CCCC 1988, Volume 53, Issue 1, Abstracts pp. 132-144, Articles by the same authors | Collection of Czechoslovak Chemical Communications

CCCC > Archive > 1988, Volume 53 > Issue 1 > p. 132 > Articles by the same authors

Collect. Czech. Chem. Commun. 1988, 53, 132-144
https://doi.org/10.1135/cccc19880132

Potentional anxiolytics and hypnotics: 1-(Alkanesulfonamidoalkyl)-6-aryl-8-halogeno-s-triazolo[4,3-a]-1,4-benzodiazepines and related compounds

Zdeněk Vejdělek^a, Jan Metyš^a, Jiří Holubek^a, Miloš Buděšínský^b, Emil Svátek^a, Oluše Matoušová^a and Miroslav Protiva^a

^a Research Institute for Pharmacy and Biochemistry, 130 60 Prague 3
^b Institute of Organic Chemistry and Biochemistry Czechoslovak Academy of Sciences, 166 10 Prague 6

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2005, Vol. 70, Issue 4, pp. 466–478 [Abstract]
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Synthesis and Biological Activity of 7a-Homo- and 7a,7b-Dihomo-5α-cholestane Analogues of Brassinolide
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2003, Vol. 68, Issue 5, pp. 931–950 [Abstract]
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A Facile Synthesis of Selectively Protected Linear Oligoamines
2003, Vol. 68, Issue 4, pp. 744–750 [Abstract]
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2002, Vol. 67, Issue 12, pp. 1805–1819 [Abstract]
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Synthesis of Linear Steroid Oligoesters Based on Etienic Acid
2002, Vol. 67, Issue 11, pp. 1709–1718 [Abstract]
Jan Mařík, Miloš Buděšínský, Jiřina Slaninová and Jan Hlaváček*
Synthesis, Bioassay and NMR Study of Methyleneoxy Isosters of Oxytocin and Vasopressin
2002, Vol. 67, Issue 3, pp. 373–392 [Abstract]
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Minor Ecdysteroid Components of Leuzea carthamoides
2002, Vol. 67, Issue 1, pp. 124–139 [Abstract]
Hana Chodounská, Miloš Buděšínský, Romana Šídová, Miroslav Šíša, Alexander Kasal and Ladislav Kohout*
Simple NMR Determination of 5α/5β Configuration of 3-Oxosteroids
2001, Vol. 66, Issue 10, pp. 1529–1544 [Abstract]
Ivan Černý*, Miloš Buděšínský, Vladimír Pouzar and Pavel Drašar
Linear Chaining of Etienic Acid Derivatives with the Amide Bond. Synthesis of Oligomeric Steroids
2001, Vol. 66, Issue 6, pp. 933–946 [Abstract]
Jindřich Karban*, Miloš Buděšínský, Miloslav Černý and Tomáš Trnka
Synthesis and NMR Spectra of 1,6-Anhydro-2,3-dideoxy-2,3-epimino- and 1,6-Anhydro-3,4-dideoxy-3,4-epimino-β-D-hexopyranoses
2001, Vol. 66, Issue 5, pp. 799–819 [Abstract]
Petr Alexander*, Antonín Holý, Miloš Buděšínský and Milena Masojídková
Synthesis of Acyclic Nucleotide Analogues Derived from N³-Substituted Isoguanine
2000, Vol. 65, Issue 11, pp. 1713–1725 [Abstract]
Ivan Černý*, Vladimír Pouzar, Miloš Buděšínský and Pavel Drašar
Synthesis of Symmetrical Bis-Steroid Pyrazines Connected via D-Rings
2000, Vol. 65, Issue 10, pp. 1597–1608 [Abstract]
Jan Hlaváček*, Renáta Marcová, Miloš Buděšínský and Jiřina Slaninová
1-Deamino-1(15)-carba and -Dicarba Analogues of Endothelin-1
2000, Vol. 65, Issue 3, pp. 407–424 [Abstract]
Martin Chadim, Miloš Buděšínský, Jana Hodačová and Jiří Závada*
A Covalently Bound Template in the Regioselective Synthesis of Bis(tetraazacrown)s
2000, Vol. 65, Issue 1, pp. 99–105 [Abstract]
Alexander Kasal*, Miloš Buděšínský, Jan Pelnař, Michael A. Bruck* and Michael F. Brown
Structures and Synthesis of 4a-Homo-7,19-dinorsteroids, X-Ray Crystallography and NMR Spectroscopy
1999, Vol. 64, Issue 12, pp. 2019–2034 [Abstract]
Barbora Slavíková, Alexander Kasal* and Miloš Buděšínský
Autoxidation vs Hydrolysis in 16α-Acyloxy Steroids
1999, Vol. 64, Issue 7, pp. 1125–1134 [Abstract]
Antonín Holý*, Miloš Buděšínský, Jaroslav Podlaha and Ivana Císařová
Synthesis of Quaternary 1-[2-(Phosphonomethoxy)ethyl] Derivatives of 2,4-Diaminopyrimidine and Related Acyclic Nucleotide Analogs
1999, Vol. 64, Issue 2, pp. 242–256 [Abstract]
Alexander Kasal, Jiří Polman and Miloš Buděšínský
Hydrogenation of a Tetrasubstituted Double Bond: Synthesis of 5-Methyl-19-nor-5β-pregnanes
1998, Vol. 63, Issue 10, pp. 1549–1563 [Abstract]
Jiří Kroutil, Tomáš Trnka, Miloš Buděšínský and Miloslav Černý
Preparation of 2,3-Dideoxy-2,3-epimino and 3,4-Dideoxy-3,4-epimino Derivatives of 1,6-Anhydro-β-D-hexopyranoses by Mitsunobu Reaction
1998, Vol. 63, Issue 6, pp. 813–825 [Abstract]
Tomáš Kraus, Miloš Buděšínský and Jiří Závada
Novel Amphiphilic Cyclodextrins: Per[6-deoxy-6-(4,5-dicarboxy-1,2,3-triazol-1-yl)-2,3-di-O-methyl] Derivatives
1998, Vol. 63, Issue 4, pp. 534–540 [Abstract]
Jaroslav Litera, Miloš Buděšínský, Ján Urban and Milan Souček
Peptide Inhibitors of Aspartic Proteinases with Hydroxyethylene Isostere Replacement of Peptide Bond. I. Preparation of Four Diastereoisomeric (2R or 2S,4R or 4S,5S)-2-Benzyl-5-[(tert-butoxycarbonyl)amino]-4-hydroxy-6-phenylhexanoic Acids
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Miloš Tichý, Luděk Ridvan, Miloš Buděšínský, Jiří Závada, Jaroslav Podlaha and Ivana Císařová
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Mária Haladová, Eva Eisenreichová, Pavel Mučaji, Miloš Buděšínský and Karel Ubik
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1998, Vol. 63, Issue 2, pp. 205–210 [Abstract]
Jan Sejbal, Jiří Klinot, Miloš Buděšínský and Jiří Protiva
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Alexander Kasal, Barbora Slavíková, Ladislav Kohout and Miloš Buděšínský
The Synthesis of A-Homo-B-norandrostanes: The Effect of a Hydroxyl on the Course of Hydrogenation of the ∆⁹-Double Bond
1997, Vol. 62, Issue 10, pp. 1631–1641 [Abstract]
Hubert Hřebabecký, Miloš Buděšínský, Milena Masojídková, Zdeněk Havlas and Antonín Holý
1-(3,5-O-Alkylidene-2-deoxy-4-C-hydroxymethyl-α-L-threo-pentofuranosyl)uracils
1997, Vol. 62, Issue 6, pp. 957–970 [Abstract]
Barbora Slavíková, Alexander Kasal and Miloš Buděšínský
Dihydrotestosterone with an Ammonium Centre in the Position 16β
1997, Vol. 62, Issue 4, pp. 656–664 [Abstract]
Miroslav Kuchař, Marie Poppová, Antonín Jandera, Vladimíra Panajotovová, Hana Zůnová, Miloš Buděšínský, Hana Tomková, Alexandr Jegorov and Jan Taimr
Chiral Forms of 4-(2',4'-Difluorobiphenyl-4-yl)-2-methyl-4-oxobutanoic Acid (Flobufen) and Its Metabolite.Synthesis and Basic Biological Properties
1997, Vol. 62, Issue 3, pp. 498–509 [Abstract]
Thi Thu Huong Nguyen, Jiří Protiva, Eva Klinotová, Jiří Urban and Miroslav Protiva
Synthesis of 24-(Piperidin-1-yl, Morpholin-4-yl and 4-Methylpiperazin-1-yl)-5β-cholan-3α-ols and Four Hydroxylated 23-(4,5-Dihydroimidazol-2-yl)-24-nor-5β-cholanes
1997, Vol. 62, Issue 3, pp. 471–478 [Abstract]
Pavel Mučaji, Mária Haladová, Eva Eisenreichová, Miloš Buděšínský and Karel Ubik
Jatropham 5-O-β-D-Glucopyranoside from Lilium candidum L.
