dibenzo[b,f]thiepin-10-carbonitrile, its 10,11-dihydro derivative, some transformation products and related compounds
1983, Vol. 48, Issue 4, pp. 1187–1211 [Abstract] - Václav Bártl, Jiří Holubek, Emil Svátek, Marie Bartošová and Miroslav Protiva
Potential anticonvulsants: Substituted N-benzylidene derivatives of 10-(4-aminopiperazino)-10,11-dihydrodibenzo[b,f]thiepins
1983, Vol. 48, Issue 4, pp. 1173–1186 [Abstract] - Jiří Jílek, Josef Pomykáček, Zdeněk Prošek, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Antonín Dlabač and Miroslav Protiva
8-Chloro and 8-methylthio derivatives of 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins; New compounds and new procedures
1983, Vol. 48, Issue 3, pp. 906–927 [Abstract] - Zdeněk Polívka, Miroslav Rajšner, Jan Metyš, Jiří Holubek, Emil Svátek, Miroslav Ryska and Miroslav Protiva
Antiaminic agents derived from thieno[2,3-c]-2-benzothiepin: 4-(1-Methyl-4-piperidylidene)-4,9-dihydrothieno[2,3-c]-2-benzothiepin and some related compounds
1983, Vol. 48, Issue 2, pp. 623–641 [Abstract] - Jiří Křepelka, Drahuše Vlčková, Jiří Holubek and Jiří Roubík
8-Substitution derivatives of D-6-methylergoline-I
1983, Vol. 48, Issue 1, pp. 312–318 [Abstract] - Jiří Křepelka, Jan Beneš, Vladimír Pouzar, Jaroslav Vachek and Jiří Holubek
Some 2-substitution derivatives of 5-(4-oxo-6-hydroxy-3,4-dihydro-5-pyrimidinyl)pentanoic acid
1983, Vol. 48, Issue 1, pp. 304–311 [Abstract] - Rudolf Kotva, Jaroslav Vachek and Jiří Křepelka
Some derivatives of 4-[(2-amino-6-hydroxy-4-oxo-3,4-dihydro-5-pyrimidinyl)methyl] benzoic acid
1983, Vol. 48, Issue 1, pp. 299–303 [Abstract] - Miloš Beran, Antonín Černý, Jiří Křepelka and Jaroslav Vachek
Substituted ω-(4-oxo-3,4-dihydro-5-pyrimidinyl) alkanoic acids, their derivatives and analogues
1983, Vol. 48, Issue 1, pp. 292–298 [Abstract] - Miroslav Rajšner, Jan Metyš, Jiří Holubek and Miroslav Protiva
Potential antidepressants: Some N-substituted derivatives of (E)-11-(3-methylaminopropylidene)-6,11-dihydrodibenzo[b,e]thiepin
1983, Vol. 48, Issue 1, pp. 163–172 [Abstract] - Karel Šindelář, Jiřina Metyšová, Jiří Holubek, Emil Svátek, Miroslav Ryska and Miroslav Protiva
Fluorinated tricyclic neuroleptics with prolonged action: 3-Fluoro-10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepins with less common substituents in position 8
1983, Vol. 48, Issue 1, pp. 144–155 [Abstract] - Rudolf Kotva, Jiří Křepelka and Miroslav Semonský
5,5-Disubstituted barbituric acids and their analogues
1983, Vol. 48, Issue 1, pp. 137–143 [Abstract] - Miloš Beran, Jan Beneš and Jiří Křepelka
Derivatives of 3-(D-6-methyl-8β-ergolin-I-yl)propanoic acid
1982, Vol. 47, Issue 12, pp. 3432–3436 [Abstract] - Zdeněk Vejdělek, Jiří Holubek, Marie Bartošová and Miroslav Protiva
4-(Aminoacylamido)-s-hydrindacenes and related compounds: Synthesis and pharmacological screening
1982, Vol. 47, Issue 12, pp. 3297–3305 [Abstract] - Miroslav Protiva, Zdeněk Šedivý, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Marie Bartošová