1996, Vol. 61, Issue 11, pp. 1662–1664 [Abstract]
Miloslav Černý, Tomáš Trnka and Miloš Buděšínský
Preparation and Reactions of 2-Chloroethyl 1-Thio-β-D-glycopyranosides Derived from D-Galactose, D-Glucose, and 2-Acetamido-2-deoxy-D-glucose
1996, Vol. 61, Issue 10, pp. 1489–1500 [Abstract]
Jan Sejbal, Jiří Klinot and Miloš Buděšínský
Functionalization of Lupane with Chromium(VI) Oxide. A Remark on the Structure of Clerodone
1996, Vol. 61, Issue 9, pp. 1371–1379 [Abstract]
Jan Sejbal, Jiří Klinot and Miloš Buděšínský
Oleanane Triterpenoids Functionalized at C-25 and C-26
1996, Vol. 61, Issue 9, pp. 1360–1370 [Abstract]
Wim F. Vranken, Miloš Buděšínský, Franky Fant, Kris Boulez, Hélène Gras-Masse and Frans A. M. Borremans
Conformational Features of a Synthetic Cyclic Peptide Corresponding to the Complete V3 Loop of the ELI HIV-1 Strain in Water
1996, Vol. 61, Issue 5, pp. 742–750 [Abstract]
Alexander Kasal and Miloš Buděšínský
Partial Modifications of Hydroxy Groups in 5-Methyl-5β-estr-9-ene Derivatives
1996, Vol. 61, Issue 2, pp. 276–287 [Abstract]
Václav Suchý, Miloš Buděšínský, Karel Ubik, Daniel Grančai and Vlasta Földešiová
NMR Determination of the Structure of Peracetylated Icariside B₂ from Veratrum Lobelianum BERNH.
1995, Vol. 60, Issue 8, pp. 1380–1385 [Abstract]
Dalibor Štys, Ján Novák, Viktor Krchňák, Josef Vágner, Petr Štrop and Miloš Buděšínský
Time Dependence of Immunoresponse of Different Epitopes of gp41 and Its Relation to the Structure of Short Peptide Fragments of gp41
1995, Vol. 60, Issue 6, pp. 1054–1064 [Abstract]
Václav Křeček, Stanislav Hilgard, Miloš Buděšínský and Alois Vystrčil
E-Homolupane Derivatives Substituted in Position 17 and 22a. ¹H NMR, ¹³C NMR and IR Spectra
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Miloš Buděšínský, Miloslav Černý, Ivan Černý, Stanislav Sámek and Tomáš Trnka
Preparation of β-D-Glucopyranosyl Derivatives of 1,6:2,3- and 1,6:3,4-Dianhydro-β-D-hexopyranoses and Their ¹H and ¹³C NMR Spectra
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X-Ray Structure Analysis and NMR Study of Sesquiterpene Lactone Hirsutolide
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Urszula Rychłewska, Miloš Buděšínský, Beata Szczepanska, Ełżbieta Błoszyk and Miroslav Holub
Two Crystalline Forms of Sesquiterpene Lactone Helenalin - X-Ray and NMR Study
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Thi Thu Huong Nguyen, Jiří Urban, Eva Klinotová, Jan Sejbal, Jiří Protiva, Pavel Drašar and Miroslav Protiva
Synthesis of Several Hydroxylated 23-(Benzimidazol-2-yl-, Benzoxazol-2-yl and Benzothiazol-2-yl)norcholanes and Some Related Compounds
1995, Vol. 60, Issue 2, pp. 257–275 [Abstract]
Dana Hocková, Milena Masojídková, Miloš Buděšínský and Antonín Holý
Acyclic Nucleoside and Nucleotide Analogs Derived from 2-Azaadenine
1995, Vol. 60, Issue 2, pp. 224–236 [Abstract]
Ivan Černý, Miloš Buděšínský, Pavel Drašar and Vladimír Pouzar
Construction of the Side-Chain in 14β-Androst-5-ene Derivatives. Preparation of 14β-Pregnenolone
1994, Vol. 59, Issue 12, pp. 2691–2704 [Abstract]
Miloš Buděšínský, Gerard Nowak, Urszula Rychłewska, Derek J. Hodgson, David Šaman, Włodzimierz M. Daniewski, Bohdan Drożdż and Miroslav Holub
Structure of Sesquiterpenic Lactones of Some Species of Subtribe Centaureinae DUMORT.
1994, Vol. 59, Issue 5, pp. 1175–1202 [Abstract]
Maria Spassova, Hana Dvořáková, Antonín Holý, Miloš Buděšínský and Milena Masojídková
Synthesis of N-(3-Azido-2-hydroxypropyl), N-(3-Phthalimido-2-hydroxypropyl) and N-(3-Amino-2-hydroxypropyl) Derivatives of Heterocyclic Bases
1994, Vol. 59, Issue 5, pp. 1153–1174 [Abstract]
Miloš Buděšínský, Nestor Perez Souto and Miroslav Holub
Sesquiterpenic Lactones of Some Species of Genus Vernonia SCHREB.
1994, Vol. 59, Issue 4, pp. 913–928 [Abstract]
Karel Šindelář, Alexandra Šilhánková, Jiří Urban, Jan Metyš, Martin Valchář and Zdeněk Polívka
Antihistamine Substances. Tricyclic Analogues of N-(4,4-Diphenyl-3-butene-1-yl)nipecotic Acid and Some Related Compounds
1994, Vol. 59, Issue 3, pp. 667–674 [Abstract]
Eva Klinotová, Jiří Klinot, Václav Křeček, Stanislav Hilgard, Miloš Buděšínský and Jan Malát
Structure of Dimeric Compounds Obtained from 3β-Acetoxy-21,22-dioxo-18α,19βH-ursan-28,20β-olide
1993, Vol. 58, Issue 7, pp. 1675–1691 [Abstract]
Urszula Rychłewska, Beata Szczepanska, Miloš Buděšínský, David Šaman, Soňa Vašíčková, Bohdan Drożdż, Halina Grabarczyk and Miroslav Holub
Crystal Structure of the Native Sesquiterpene Lactone Arctolide
1993, Vol. 58, Issue 4, pp. 909–917 [Abstract]
Jaroslav Píš, Jiří Hykl, Miloš Buděšínský and Juraj Harmatha
Cyclic Phenylboronates of Ecdysteroids as Products of Regiospecific Reaction with Phenylboronic Acid
1993, Vol. 58, Issue 3, pp. 612–618 [Abstract]
Eva Klinotová, Jiří Klinot, Václav Křeček, Miloš Buděšínský and Bohumil Máca
21,22-Disubstituted 18α,19βH-Ursane Derivatives with Oxabicyclooctane System in Ring E
1993, Vol. 58, Issue 1, pp. 173–190 [Abstract]
Juraj Bernát, Ladislav Kniežo, Gabriela Birošová, Miloš Buděšínský, Jaroslav Podlaha, Jana Podlahová and Jiří Novotný
Reactions of PO(NCS)₃ with 4-Hydroxy-1,3-dioxanes. Crystal Structure of rel-(2S,4R,5S,6S)-2,6-Diethyl-5-methyl-4-(N'-benzylthioureido)-1,3-dioxane
1992, Vol. 57, Issue 6, pp. 1299–1313 [Abstract]
Ełżbieta Błoszyk, Urszula Rychłewska, Beata Szczepanska, Miloš Buděšínský, Bohdan Drożdż and Miroslav Holub
Sesquiterpene Lactones of Ambrosia artemisiifolia L. and Ambrosia trifida L. Species
1992, Vol. 57, Issue 5, pp. 1092–1102 [Abstract]
Karel Stránský, Marta Semerdžieva, Miroslav Otmar, Želimír Procházka, Miloš Buděšínský, Karel Ubik, Jitka Kohoutová and Ludvík Streinz
Antifungal Antibiotic from the Mushroom Agrocybe aegerita (BRIG.) SING.
1992, Vol. 57, Issue 3, pp. 590–603 [Abstract]
Václav Křeček, Miloš Buděšínský and Alois Vystrčil
Preparation of 20R and 20S Acetylamino-30-norlupane Derivatives
1992, Vol. 57, Issue 3, pp. 556–564 [Abstract]
Otto Exner and Miloš Buděšínský
Carbon-13 Substituent-Induced Chemical Shifts: Monosubstituted Benzene Derivatives
1992, Vol. 57, Issue 3, pp. 497–507 [Abstract]
Irena Valterová, Miloš Buděšínský and Jan Vrkoč
Defensive substances from the frontal gland secretion of Nasutitermes nigriceps termite soldiers
1991, Vol. 56, Issue 12, pp. 2969–2977 [Abstract]
Jindřich Jindřich, Miloslav Černý, Tomáš Trnka and Miloš Buděšínský
The synthesis of 4-O-oligoethylene glycol derivatives of 1,6-anhydro-β-D-glucopyranose and crown-ethers formed by their intramolecular cyclization
1991, Vol. 56, Issue 12, pp. 2950–2963 [Abstract]
Jan Sejbal, Jiří Klinot, Miloš Buděšínský and Jiří Protiva
Functionalization of 3β,28-lupanediol diacetate with chromium(VI) oxide
1991, Vol. 56, Issue 12, pp. 2936–2949 [Abstract]
Eva Klinotová, Václav Křeček, Jiří Klinot, Miloš Buděšínský, Jaroslav Podlaha, Jana Podlahová and Jiří Ječný
An unusual reaction of a bridged triterpenoid α-diketone with acetic anhydride
1991, Vol. 56, Issue 12, pp. 2917–2935 [Abstract]
Miroslav Protiva
Fifty years in chemical drug research
1991, Vol. 56, Issue 11, pp. 2501–2772 [Abstract]
Karel Šindelář, Jiří Holoubek, Emil Svátek, Jan Metyš, Hana Blehová and Zdeněk Polívka
Potential antihistaminics: Tricyclic carboxylic acids derived from 6,11-dihydrodibenzo[b,e]thiepine and 4,9-dihydrothieno[2,3-c]-2-benzothiepine
1991, Vol. 56, Issue 11, pp. 2482–2493 [Abstract]
Vojtěch Kmoníček, Josef Pomykáček, Jiří Holoubek, Emil Svátek, Martin Valchář, Jiřina Metyšová and Zdeněk Polívka
Potential antidepressants: 2-(fluoro-, chloro-, bromo- and cyanophenylthio)benzylamines as inhibitors of 5-hydroxytryptamine and noradrenaline re-uptake in brain
1991, Vol. 56, Issue 11, pp. 2468–2481 [Abstract]
Otto Exner and Miloš Buděšínský*
Correlation of substituent – inducted chemical shifts of aromatic protons: Substituted benzonitriles and methyl benzoates
1991, Vol. 56, Issue 11, pp. 2234–2250 [Abstract]
Jan Sejbal, Jiří Klinot and Miloš Buděšínský
Photolyses and pyrolyses of triterpenoid nitrites
1991, Vol. 56, Issue 8, pp. 1732–1743 [Abstract]
Miloš Buděšínský, Alexander Kasal, Želimír Procházka, Huynh Kim Thoa, Soňa Vašíčková and Pavel Kočovský
Revision of the structure of 3-methoxy-14α-hydroxy-D-homo-1,3,5-(10)-estratrien-17a-one. A simple ¹H NMR method for the determination of configuration of hydroxy group in position 5 and/or 14 of the D-homo-steroid skeleton
1991, Vol. 56, Issue 7, pp. 1512–1524 [Abstract]
Zdeněk Arnold, Miloš Buděšínský and Magdalena Pánková
Reactivity of triformylmethane. I. Reactions of triformylmethane with selected types of amino compounds
1991, Vol. 56, Issue 5, pp. 1019–1031 [Abstract]
Alois Vystrčil, Václav Křeček, Jiří Protiva and Miloš Buděšínský
Anhydrobetulin and its derivatives
1991, Vol. 56, Issue 4, pp. 886–904 [Abstract]
Karel Šindelář, Josef Pomykáček, Jiří Holubek, Emil Svátek, Martin Valchář, Karel Dobrovský, Jiřina Metyšová and Zdeněk Polívka
Potential antidepressants and selective inhibitors of 5-hydroxytryptamine re-uptake in the brain: Synthesis of several potential metabolites of moxifetin and of two A-ring fluorinated analogues
1991, Vol. 56, Issue 2, pp. 459–477 [Abstract]
Miloš Buděšínský, Dan Johnels, Ulf Edlund and Otto Exner
Carbon-13 substituent-induced chemical shifts in benzene derivatives: Substituted anilines
1991, Vol. 56, Issue 2, pp. 368–385 [Abstract]
Vladimír Valenta, Jiří Holubek, Emil Svátek, Martin Valchář, Ivan Krejčí and Miroslav Protiva
Potential nootropic agents: Synthesis of some (2-oxo-1-pyrrolidinyl)acetamides and some related compounds
1990, Vol. 55, Issue 11, pp. 2756–2764 [Abstract]
Václav Černý and Miloš Buděšínský
A route to 24-epibrassinolide from ergosterol avoiding the use of osmium tetroxide
1990, Vol. 55, Issue 11, pp. 2738–2755 [Abstract]
Ivan Černý, Vladimír Pouzar, Miloš Buděšínský, Pavel Drašar and Miroslav Havel
Epimeric 17-hydroxy derivatives of 14β-androst-5-en-3β-yl acetate
1990, Vol. 55, Issue 10, pp. 2510–2520 [Abstract]
Zdeněk Vejdělek and Miroslav Protiva
Synthetic experiments aiming at 1,2,4,5-tetrahydro-3-benzothiepin derivatives
1990, Vol. 55, Issue 9, pp. 2351–2356 [Abstract]
Zdeněk Vejdělek and Miroslav Protiva
Synthesis of some derivatives of 1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine and 11-phenyl-5,6-dihydro-11H-s-triazolo[3,4-b]-3-benzazepine
1990, Vol. 55, Issue 9, pp. 2345–2350 [Abstract]
Vladimír Valenta, Jiří Holubek, Emil Svátek and Miroslav Protiva
Potential cholinergic and anticholinergic compounds: Synthesis of 2,8-substituted 2,8-diazaspiro[4,5]decane-1,3-diones
1990, Vol. 55, Issue 9, pp. 2304–2316 [Abstract]
Karel Šindelář, Jiří Jílek, Josef Pomykáček, Vladimír Valenta, Marta Hrubantová, Marie Vlková, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiřina Metyšová and Miroslav Protiva
Tricyclic neuroleptics: Synthesis of metabolites of isofloxythepin and some related compounds
1990, Vol. 55, Issue 9, pp. 2282–2303 [Abstract]
Jiří Jílek, Miroslav Rajšner, Vladimír Valenta, Miloš Borovička, Jiří Holubek, Miroslav Ryska, Emil Svátek, Jan Metyš and Miroslav Protiva
Synthesis of piperidine derivatives as potential analgetic agents
1990, Vol. 55, Issue 7, pp. 1828–1853 [Abstract]
Vojtěch Kmoníček, Emil Svátek, Jiří Holubek, Miroslav Ryska, Martin Valchář and Miroslav Protiva
Synthesis of 1-acyl- and 1-(thioacyl)-4-benzylpiperazines as potential antidepressants
1990, Vol. 55, Issue 7, pp. 1817–1827 [Abstract]
Vladimír Valenta, Karel Šindelář, Jiří Holubek, Miroslav Ryska, Ivan Krejčí, Antonín Dlabač and Miroslav Protiva
Potential nootropic agents: Synthesis of a series of (2-oxo-1-pyrrolidinyl)acetic acid piperazides
1990, Vol. 55, Issue 6, pp. 1613–1629 [Abstract]
Vojtěch Kmoníček, Zdeněk Vejdělek and Miroslav Protiva
Synthesis of a series of 5-methyl-1H-imidazole-4-ylmethyl sulfides
1990, Vol. 55, Issue 6, pp. 1602–1612 [Abstract]
Karel Šindelář, Jiří Holubek, Ivan Koruna, Marta Hrubantová and Miroslav Protiva
Modified syntheses of 2-(methylthio)-10-(2-(1-methyl-2-piperidinyl)ethyl)phenothiazine (thioridazine) and 1-(3-(2-(methylsulfonyl)-10-phenothiazinyl)propyl)-piperidine-4-carboxamide (metopimazine)
1990, Vol. 55, Issue 6, pp. 1586–1601 [Abstract]
Irena Valterová, Miloš Buděšínský, Jan Vrkoč and Glenn D. Prestwich
(8Z)-1(15),8(9)-Trinervitadien-3α-ol from Nasutitermes nigriceps termites. The revised structure for a deffense compound of Trinervitermes gratiosus termites
1990, Vol. 55, Issue 6, pp. 1580–1585 [Abstract]
Sergazy M. Adekenov, Miloš Buděšínský, Metram A. Abdikalikov, Coblandy M. Turdybekov, David Šaman, Ełżbieta Błoszyk, Bohdan Drożdż and Miroslav Holub
Sesquiterpenic lactones of the Inula caspica BLUME species
1990, Vol. 55, Issue 6, pp. 1568–1579 [Abstract]
Ełżbieta Błoszyk, Miloš Buděšínský, Włodzimierz M. Daniewski, Eva Pešková, Bohdan Drożdż and Miroslav Holub