Potential psychotropic and antihistamine agents: 1- and 3-alkyl-9-(3-dimethylaminopropylidene)-thioxanthenes and 3-alkyl-11-piperazino-10,11-dihydrodibenzo[b,f]thiepins
1982, Vol. 47, Issue 11, pp. 3134–3147 [Abstract] - Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Antonín Dlabač, Jiřina Metyšová and Miroslav Protiva
Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: 2-Fluoro-8-substituted 6-(4-piperidyl)-6H-dibenz[b,e]-1,4-oxathiepins
1982, Vol. 47, Issue 11, pp. 3114–3133 [Abstract] - Miroslav Protiva, Karel Šindelář, Vladimír Valenta, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiří Schlanger, Jiří Urban and Marta Hrubantová
Reactions of 11-chloro-11-phenyl-6,11-dihydrodibenzo[b,e]-thiepin with piperidine and some further nucleophiles
1982, Vol. 47, Issue 11, pp. 3094–3113 [Abstract] - Karel Šindelář, Jiřina Metyšová, Jiří Holubek, Emil Svátek, Jiří Protiva and Miroslav Protiva
Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: 8-Substituted 6-(4-piperidyl)-6H-dibenz[b,e]-1,4-oxathiepins
1982, Vol. 47, Issue 11, pp. 3077–3093 [Abstract] - Josef Hájíček, Jiří Holubek and Jan Trojánek
Synthesis of 4,4- and 5,5-disubstituted 4,5-dihydro-6H-canthin-6-ones
1982, Vol. 47, Issue 10, pp. 2749–2762 [Abstract] - Rudolf Kotva, Jiří Křepelka and Jaroslav Vachek
2-Substituted derivatives of 5-(4-oxo-3,4-dihydro-5-pyrimidinyl)pentanoic acid
1982, Vol. 47, Issue 9, pp. 2525–2529 [Abstract] - Iva Vančurová, Jiří Křepelka and František Šmejkal
Derivatives of benzo(c)fluorenes. III. Synthesis and biological action of some dibasic derivatives of 7-oxo-7H-benzo(c)fluorene
1982, Vol. 47, Issue 7, pp. 1867–1872 [Abstract] - Jiří Křepelka, Iva Vančurová, Jiří Holubek, Milan Mělka and Karel Řežábek
Derivatives of benzo(c)fluorene: II. Synthesis and biological effect of basic ethers of 7-oxo-7H-benzo(c)fluorene
1982, Vol. 47, Issue 7, pp. 1856–1866 [Abstract] - Jan Beneš and Jiří Křepelka
2-Acylated derivatives of ergoline
1982, Vol. 47, Issue 6, pp. 1757–1761 [Abstract] - Jan Beneš and Jiří Holubek
1,2-Fused derivatives of ergoline
1982, Vol. 47, Issue 6, pp. 1641–1644 [Abstract] - Jan Beneš and Jiří Holubek
Wittig type reactions of 2-formylated derivatives of 6-methylergoline - I
1982, Vol. 47, Issue 6, pp. 1636–1640 [Abstract] - Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Antonín Dlabač and Miroslav Protiva
Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: Synthesis of 6-(aminoalkyl) derivatives of 6H-dibenz[b,e]-1,4-oxathiepin
1982, Vol. 47, Issue 5, pp. 1367–1381 [Abstract] - Jiří Křepelka, Jiří Roubík, Jiří Holubek and Iva Vančurová
5-, 6- And 7-substitution derivatives of 7-oxo-7H-benzo(c)fluorene
1982, Vol. 47, Issue 4, pp. 1258–1266 [Abstract] - Jiří Křepelka, Iva Vančurová and Jiří Holubek
Reactions of 4-aryl-1-methoxynaphtalene-2,3-dicarboxylic acid anhydrides and naphtho(2,3-c)furan-1-(3H)-one derivatives with hydrazines