Sesquiterpenic lactones of Inula aschersoniana JANKA var. aschersoniana species
1990, Vol. 55, Issue 6, pp. 1562–1567 [Abstract]
Jan Ježek, Evgenii A. Makarov, Tamara A. Balashova, Miloš Buděšínský, Tatyana M. Andronova and Vadim T. Ivanov
Synthesis of tetrasaccharide containing glycopeptides related to bacterial cell wall starting from free tetrasaccharide by the pentafluorophenyl ester method
1990, Vol. 55, Issue 5, pp. 1326–1335 [Abstract]
Vladimír Valenta, Jiří Holubek, Emil Svátek, Oluše Matoušová, Jiřina Metyšová and Miroslav Protiva
Potential neuroleptics of the orthopramide series; synthesis of heterocyclic 5-amino-2-methoxybenzamides and of some related compounds
1990, Vol. 55, Issue 5, pp. 1297–1310 [Abstract]
Zdeněk Vejdělek and Miroslav Protiva
Potential antidepressants and tranquillizers: Synthesis of some 9-(aminoalkoxy)-2,3,6,7-tetrahydro-1H,5H-benzo[ij] quinolizines and 1-(substituted amino)-3-(1-naphthoxy)-2-propanols
1990, Vol. 55, Issue 5, pp. 1290–1296 [Abstract]
Miroslav Protiva, Vladimír Valenta, Zdeňka Kopicová, Juraj Lukáč, Jiří Holubek and Ivan Krejčí
Potential cerebral stimulants: Esters of 2-dimethylaminoethanol with some lipophilic carboxylic acids
1990, Vol. 55, Issue 5, pp. 1278–1289 [Abstract]
Jiří Jílek, Karel Šindelář, Jaroslava Grimová, Eva Maturová, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Jan Metyš, Marta Hrubantová and Miroslav Protiva
Potential antidepressant and anti-inflammatory agents: 4-(2-Propylthio)acetophenone oximes and 4-(2-propylthio)phenylalkanoic acids
1990, Vol. 55, Issue 5, pp. 1266–1277 [Abstract]
Jiří Urban, Zdeněk Šedivý, Jiří Holubek, Emil Svátek, Miroslav Ryska, Ivan Koruna, Antonín Dlabač, Martin Valchář, Jiřina Metyšová, Zdeněk Polívka, Karel Šindelář, Josef Pomykáček, Marta Hrubantová and Miroslav Protiva
Potential antidepressants: 1-(2-(Methoxy- and hydroxyphenylthio)phenyl)-2-propylamines
1990, Vol. 55, Issue 4, pp. 1077–1098 [Abstract]
Vladimír Valenta, Zdeněk Vejdělek, Karel Šindelář and Miroslav Protiva
Potential anticonvulsants: Some derivatives and analogues of 2-propylpentanoic acid
1990, Vol. 55, Issue 4, pp. 1067–1076 [Abstract]
Miloš Beran, Antonín Černý, Miroslav Kuchař, Hana Adamírová, Jiří Holubek, Jan Taimr, Jaroslav Vachek, Maria Frühaufová, Karel Řežábek, Martin Valchář and Ivan Krejčí
9,10-Dihydroergopeptines modified in position 6
1990, Vol. 55, Issue 3, pp. 819–832 [Abstract]
Vladimír Valenta, Marie Vlková, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
Potential neuroleptics of the orthopramide series; Synthesis of N-(3-(tert.amino)propyl)-5-sulfamoyl-2-methoxybenzamides
1990, Vol. 55, Issue 3, pp. 797–808 [Abstract]
Karel Šindelář, Jiří Holubek, Emil Svátek, Jiří Schlanger, Antonín Dlabač, Martin Valchář, Marta Hrubantová and Miroslav Protiva
Open-ring models of hetero-cannabinoids: Synthesis of 2-(alkylthio)-5-(2-aminoethyl)hydroquinone derivatives
1990, Vol. 55, Issue 3, pp. 782–796 [Abstract]
Jiří Klinot, Miloš Buděšínský and Jarmil Světlý
Conformation of ring A in triterpenoid and 4,4-dimethylsteroid 3-ketones. Chemical shifts of methyl protons and lanthanide and benzene induced shifts
1990, Vol. 55, Issue 3, pp. 766–781 [Abstract]
Miroslav Kuchař, Jaroslava Grimová, Václav Rejholec, Hana Tomková, Magda Jelínková and Jiří Holubek
Use of QSAR in design of antiinflammatory fluorinated arylalkanoic acids
1990, Vol. 55, Issue 1, pp. 296–306 [Abstract]
Karel Šindelář, Vladimír Valenta, Jiří Holubek, Oluše Matoušová and Miroslav Protiva
Potential antidepressants. Synthesis of 6,11-dihydrodibenzo[b,e]thiepin-11-yl (dimethylaminomethyl)phenyl ethers, sulfides, amines and some related compounds
1990, Vol. 55, Issue 1, pp. 282–295 [Abstract]
Jiří Jílek, Karel Šindelář, Josef Pomykáček, Vojtěch Kmoníček, Zdeněk Šedivý, Marta Hrubantová, Jiří Holubek, Emil Svátek, Miroslav Ryska, Ivan Koruna, Martin Valchář, Antonín Dlabač, Jiřina Metyšová, Nataša Dlohožková and Miroslav Protiva
Potential antidepressants: 2-(Methoxy- and hydroxyphenylthio)benzylamines as selective inhibitors of 5-hydroxytryptamine re-uptake in the brain
1989, Vol. 54, Issue 12, pp. 3294–3338 [Abstract]
Jaroslav Podlaha, Miloš Buděšínský, Jana Podlahová and Jindřich Hašek
Crystal and solution structure of (E)-1,2-bis(ethylsulphonyl)cyclobutane-1,2-dicarbonitrile
1989, Vol. 54, Issue 12, pp. 3253–3259 [Abstract]
Marcela Krečmerová, Miloslav Černý, Miloš Buděšínský and Antonín Holý
Utilization of 1,6-anhydrohexoses for the preparation of some aliphatic adenosine analogs
1989, Vol. 54, Issue 10, pp. 2753–2766 [Abstract]
Zdeněk Polívka, Miloš Buděšínský, Jiří Holubek, Bohdan Schneider, Zdeněk Šedivý, Emil Svátek, Oluše Matoušová, Jan Metyš, Martin Valchář, Radomír Souček and Miroslav Protiva
4H-Benzo[4,5]cyclohepta[1,2-b]thiophenes and 9,10-dihydro derivatives - Sulfonium analogues of pizotifen and ketotifen; Chirality of ketotifen; Synthesis of the 2-bromo derivative of ketotifen
1989, Vol. 54, Issue 9, pp. 2443–2469 [Abstract]
Jiří Jílek, Jiří Urban, Vojtěch Kmoníček, Josef Pomykáček, Jiří Holubek, Emil Svátek, Oluše Matoušová, Jan Metyš, Martin Valchář, Stanislav Wildt and Miroslav Protiva
Potential anticonvulsants: 3-Chlorobenzophenone derivatives
1989, Vol. 54, Issue 8, pp. 2248–2260 [Abstract]
Karel Šindelář, Marta Hrubantová, Emil Svátek, Oluše Matoušová, Jiřina Metyšová, Martin Valchář and Miroslav Protiva
Potential antidepressants: 4-(Thioaryloxy)piperidines
1989, Vol. 54, Issue 8, pp. 2240–2247 [Abstract]
Jiří Jílek, Jiří Urban, Petr Taufmann, Jiří Holubek, Antonín Dlabač, Martin Valchář and Miroslav Protiva
Potential antidepressants: 2-(Phenylthio)aralkylamines
1989, Vol. 54, Issue 7, pp. 1995–2008 [Abstract]
Vladimír Valenta, Marie Vlková, Jiří Holubek, Jiřina Metyšová and Miroslav Protiva
Potential antidepressants: 10-Amino-2-chloro-10,11-dihydrodibenzo[b,f]thiepins
1989, Vol. 54, Issue 7, pp. 1979–1994 [Abstract]
Irena Červená, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
Potential antidepressants: 2-(Aminoalkoxy)biphenyls and some related ω-substituted 2-alkoxybiphenyls
1989, Vol. 54, Issue 7, pp. 1966–1978 [Abstract]
Irena Červená, Jiří Holubek, Emil Svátek, Miroslav Ryska and Miroslav Protiva
Potential antidepressants: 6-(Aminoalkoxy)dibenzo[b,f]thiepin-10(11H)-ones and 6-(aminoalkoxy)-10,11-dihydrodibenzo[b,f]thiepin-10-ols
1989, Vol. 54, Issue 7, pp. 1955–1965 [Abstract]
Miloš Buděšínský and Jiří Klinot
Conformation of ring A in triterpenoid ketones. Carbon-13 chemical shifts and spin-lattice relaxation times of lupane and 18α-oleanane derivatives
1989, Vol. 54, Issue 7, pp. 1928–1939 [Abstract]
Miloš Buděšínský, Halina Grabarczyk, Włodzimierz M. Daniewski, Andrzej Wawrzuń, Maria Gulumka, David Šaman, Bohdan Drożdż and Miroslav Holub
Sesquiterpene lactones from Venidium hirsutum BEROL. species
1989, Vol. 54, Issue 7, pp. 1919–1927 [Abstract]
Ełżbieta Błoszyk, Aleksandra Dudek, Zofia Kosturkiewicz, Urszula Rychłewska, Włodzimierz M. Daniewski, Maria Gulumka, Jan Nawrot, Miloš Buděšínský, Soňa Vašíčková and Miroslav Holub
Sesquiterpene lactones of Cephalophora aromatica (HOOK.) SCHRADER and their deterrent activity. The stereostructure of geigerinin
1989, Vol. 54, Issue 7, pp. 1903–1918 [Abstract]
Martin Mandel, Ludvík Novák, Miroslav Rajšner, Jiří Holubek and Vladislava Holá
New synthesis of oxime-type beta-lactam antibiotics
1989, Vol. 54, Issue 6, pp. 1734–1745 [Abstract]
Vojtěch Kmoníček, Zdeněk Vejdělek, Jiří Holubek, Martin Valchář and Miroslav Protiva
Potential antidepressants: 1-(4-Aminoalkoxy)phenyl)-2-propylamines
1989, Vol. 54, Issue 6, pp. 1721–1733 [Abstract]
Vladimír Valenta, Marie Vlková and Miroslav Protiva
Potential neurotropic and antiinflammatory agents: 2-Chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yl sulfides
1989, Vol. 54, Issue 5, pp. 1403–1421 [Abstract]
Hana Hulinská, Miroslav Ryska, Ivan Koruna, Jiří Holubek, Jan Taimr, Emil Svátek and Miroslav Protiva
Some further 2-(4-substituted 1-piperazinyl)acetamides derived from 6,11-dihydrodibenzo[b,e]thiepin. Transformations of 6,11-dihydrodibenzo[b,e]thiepin derivatives into anthraquinones, anthrones and anthracenes
1989, Vol. 54, Issue 5, pp. 1388–1402 [Abstract]
Hana Hulinská, Miloš Buděšínský, Jiří Holubek, Oluše Matoušová, Hana Frycová and Miroslav Protiva
Reactions of N-substituted 2-aminopyridines with chloroacetyl chloride; Formation of a new series of heterocyclic betaines: 1-Substituted 4-chloromethyl-2-oxopyrido[1,2-a]pyrimidin-5-ium-3-olates
1989, Vol. 54, Issue 5, pp. 1376–1387 [Abstract]
Jan Sejbal, Eva Klinotová, Markéta Bludská, Jiří Klinot and Miloš Buděšínský
Conversion of betulin into careyagenolide (2α,3β-dihydroxy-18α,19βH-ursan-28,20β-olide)
1989, Vol. 54, Issue 4, pp. 1036–1042 [Abstract]
Jiří Protiva, Václav Křeček, Bohumil Máca, Jiří Urban, Miloš Buděšínský and Miloš Procházka
Synthesis of 4-(N-acetyl-L-tyrosyl)amino-2-iodobenzoic acid
1989, Vol. 54, Issue 4, pp. 1012–1018 [Abstract]
Miloš Buděšínský, Le Viet Ngoc Phuong, Nestor Perez Souto, Włodzimierz M. Daniewski, Andrzej Wawrzuń, Maria Gumułka, Soňa Vašíčková, David Šaman, Bohdan Drożdż, Halina Grabarczyk, Urszula Rychłewska and Miroslav Holub
Isolation and structures of sesquiterpene lactones: Aerial parts of Arctotis grandis THUNB. species
1989, Vol. 54, Issue 2, pp. 473–486 [Abstract]
Jiří Klinot, Jiří Liška, Alena Forgáčová, Miloš Buděšínský, Jiří Protiva, Stanislav Hilgard and Alois Vystrčil
Acid-catalyzed rearrangements of an A(1)-nor-triterpenoid 2α,3α-epoxide
1989, Vol. 54, Issue 2, pp. 413–429 [Abstract]
Zdeněk Polívka, Vladimír Valenta, Karel Šindelář, Jiří Holubek, Miloš Buděšínský, Miroslav Ryska, Ivan Koruna, Jitka Kohoutová, Jan Metyš, Jiřina Metyšová, Martin Valchář and Miroslav Protiva
Potential antidepressants: Saturated side chain amines derived from 6,11-dihydrodibenzo[b,e]thiepin and 4,9-dihydrothieno[2,3-c]-2-benzothiepin
1989, Vol. 54, Issue 1, pp. 235–247 [Abstract]
Karel Šindelář, Jiřina Metyšová and Miroslav Protiva
Potential antidepressants: 2-(6,11-Dihydrodibenzo[b,e]thiepin-11-yl)-4,5-dihydroimidazoles
1989, Vol. 54, Issue 1, pp. 229–234 [Abstract]
Irena Červená, Jiří Holubek, Emil Svátek, Jan Metyš, Martin Valchář and Miroslav Protiva
Potential antidepressants: Synthesis of two 4-(aminoalkoxy)dibenzo[b,e]thiepin-11(6H)-ones
1989, Vol. 54, Issue 1, pp. 225–228 [Abstract]
Miloš Buděšínský, David Šaman, Jan Pelnař, Soňa Vašíčková, Bohdan Drożdż, Halina Grabarczyk, Le Viet Ngoc Phuong and Miroslav Holub
Arctolide-revision of its stereostructure and determination of absolute configuration. Detailed ¹H and ¹³C NMR analysis
1989, Vol. 54, Issue 1, pp. 166–188 [Abstract]
Jan Ježek, Milan Zaoral, Miloš Buděšínský, Jiří Günther and Jiří Rotta
Muramyl-dipeptide analogues: Synthesis and biological activities
1988, Vol. 53, Issue 11, pp. 2897–2906 [Abstract]
Jiří Jílek, Martin Valchář, Jiří Holubek, Nataša Dlohožková, Josef Pomykáček, Oluše Matoušová, Jiřina Metyšová and Miroslav Protiva
Noncataleptic neuroleptic agents: 2-(4-(2-(2-Chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yloxy)ethyl)piperazine-1-yl)ethanol and some related compounds
1988, Vol. 53, Issue 11, pp. 2731–2741 [Abstract]
Zdena Koblicová, Jiří Holubek and Jan Trojánek
Synthesis of stereoisomeric vincamines
1988, Vol. 53, Issue 11, pp. 2722–2730 [Abstract]
Zdenko Procházka, Juris E. Ancans, Jiřina Slaninová, Alena Machová, Tomislav Barth, Jana Škopková, Miloš Buděšínský, Františka Pavlíková and Michal Lebl
Synthesis and properties of analogues of vasopressin with 1-aminocyclopropane-1-carboxylic acid in position 9
1988, Vol. 53, Issue 11, pp. 2604–2616 [Abstract]
Jan Hlaváček, Ivo Frič, Miloš Buděšínský and Karel Bláha
An alternative route to N^α-methylamino acid derivatives: Synthesis and conformation of some N^α-acetyl-N^α-methylamino acid methylamides
1988, Vol. 53, Issue 11, pp. 2473–2494 [Abstract]
Petr Maloň, C. L. Barness, Miloš Buděšínský, Rina K. Dukor, Dick Van der Helm, Timothy A. Keiderling, Zdena Koblicová, Františka Pavlíková, Miloš Tichý and Karel Bláha
(1S,7S)-7-Methyl-6,9-diazatricyclo[6,3,0,0^1,6]tridecane-5,10-dione, a tricyclic spirodilactam containing non-planar amide groups: Synthesis, NMR, crystal structure, absolute configuration, electronic and vibrational circular dichroism
1988, Vol. 53, Issue 11, pp. 2447–2472 [Abstract]
Miroslav Kuchař, Eva Maturová, Bohumila Brunová, Jaroslava Grimová, Hana Tomková and Jiří Holubek
Quantitative relations between structure and antiinflammatory activity of aryloxoalkanoic acids
1988, Vol. 53, Issue 8, pp. 1862–1872 [Abstract]
Hana Hulinská, Zdeněk Polívka, Jiří Jílek, Karel Šindelář, Jiří Holubek, Emil Svátek, Oluše Matoušová, Miloš Buděšínský, Hana Frycová and Miroslav Protiva
Experimental antiulcer agents: N-substituted 2-(4-methyl-1-piperazinyl)acetamides as pirenzepine models and some related compounds
1988, Vol. 53, Issue 8, pp. 1820–1844 [Abstract]
Zdeněk Polívka, Jan Metyš and Miroslav Protiva
6,11-Dihydrodibenzo[b,e]thiepin-11-yl 3-quinuclidinyl ethers: New potential intidepressants and antihistamine agents
1988, Vol. 53, Issue 8, pp. 1806–1811 [Abstract]
Václav Černý, Miloš Buděšínský, Miloš Ryba and František Tureček
A contribution to peroxy acid oxidation of α,β-unsaturated ketones and linearly conjugated dienones: Reactions in the cholestane series
1988, Vol. 53, Issue 7, pp. 1549–1567 [Abstract]
Irena Červená, Jiří Holubek, Emil Svátek and Miroslav Protiva
Potential antidepressants: 4-(Aminoalkoxy)thioxanthones
1988, Vol. 53, Issue 6, pp. 1307–1316 [Abstract]
Zdeněk Polívka, Jiřina Metyšová, Martin Valchář and Miroslav Protiva
Potential antidepressants: N-phenacyl derivatives of (E)-N-methyl-3-(6,11-dihydrodibenzo[b,e]thiepin-11-ylidene)propylamine
1988, Vol. 53, Issue 4, pp. 884–888 [Abstract]
Jiří Jílek, Jiří Holubek, Emil Svátek, Jan Metyš, Hana Frycová, Josef Pomykáček and Miroslav Protiva
Tricyclic analogues of the antiallergic agent oxatomide: 1-(3-(4-(10,11-Dihydro-5H-dibenzo[a,d]cycloheptene-5-yl)-1-piperazinyl)propyl)-1,3-dihydro-2H-benzimidazol-2-one and the related 6,11-dihydrodibenzo[b,e]thiepin, 4,9-dihydrothieno[2,3-c]-2-benzothiepin, and 10,11-dihydrodibenzo[b,f]thiepin derivatives