1982, Vol. 47, Issue 4, pp. 1252–1257 [Abstract] - Pavel Drašar, Vladimír Pouzar, Ivan Černý, Miroslav Havel, Sofia N. Ananchenko and Igor V. Torgov
Use of malonic acid derivatives for the construction of substituted side chains in the position 17β of steroids
1982, Vol. 47, Issue 4, pp. 1240–1251 [Abstract] - Karel Šindelář, Jiří Holubek, Miroslav Ryska, Antonín Dlabač, Jiřina Metyšová, Emil Svátek, Marta Hrubantová, Jiří Protiva and Miroslav Protiva
Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: Derivatives of 11H-dibenz[b,f]-1,4-oxathiepin
1982, Vol. 47, Issue 3, pp. 967–983 [Abstract] - Jiří Křepelka, Iva Vančurová, Jiří Holubek, Jiří Roubík and Drahuše Vlčková
Syntheses and antineoplastic effects of some N-substituted imides of 1-substituted 4-aryl-naphthalene-2,3-dicarboxylic acids
1982, Vol. 47, Issue 1, pp. 304–314 [Abstract] - Pavel Kočovský, Pavel Drašar, Vladimír Pouzar and Miroslav Havel
Synthesis of some westphalen-type cardenolide analogs
1982, Vol. 47, Issue 1, pp. 108–116 [Abstract] - Vladimír Pouzar, Pavel Drašar, Pavel Kočovský and Miroslav Havel
Synthesis of some isocardenolide analogs and 17β-maleimidoandrostane of westphalen structural type
1982, Vol. 47, Issue 1, pp. 96–107 [Abstract] - Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Antonín Dlabač, Marta Hrubantová and Miroslav Protiva
Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: Synthesis of 11-(dimethylaminoalkyl) derivatives of 11H-dibenzo[b,e]-1,4-dioxepin and 11H-dibenzo[b,e]-1,4-dithiepin
1982, Vol. 47, Issue 1, pp. 72–87 [Abstract] - Vladimír Pouzar and Miroslav Havel
Synthesis and absolute configuration at C(20) of 21,26,27-trinor-5α-cholestan-25→20-olide derivatives
1981, Vol. 46, Issue 11, pp. 2758–2765 [Abstract] - Miroslav Protiva, Zdeněk Šedivý, Josef Pomykáček, Václav Bártl, Jiří Holubek and Emil Svátek
Potential metabolites of the noncataleptic neuroleptics: Synthesis of 2-chloro-6-hydroxy(and methoxy)-10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
1981, Vol. 46, Issue 9, pp. 2245–2253 [Abstract] - Zdeněk Vejdělek, Jiří Holubek, Marie Bartošová and Miroslav Protiva
1-(4-Cyclopentylphenyl)ethylamine and derivatives: Synthesis and pharmacological screening
1981, Vol. 46, Issue 9, pp. 2234–2244 [Abstract] - Zdeněk Polívka, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
Fluorinated tricyclic neuroleptics: Synthesis and pharmacology of 2-chloro-8-fluoro-4-(4-methylpiperazino)-4,5-dihydrothieno[2,3-b]-1-benzothiepin
1981, Vol. 46, Issue 9, pp. 2222–2233 [Abstract] - Rudolf Kotva, Jiří Křepelka, Karel Řežábek and Jaroslav Vachek
4-(ω-(2-Amino-6-hydroxy-4-oxo-3,4-dihydro-5-pyrimidinyl)alkyl)benzoic acids with an antineoplastic effect
1981, Vol. 46, Issue 9, pp. 2217–2221 [Abstract] - Jiří Křepelka, Iva Vančurová, Jiří Holubek and Jiří Roubík
Hydrolytic products of 4-aryl-2,3-dicyano-1-naphthol derivatives
1981, Vol. 46, Issue 9, pp. 2207–2216 [Abstract] - Jiří Křepelka and Jiří Holubek
The synthesis of model lactones of cyclolignan type
1981, Vol. 46, Issue 9, pp. 2123–2128 [Abstract] - Jiří Křepelka, Jiří Roubík and Jiří Holubek
1-Substitution derivatives of 4-aryl-2,3-dibromo-1-naphthol
1981, Vol. 46, Issue 9, pp. 2116–2122 [Abstract] - Miroslav Protiva, Karel Šindelář, Zdeněk Šedivý, Jiří Holubek and Marie Bartošová
Potential metabolites of tricyclic neuroleptics: 3,7-Dimethoxy and 7,8-dimethoxy derivatives of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1981, Vol. 46, Issue 8, pp. 1808–1817 [Abstract] - Miroslav Protiva, Karel Šindelář, Jiřina Metyšová, Jiří Holubek, Miroslav Ryska, Emil Svátek, Zdeněk Šedivý and Josef Pomykáček
Fluorinated tricyclic neuroleptics with prolonged action: 3-Fluoro-8-halogeno derivatives of 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
1981, Vol. 46, Issue 8, pp. 1788–1799 [Abstract] - Jiří Křepelka, Iva Vančurová and Jiří Holubek
Some derivatives of 4-aryl-2,3-dicyano-1-naphthol
1981, Vol. 46, Issue 6, pp. 1523–1529 [Abstract] - Rudolf Kotva, Jiří Křepelka, Antonín Černý, Vojtěch Pujman and Miroslav Semonský
Some 2-substituted derivatives of 5-(2-amino-6-hydroxy-4-oxo-3,4-dihydro-5-pyrimidinyl)pentanoic acid
1981, Vol. 46, Issue 6, pp. 1397–1404 [Abstract] - Miroslav Protiva, Zdeněk Šedivý, Josef Pomykáček, Emil Svátek and Jiří Holubek
Potential metabolites of the neuroleptic agent octoclothepin; Synthesis of 8-chloro-2,6-dihydroxy and 8-chloro-3,6-dihydroxy derivatives of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1981, Vol. 46, Issue 5, pp. 1199–1209 [Abstract] - Vladimír Pouzar and Miroslav Havel
Preparation and absolute configuration at C(20) of 21-nor-5α-chol-22-en-24→20-olide derivatives
1981, Vol. 46, Issue 4, pp. 917–925 [Abstract] - Karel Šindelář, Jiří Holubek, Jan Metyš, Marie Bartošová and Miroslav Protiva
Synthesis of 3-(2-alkoxyphenoxy)-2-methyl (or phenyl)propylamines as potential antidepressants
1981, Vol. 46, Issue 3, pp. 597–606 [Abstract] - Zdeněk Vejdělek, Emil Svátek, Jiří Holubek, Jan Metyš, Marie Bartošová and Miroslav Protiva
Synthesis and pharmacological screening of 1-[2-tert-aminoethyl]-8-fluoro-5-[4-fluorophenyl]-2,3,4,5-tetrahydro-1H-1-benzazepines, their 1-[aminoacetyl] analogues and 1-substituted 9-fluoro-6-[4-fluorophenyl]-5,6-dihydro-4H-s-triazolo[4,3-a]-1-benzazepines
1981, Vol. 46, Issue 1, pp. 148–160 [Abstract] - Karel Šindelář, Miroslav Ryska, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Jiří Protiva and Miroslav Protiva
Fluorinated tricyclic neuroleptics with prolonged action: 3-Fluoro-8-trifluoromethyl derivatives of 10-(4-methylpiperazino)- and 10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo-[b,f]thiepin
1981, Vol. 46, Issue 1, pp. 118–140 [Abstract] - Vladimír Pouzar and Miroslav Havel
Preparation and absolute configuration at C(20) of 21-nor-5α-cholan-24→20-olide derivatives
1981, Vol. 46, Issue 1, pp. 107–117 [Abstract] - Zdeněk Vejdělek, Miroslav Rajšner, Antonín Dlabač, Miroslav Ryska, Jiří Holubek, Emil Svátek and Miroslav Protiva