1988, Vol. 53, Issue 4, pp. 870–883 [Abstract]
Vladimír Valenta, Hana Hulinská, Jiří Holubek, Antonín Dlabač, Jan Metyš, Hana Frycová and Miroslav Protiva
N-substituted derivatives of 6,11-dihydrodibenzo[b,e]thiepin-11-amine and related compounds; Synthesis and pharmacological screening
1988, Vol. 53, Issue 4, pp. 860–869 [Abstract]
Karel Šindelář, Zdeněk Šedivý, Marta Hrubantová, Martin Valchář, Jiřina Metyšová and Miroslav Protiva
Synthesis of (2-(phenylthio)phenyl)acetamidines and related amidoximes as potential antidepressants
1988, Vol. 53, Issue 2, pp. 381–388 [Abstract]
Hana Hulinská, Petr Taufmann, Hana Frycová and Miroslav Protiva
1-Methyl-, 1-phenyl-, and 1-(2-(2-dimethylaminoethoxy)-phenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole and their 2-substituted derivatives: Synthesis and pharmacological screening
1988, Vol. 53, Issue 2, pp. 373–380 [Abstract]
Zdeněk Vejdělek, Jiří Holubek, Miloš Buděšínský, Miroslav Ryska, Emil Svátek and Miroslav Protiva
Reactions of 4-chloro-1-nitrobenzene with (3-chloro-4-methoxyphenyl)acetonitrile and (3,4-dimethoxyphenyl)acetonitrile; Synthesis of 8-chloro-1-methyl (and methylthiomethyl-6-(3,4-disubstituted phenyl)-4H-s-triazolo[4,3-a]-1,4-benzodiazepines
1988, Vol. 53, Issue 2, pp. 361–372 [Abstract]
Karel Šindelář, Jiří Holubek, Oluše Matoušová, Emil Svátek, Martin Valchář, Antonín Dlabač, Nataša Dlohožková, Marta Hrubantová and Miroslav Protiva
Aminoalkylidene and aminoalkyl derivatives of 6,11-dihydrodibenzo[b,e]thiepin-2- and -9-carbonitrile and 4,10-dihydrothieno[2,3-c]-1-benzothiepin-6-carbonitrile; Antidepressants with a new activity profile
1988, Vol. 53, Issue 2, pp. 340–360 [Abstract]
Vladimír Valenta, Jiří Holubek, Emil Svátek and Miroslav Protiva
Synthesis of 4-methoxyphenoxyacetic and 3,4,5-trimethoxyphenoxyacetic acid amides and hydrazides as potential neurotropic and cardiovascular agents
1987, Vol. 52, Issue 12, pp. 3013–3023 [Abstract]
Dalimil Dvořák, David Šaman, Miloš Buděšínský and Zdeněk Arnold
Arbuzov rearrangement in the reaction of arylmethylenemalonaldehydes with trimethyl phosphite: Formation of 2-(α-dimethoxyphosphonylbenzyl)-3-methoxyacroleins
1987, Vol. 52, Issue 12, pp. 2926–2935 [Abstract]
Zdeněk Polívka, Jiří Holubek, Miloš Buděšínský, Oluše Matoušová, Emil Svátek, Jan Metyš and Miroslav Protiva
Potential antihistamine agents: 4-(6,11-Dihydrodibenzo[b,e]thiepin-11-ylidene)-1-methyltetrahydrothiopyranium iodide and similar sulfonium salts derived from related tricyclic systems
1987, Vol. 52, Issue 11, pp. 2758–2774 [Abstract]
Irena Červená, Jiří Holubek, Emil Svátek, Martin Valchář and Miroslav Protiva
Potential antidepressants: 3-Methyl-6-dimethylamino-1,2-diphenylhexan-3-ol and related compounds
1987, Vol. 52, Issue 10, pp. 2564–2571 [Abstract]
Zdeněk Vejdělek, Jiří Holubek, Miroslav Ryska, Ivan Koruna, Emil Svátek, Miloš Buděšínský and Miroslav Protiva
Reactions of 4-chloro-1-nitrobenzene with o-substituted phenylacetonitriles; Synthesis of 8-chloro-1-methyl(and methylthiomethyl)-6-(2-substituted phenyl)-4H-s-triazolo[4,3-a]-1,4-benzodiazepines
1987, Vol. 52, Issue 10, pp. 2545–2563 [Abstract]
Vladimír Valenta, Jiří Holubek, Emil Svátek, Vladimír Miller, Marie Vlková and Miroslav Protiva
2-Diethylaminoethyl esters of 1,3-disubstituted propane-2-carboxylic acids
1987, Vol. 52, Issue 10, pp. 2534–2544 [Abstract]
Zdeněk Wimmer, Miloš Buděšínský, Tomáš Macek, Aleš Svatoš, David Šaman, Soňa Vašíčková and Miroslav Romaňuk
Biotransformation of 2-(4-methoxybenzyl)-1-cyclohexanone by means of Saccharomyces cerevisiae
1987, Vol. 52, Issue 9, pp. 2326–2337 [Abstract]
Karel Bláha, Miloš Buděšínský, Ivo Frič, Jan Pospíšek and Jindřich Symerský
Conformation of diastereoisomeric cyclo(neopentylglycyl-prolyls): NMR, X-ray, and CD studies
1987, Vol. 52, Issue 9, pp. 2295–2308 [Abstract]
Karel Šindelář, Miloš Buděšínský, Tomáš Vaněk, Jiří Holubek, Emil Svátek, Oluše Matoušová, Charles Wayne Rees and Miroslav Protiva
Reaction of 6,11-dihydrodibenzo[b,e]thiepin-11-carbonitrile with 1,2-dibromoethane, a reinvestigation. Formation of 11,12-dihydro-6H-6,12-methanodibenzo[b,f]thiocin-12-carbonitrile
1987, Vol. 52, Issue 9, pp. 2281–2294 [Abstract]
Vladimír Valenta and Miroslav Protiva
Potential neuroleptics of the orthopramide series; Synthesis of N-substituted 5-(aminosulfonyl)-2-methoxybenzamides
1987, Vol. 52, Issue 8, pp. 2095–2106 [Abstract]
Zdeněk Vejdělek and Miroslav Protiva
1-(4-Cyclopentylphenyl)piperazine and its 4-substituted derivatives; Synthesis and biological screening
1987, Vol. 52, Issue 7, pp. 1834–1840 [Abstract]
Miroslav Protiva, Jiří Jílek, Miroslav Rajšner, Karel Šindelář, Václav Bártl, Miroslav Ryska, Ivan Koruna, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Antonín Dlabač, Josef Pomykáček and František Mikšík
Fluorinated tricyclic neuroleptics with prolonged action: derivatives and analogues of 2-(4-(7-fluoro-2-isopropyl-10,11-dihydrodibenzo[b,f]thiepin-11-yl)-piperazine-1-yl)ethanol
1987, Vol. 52, Issue 7, pp. 1811–1833 [Abstract]
Ladislav Novotný, Miloš Buděšínský, Josef Jizba, Juraj Harmatha, Vít Lukeš, Wolfgang Lindner, Rolf Grosser and Günther Snatzke
Configuration of natural 9-hydroxyfuroeremophilane, its 9-hydroxy epimer and furanopetasin: NMR and CD studies
1987, Vol. 52, Issue 7, pp. 1786–1802 [Abstract]
Zdeněk Polívka, Irena Lichá, Petr Taufmann, Emil Svátek, Jiří Holubek and Miroslav Protiva
Synthesis of 3-(6,11-dihydrodibenzo[b,e]thiepin-11-ylidene)propanoic acid and related compounds
1987, Vol. 52, Issue 6, pp. 1566–1582 [Abstract]
Jiří Urban, Emil Svátek, Miroslav Ryska, Jan Metyš, Stanislav Wildt and Miroslav Protiva
4-Aryl-3-(dimethylaminomethyl)thiacyclohexan-4-ols including the thia analogue of tramadol; Synthesis and analgetic activity
1987, Vol. 52, Issue 5, pp. 1340–1351 [Abstract]
Zdeněk Vejdělek and Miroslav Protiva
4-Amino-1-(4-cyclopentylphenyl)butan-1-ones; Synthesis and biological screening
1987, Vol. 52, Issue 4, pp. 1073–1078 [Abstract]
Vladimír Valenta, Jiří Holubek and Miroslav Protiva
4-Substituted 1-(1-(2-(arylthio)-5-halogenophenyl)ethyl)piperazines; Synthesis and biological screening
1987, Vol. 52, Issue 4, pp. 1062–1072 [Abstract]
Vojtěch Kmoníček, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
2-(tert.amino)-11-(4-methylpiperazino)dibenzo[b,f]thiepins and their 10,11-dihydro derivatives; Synthesis and neuroleptic activity
1987, Vol. 52, Issue 3, pp. 793–803 [Abstract]
Silvio Cerrini, Doriano Lamba, Irena Valterová, Miloš Buděšínský, Jan Vrkoč and František Tureček
Methyl 3α,6α-diacetoxy-10-oxo-(7α)-kemp-11-en-20-oate: The revised structure for the kempane derivative from the frontal gland secretion of Nasutitermes costalis soldiers
1987, Vol. 52, Issue 3, pp. 707–713 [Abstract]
Miloš Buděšínský and David Šaman
Identification of acyl groups occurring in sesquiterpene lactones: Proton and carbon-13 NMR study
1987, Vol. 52, Issue 2, pp. 453–475 [Abstract]