Psychotropic derivatives of 5-phenyl-7-chloro-1,3-dihydro-1,4-benzodiazepin-2-one and contribution to the synthesis of its 5-(2-chlorophenyl) analogue
1980, Vol. 45, Issue 12, pp. 3593–3615 [Abstract] - Miroslav Semonský, Antonín Černý, Jiří Křepelka, Rudolf Kotva, Bohumil Kakáč, Jiří Holubek and Jaroslav Vachek
Some ω-(2-amino-6-hydroxy-4-oxo-3,4-dihydro-5-pyrimidinyl) alkanoic acids, their derivatives and analogues
1980, Vol. 45, Issue 12, pp. 3583–3592 [Abstract] - Karel Šindelář, Jiří Jílek, Jiří Körbl, Fedir Jančik, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
Potential metabolites of the neuroleptic agent chlorprothixene; synthesis and pharmacology of the 3-, 4-, 6- and 7-hydroxy and methoxy derivatives of 2-chloro-9-(3-dimethylaminopropylidene)-thioxanthenes
1980, Vol. 45, Issue 11, pp. 3166–3181 [Abstract] - Jiří Křepelka, Viktor Zikán, Jiří Holubek and Miroslav Semonský
Derivatives of 4-aryl-2,3-dihalogeno-1-naphthol
1980, Vol. 45, Issue 10, pp. 2700–2705 [Abstract] - Jiří Křepelka, Jiří Holubek and Miroslav Semonský
Esters of 4,4-bis(4-ethylphenyl)-2,3-dibromo-2-butenoic acid and 7-ethyl-4-(4-ethylphenyl)-2,3-dibromo-1-naphthol
1980, Vol. 45, Issue 10, pp. 2695–2699 [Abstract] - Irena Červená, Marta Hrubantová, Emil Svátek, Jiří Holubek, Miroslav Ryska, Jiřina Metyšová and Miroslav Protiva
Fluorinated analogues of tricyclic neuroleptics: 6,9-difluoro derivative of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1980, Vol. 45, Issue 10, pp. 2688–2694 [Abstract] - Vladimír Pouzar and Miroslav Havel
Absolute configuration at C(20) of the derivatives of 21-nor-5α-cholane-20,24-diol
1980, Vol. 45, Issue 9, pp. 2443–2451 [Abstract] - Miroslav Kuchař, Bohumila Brunová, Zdeněk Roubal, Jiří Schlanger and Oldřich Němeček
Synthesis of arylacetic acids and their effect on activation of fibrinolysis. Quantitative relations between structure and biological activity
1980, Vol. 45, Issue 5, pp. 1401–1409 [Abstract] - Karel Šindelář, Emil Svátek, Jiří Holubek, Miroslav Ryska, Jiřina Metyšová, Zdeněk Šedivý and Miroslav Protiva
Fluorinated analogues of the tricyclic neuroleptics; 7-Fluoro and 7-trifluoromethyl derivative of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1980, Vol. 45, Issue 4, pp. 1086–1098 [Abstract] - Jiří Křepelka, Jiří Holubek and Miroslav Semonský
Some condensation products of ergoline - I Derivatives with ketones
1980, Vol. 45, Issue 3, pp. 755–760 [Abstract] - Zdeněk Buděšínský, Josef Vavřina, Leon Langšádl and Jiří Holubek
On the synthesis of 4- and 5-pyrimidinyl-diphenyl-(1-imidazolyl)methanes and their antifungal activity
1980, Vol. 45, Issue 2, pp. 539–547 [Abstract] - Karel Šindelář, Jiří Holubek, Emil Svátek and Miroslav Protiva
Synthesis of 3-chloro-5-(4-methylpiperazino)-6,7-dihydro-5H-dibenzo[b,g]thiocin, an eight-membered ring homologue of the neuroleptic agent octoclothepin
1980, Vol. 45, Issue 2, pp. 491–503 [Abstract] - Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiřina Metyšová, Zdeněk Šedivý and Miroslav Protiva
Potential metabolites of the neuroleptic agents noroxyclothepin and oxyclothepin; Synthesis of 8-chloro-3-hydroxy-10-[4-(2-hydroxyethyl)piperazino]- and -10-[4-(3-hydroxypropyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
1979, Vol. 44, Issue 12, pp. 3617–3626 [Abstract] - Zdeněk Vejdělek, Miroslav Rajšner, Emil Svátek, Jiří Holubek and Miroslav Protiva
Synthesis of 7-chloro-5-(6,7,8,9-tetrahydro-5H-benzocyclohepten-2-yl)-2-methylamino-3H-1,4-benzodiazepine 4-oxide and of some related compounds
1979, Vol. 44, Issue 12, pp. 3604–3616 [Abstract] - Miloš Beran, Jiří Křepelka and Miroslav Semonský
Some 6-alkyl derivatives of D-8-ergolin-I-ylacetamide
1979, Vol. 44, Issue 11, pp. 3385–3390 [Abstract] - Miroslav Rajšner, Václav Bártl, Karel Šindelář, Emil Svátek, Jiří Holubek, Jan Metyš and Miroslav Protiva
Synthesis of new dibenzo[b,e]thiepin derivatives related to the antidepressant agent prothiadene
1979, Vol. 44, Issue 8, pp. 2536–2549 [Abstract] - Jiří O. Jílek, Jiří Holubek, Emil Svátek, Miroslav Ryska, Josef Pomykáček and Miroslav Protiva
Reaction of some 3-(phenylthioaryl)propionic acids with polyphosphoric acid; Formation of 2H-cyclopenta[k,l]thioxanthenes
1979, Vol. 44, Issue 7, pp. 2124–2138 [Abstract] - Antonín Černý, Jiří Křepelka and Miroslav Semonský
Some 6-substituted derivatives of D-8-cyanomethylergoline-I and D-8-methylergoline-I
1979, Vol. 44, Issue 3, pp. 946–951 [Abstract] - Vladimír Pouzar and Alois Vystrčil
Preparation of 12,20-disubstituted lupane derivatives
1979, Vol. 44, Issue 1, pp. 194–210 [Abstract] - Jiří Jílek, Jiří Holubek, Emil Svátek, Marie Bartošová, Jiřina Metyšová, Josef Pomykáček and Miroslav Protiva
8-Chloro-3-hydroxy-10-piperazino-10,11-dihydrodibenzo[b,f]thiepins, their O-methyl derivatives and further potential metabolites of the neuroleptic agent octoclothepin
1978, Vol. 43, Issue 11, pp. 3092–3102 [Abstract] - Václav Bártl, Jiří Holubek, Jiří Němec, Marie Bartošová and Miroslav Protiva
Derivatives of 8-chloro-10,11-dihydrodibenzo[b,f]thiepin-10-amine, -10-ol and -10-thiol; Synthesis and pharmacological screening
1978, Vol. 43, Issue 9, pp. 2427–2443 [Abstract] - Vladimír Pouzar and Alois Vystrčil
Preparation of 29-acetoxy-30-norlupan-20-one derivatives with the substituted ring C
1978, Vol. 43, Issue 8, pp. 2190–2203 [Abstract] - Miroslav Rajšner, Zdeňka Kopicová, Jiří Holubek, Emil Svátek, Jan Metyš, Marie Bartošová, František Mikšík and Miroslav Protiva
4,4-Bis(4-fluorophenyl)butylamines and their cyclic analogues; An efficient synthesis of the neuroleptic penfluridol
1978, Vol. 43, Issue 7, pp. 1760–1777 [Abstract] - Viktor Zikán, Miroslav Semonský, Bohumil Kakáč, Jiří Holubek and Karel Řežábek
Reactions of methyl esters of 3-bromo-4-(4-alkoxyphenyl)-4-oxo-2-butenoic acids with diethyl sodium malonate
1978, Vol. 43, Issue 7, pp. 1727–1731 [Abstract] - Jiří Křepelka and Miroslav Semonský
Some N-nitrososubstituted derivatives of ergoline I
1978, Vol. 43, Issue 7, pp. 1723–1726 [Abstract]