Zdeněk Veselý, Jiří Holubek and Jan Trojánek
Reactions in the series of substituted isoindolo[1,2-b][3]-benzazepin-5-ones
1987, Vol. 52, Issue 1, pp. 233–241 [Abstract]
Miroslav Kuchař, Bohumila Brunová, Jaroslava Grimová, Stanislav Vaněček and Jiří Holubek
Synthesis of cyclohexylaliphatic acids and their pharmacological properties
1986, Vol. 51, Issue 12, pp. 2896–2908 [Abstract]
Irena Valterová, Soňa Vašíčková, Miloš Buděšínský and Jan Vrkoč
Constituents of frontal gland secretion of peruvian termites Nasutitermes ephratae
1986, Vol. 51, Issue 12, pp. 2884–2895 [Abstract]
Jiří Klinot, Jarmil Světlý, Eva Klinotová, Miloš Buděšínský and Alois Vystrčil
Preparation of isomeric 2-methyl-1-oxotriterpenoids of the 18α-oleanane series; Conformation of ring A
1986, Vol. 51, Issue 12, pp. 2869–2878 [Abstract]
Karel Šindelář, Jiří Holubek, Miroslav Ryska, Ivan Koruna and Miroslav Protiva
5-Substituted and 5,7-disubstituted 5,7-dihydrodibenzo[c,e]thiepins and the corresponding S-oxygenated compounds: Alkylamines, carboxylic acids, and carboxamides; synthesis and pharmacological screening
1986, Vol. 51, Issue 12, pp. 2848–2868 [Abstract]
Miroslav Protiva, Jiří Jílek, Irena Červená, Josef Pomykáček, Václav Bártl, Antonín Dlabač, Martin Valchář, Jiřina Metyšová, Jiří Holubek and Emil Svátek
Noncataleptic neuroleptic agents: 4-Substituted 1-(2-chloro-7-fluoro-10,11-dihydrodibenzo[b,f]thiepin-10-yl)piperazines and related compounds
1986, Vol. 51, Issue 11, pp. 2598–2616 [Abstract]
Ludvík Streinz, Irena Valterová, Zdeněk Wimmer, Miloš Buděšínský, David Šaman, Jitka Kohoutová, Miroslav Romaňuk and Jan Vrkoč
Direct esterification of α-methoxy-α-(trifluoromethyl)phenylacetic acid
1986, Vol. 51, Issue 10, pp. 2207–2213 [Abstract]
Zdeněk Polívka, Jan Metyš and Miroslav Protiva
Heterocyclic ethers derived from 6,11-dihydrodibenzo[b,e]thiepin-11-ols and 4,9-dihydrothieno[2,3-c]-2-benzothiepin-4-ol; A new series of potential antidepressants and antihistamine agents
1986, Vol. 51, Issue 9, pp. 2034–2049 [Abstract]
Włodzimierz M. Daniewski, Wojciech Kroszczyṅski, Ełżbieta Błoszyk, Bohdan Drożdż, Jan Nawrot, Urszula Rychłewska, Miloš Buděšínský and Miroslav Holub
Sesquiterpenoids from Dittrichia viscosa (L.) GREUTER. Their structure and deterrent activity
1986, Vol. 51, Issue 8, pp. 1710–1721 [Abstract]
Urszula Rychłewska, Derek J. Hodgson, Halina Grabarczyk, Bohdan Drożdż, Włodzimierz M. Daniewski, Wojciech Kroszczyṅski, Miloš Buděšínský and Miroslav Holub
Sesquiterpene lactones of Urospermum dalechampii SCHMIDT
1986, Vol. 51, Issue 8, pp. 1698–1709 [Abstract]
Jiří Jílek, Martin Valchář, Josef Pomykáček, Antonín Dlabač and Miroslav Protiva
Noncataleptic neuroleptic agents: Synthesis of some esters of 2-chloro-10-(4-(2-hydroxyethyl)piperazino)-10,11-dihydrodibenzo[b,f]thiepin
1986, Vol. 51, Issue 7, pp. 1503–1508 [Abstract]
Zdeněk Vejdělek and Miroslav Protiva
N-(piperazinoacyl) and N-(piperazinoalkyl) derivatives of 4-cyclopentylaniline and related compounds: Synthesis and pharmacological screening
1986, Vol. 51, Issue 7, pp. 1494–1502 [Abstract]
Zdeněk Vejdělek, Jiří Němec and Miroslav Protiva
Synthesis of N-(1-phenyl-2-propyl)-2,5-diphenylpentylamine and some related compounds as potential neurotropic and cardiovascular drugs
1986, Vol. 51, Issue 7, pp. 1487–1493 [Abstract]
Zdenka Smítalová, Miloš Buděšínský, David Šaman and Miroslav Holub
Minor sesquiterpenic lactones of Laser trilobum (L) BORKH. species
1986, Vol. 51, Issue 6, pp. 1323–1339 [Abstract]
Miloš Buděšínský, Antonín Trka, Karel Stránský and Milan Streibl
Heterocyclic nitrogen-containing compounds from the extract of the springtail Tetrodontophora bielanensis (WAGA)
1986, Vol. 51, Issue 4, pp. 956–963 [Abstract]
Karel Stránský, Antonín Trka, Miloš Buděšínský and Milan Streibl
Lipidic compounds from the extract of the springtail Tetrodontophora bielanensis (WAGA)
1986, Vol. 51, Issue 4, pp. 948–955 [Abstract]
Vojtěch Kmoníček, Emil Svátek, Jiří Holubek and Miroslav Protiva
Synthesis of potential neuroleptics and tranquillizers: 2-(tert.Amino)-9-(3-dimethylaminopropylidene)thioxanthenes
1986, Vol. 51, Issue 4, pp. 937–947 [Abstract]
Miroslav Holub, Miloš Buděšínský, Zdenka Smítalová, David Šaman and Urszula Rychłewska
Structure of isosilerolide, relative and absolute configuration of silerolide and lasolide - Sesquiterpenic lactones of new stereoisomeric type of eudesmanolides
1986, Vol. 51, Issue 4, pp. 903–929 [Abstract]
Miroslav Protiva, Jiří Jílek, Miroslav Rajšner, Josef Pomykáček, Miroslav Ryska, Jiří Holubek, Emil Svátek and Jiřina Metyšová
Fluorinated tricyclic neuroleptics with prolonged action: 7-Fluoro-11-[4-(2-hydroxyethyl)piperazino]-2-isopropyl-10,11-dihydrodibenzo[b,f]thiepin
1986, Vol. 51, Issue 3, pp. 698–722 [Abstract]
Václav Křeček, Jiří Protiva, Miloš Buděšínský, Eva Klinotová and Alois Vystrčil
Preparation of C₍₁₈₎-empiric 20,29,30-trinorlupane derivatives. ¹H, ¹³C NMR and mass spectra
1986, Vol. 51, Issue 3, pp. 621–635 [Abstract]
Jiří Klinot, Miloš Buděšínský, Eva Klinotová and Alois Vystrčil
Conformation of the A ring in 1-oxo and 3-oxotriterpenoids. Vicinal interproton coupling constants
1986, Vol. 51, Issue 3, pp. 593–610 [Abstract]
Alois Vystrčil, Václav Křeček, Miloš Buděšínský and Jiří Protiva
Isomeric oximes of 30-norlupan-20-one and its derivatives
1986, Vol. 51, Issue 3, pp. 581–592 [Abstract]
Miroslav Protiva, Antonín Dlabač, Martin Valchář, Stanislav Wildt, Irena Červená and Zdeněk Šedivý
Potential noncataleptic neuroleptic agents; 2,6-Dichloro-, 2,7-dichloro- and 2,8-dichloro-10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
1986, Vol. 51, Issue 1, pp. 156–166 [Abstract]
Irena Červená, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Martin Valchář, Antonín Dlabač, Stanislav Wildt and Miroslav Protiva
6-Substituted and 2-chloro-6-substituted 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins as potential antidepressants; Synthesis and pharmacology
1986, Vol. 51, Issue 1, pp. 141–155 [Abstract]
Urszula Rychłewska, Derek J. Hodgson, Miroslav Holub, Miloš Buděšínský and Zdenka Smítalová
The structure of 2-oxo-8α-angeloyloxy-11α-acetoxy-5βH,6αH,7αH-guai-1(10),3-dien-6,12-olide, a sesquiterpenic lactone from Laserpitium prutenicum L. revision of the stereostructures of native 2-oxoguai-1(10),3-dien-6,12-olides from the species of the Umbelliferae family
1985, Vol. 50, Issue 11, pp. 2607–2624 [Abstract]
Dalimil Dvořák, Miloš Buděšínský, David Šaman and Zdeněk Arnold
Benzylidenemalonaldehydes: A redox reaction during the attempted cycloaddition on nitrosobenzene
1985, Vol. 50, Issue 10, pp. 2260–2264 [Abstract]
Jiří Jílek, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Josef Pomykáček, Zdeněk Šedivý and Miroslav Protiva
Potential metabolites of the neuroleptic agents belonging to the 8-methylthio-10-piperazino-10,11-dihydrodibenzo[b,f]thiepin series; Synthesis of 2-hydroxy and 3-hydroxy derivatives
1985, Vol. 50, Issue 10, pp. 2179–2190 [Abstract]
Milena Masojídková, Jaroslav Zajíček, Miloš Buděšínský, Ivan Rosenberg and Antonín Holý
Conformational study on ribonucleoside O-phosphonylmethyl derivatives by ¹H NMR spectroscopy
1985, Vol. 50, Issue 8, pp. 1899–1905 [Abstract]
Miroslav Protiva, Zdeněk Šedivý, Jiří Holubek, Emil Svátek and Jiří Němec
Cyclic amidines derived from benz[c,d]indole and 4,5-dihydro-3H-1-benzazepine including some related compounds: Synthesis and pharmacological screening
1985, Vol. 50, Issue 8, pp. 1888–1898 [Abstract]
Miroslav Holub, Miloš Buděšínský, Zdenka Smítalová, David Šaman and Urszula Rychłewska
Structure of laserolide and isolaserolide: Revision of constitution and determination of relative and absolute configuration
1985, Vol. 50, Issue 8, pp. 1878–1887 [Abstract]
Zdeněk Vejdělek, Václav Bártl, Emil Svátek and Miroslav Protiva
Synthesis of several compounds related to 1-(4-methylsulfonylphenacyl)-4-phenylpiperazine and their pharmacological screening
1985, Vol. 50, Issue 7, pp. 1498–1506 [Abstract]
Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Martin Valchář and Miroslav Protiva
Butaclamol-like neuroleptic agents: Synthesis of 1-(11H-dibenz[b,f]-1,4-oxathiepin-11-yl)methyl-4-isobutylpiperidin-4-ol and of some related compounds
1985, Vol. 50, Issue 7, pp. 1484–1497 [Abstract]
Karel Šindelář, Jan Metyš and Miroslav Protiva
Potential antidiarrheal agents: 1-(11-Cyano-6,11-dihydrodibenzo[b,e]thiepin-11-yl-alkyl)- and 1-(10-cyano-10,11-dihydrodibenzo[b,f]thiepin-10-yl-alkyl)-4-substituted piperidines
1985, Vol. 50, Issue 5, pp. 1089–1096 [Abstract]
Zdeněk Polívka, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
Synthesis of the semi-rigid analogues of prothiadene and dithiadene as potential antidepressant and antihistamine agents: 11-[2-(Dimethylaminomethyl)cyclohexylidene]-6,11-dihydrodibenzo[b,e]thiepins and 4-[2-(dimethylaminomethyl)cyclohexylidene]-4,9-dihydrothieno-[2,3-c]-2-benzothiepins
1985, Vol. 50, Issue 5, pp. 1078–1088 [Abstract]
Vladimír Valenta, Zdeněk Prošek, Jiřina Metyšová, Martin Valchář, Antonín Dlabač and Miroslav Protiva
Cataleptic and noncataleptic neuroleptic agents: Synthesis and pharmacology of 4-(2-chloro and 8-chloro substituted 10,11-dihydrodibenzo[b,f]thiepin-10-yl)piperazine-1-ylalkyl ethers and sulfides
1985, Vol. 50, Issue 5, pp. 1070–1077 [Abstract]
Zdeněk Vejdělek, Zdeněk Polívka and Miroslav Protiva
Synthesis of 7-chloro-5-(4-chlorophenyl)-1-methyl-1,3-dihydro-1,4-benzodiazepin-2-one
1985, Vol. 50, Issue 5, pp. 1064–1069 [Abstract]
Jan Šmidrkal, Jiří Holubek and Jan Trojánek
The synthesis of 2,3,7,8-bismethylenedioxy-11-methoxy-5-methylbenzo[c]phenanthridinium chloride
1985, Vol. 50, Issue 4, pp. 984–990 [Abstract]
Jan Šmidrkal, Jiří Holubek, Jiří Šlanger and Jan Trojánek
Attempts at the synthesis of 11-methoxysubstituted benzo[c]phenantridines
1985, Vol. 50, Issue 4, pp. 861–868 [Abstract]
Jiří Jílek, Jiří Holubek, Emil Svátek, Jiří Schlanger, Josef Pomykáček and Miroslav Protiva
Highly polar potential metabolites of the neuroleptic agent oxyprothepin: Synthesis of 2-hydroxy-8-methylsulfonyl and 3-hydroxy-8-methylsulfonyl derivatives of 10-[4-(3-hydroxypropyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
1985, Vol. 50, Issue 2, pp. 519–537 [Abstract]
Vladimír Valenta and Miroslav Protiva
Synthesis of several 4-hydroxy-3,5-dimethoxybenzamides, their O-substituted derivatives and some related compounds as potential neurotropic agents
1985, Vol. 50, Issue 2, pp. 510–518 [Abstract]
Karel Šindelář, Jiří Holubek, Jiří Schlanger, Antonín Dlabač, Martin Valchář and Miroslav Protiva
Synthesis of spiro(piperidine-4,6'-dibenz[b,e]-1,4-oxathiepin) and its 1-methyl derivative as potential antidepressant agents
1985, Vol. 50, Issue 2, pp. 503–509 [Abstract]
Wojciech Kroszczyṅski, Włodzimierz M. Daniewski, Miloš Buděšínský, David Šaman, Halina Grabarczyk, Bohdan Drożdż and Miroslav Holub
Minor sesquiterpenic lactones from Ursinia anthemoides (L.) POIRET
1985, Vol. 50, Issue 1, pp. 94–102 [Abstract]
Karel Konečný, Milan Streibl, Soňa Vašíčková, Miloš Buděšínský, David Šaman, Karel Ubik and Vlastimil Herout
Constituents of the liverwort Bazzania trilobata of Czech origin
1985, Vol. 50, Issue 1, pp. 80–93 [Abstract]
Antonín Černý, Jiří Křepelka, Viktor Zikán, Drahuše Vlčková, Jaroslav Vachek, Jiří Holubek, Karel Řežábek, Maria Frühaufová, Miroslav Šeda, Jana Chlebounová and Otakar Marhan
Some 6-substituted 1-[(5R,8S,10R)-8-ergolinyl]-3,3-diethylureas
1984, Vol. 49, Issue 12, pp. 2828–2836 [Abstract]
Urszula Rychłewska, Miroslav Holub, Miloš Buděšínský and Zdenka Smítalová
Stereostructure of slovanolides: X-ray crystallography of the 3-oxo-4αH,8α-benzoyloxy-10β,11α-diacetoxyslovanolide
1984, Vol. 49, Issue 12, pp. 2790–2800 [Abstract]
Zdeněk Vejdělek, Jan Metyš, Jiří Holubek, Emil Svátek and Miroslav Protiva
Potential antiparkinsonic agents: Synthesis and pharmacology of some 4-fluoro-4'-halogen'benzhydryl 2-(N,N-disubstituted amino)ethyl ethers
1984, Vol. 49, Issue 11, pp. 2649–2660 [Abstract]
Jiří Jílek, Miroslav Rajšner, Jiřina Metyšová, Josef Pomykáček and Miroslav Protiva
Fluorinated tricyclic neuroleptics with prolonged action: 8-Alkyl derivatives of 3-fluoro-10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
1984, Vol. 49, Issue 11, pp. 2638–2648 [Abstract]
Karel Šindelář, Jiří Holubek, Miroslav Ryska, Antonín Dlabač, Martin Valchář, Jiřina Metyšová and Miroslav Protiva
Tricyclic compounds containing two chalcogen atoms in the central seven-membered rings as potential drugs: Synthesis of 3-chloro-6-(1-methyl-4-piperidyl)-6H-dibenz[b,e]-1,4-oxathiepin and 6-oxodibenz[b,e]-1,4-oxathiepin-2-acetic acid
1984, Vol. 49, Issue 11, pp. 2531–2540 [Abstract]
Václav Bártl, Karel Šindelář, Vladimír Valenta, Jiří Holubek, Emil Svátek, Jiří Schlanger, Antonín Dlabač, Jiřina Metyšová and Miroslav Protiva
Potential antipsychotic agents: 2-Chloro- and 2-methyl-11-(2-piperazinoethoxy)-6,11-dihydrodibenzo[b,e]thiepins and some related compounds; Synthesis and pharmacology
1984, Vol. 49, Issue 11, pp. 2520–2530 [Abstract]
Václav Bártl, Vojtěch Kmoníček, Zdeněk Šedivý, Emil Svátek, Jiří Protiva and Miroslav Protiva
Thioxanthene derivatives of pharmacological interest: 1,2,4-Trichloro and 2,4,5,6-tetrachloro derivatives of 9-(3-dimethylaminopropylidene)thioxanthene
1984, Vol. 49, Issue 10, pp. 2295–2308 [Abstract]
Irena Valterová, Miloš Buděšínský, František Tureček and Jan Vrkoč
Minor diterpene components of the defense secretion from the frontal gland of soldiers of the species Nasutitermes costalis (HOLMGREN)
1984, Vol. 49, Issue 9, pp. 2024–2039 [Abstract]
Václav Bártl, Emil Svátek, Antonín Dlabač, Stanislav Wildt and Miroslav Protiva
11-(3-[4-(2-Hydroxyethyl)piperazino]propylidene)-6,11-dihydrodibenzo[b,e]thiepin, its 2-chloro derivative and some related compounds as potential antipsychotic agents; Synthesis and pharmacology
1984, Vol. 49, Issue 8, pp. 1816–1826 [Abstract]
Václav Bártl, Jiří Jílek, Jiřina Metyšová, Martin Valchář, Antonín Dlabač, Stanislav Wildt and Miroslav Protiva
Neuroleptic 2-chloro-11-(2-piperazineethoxy)-10,11-dihydrodibenzo[b,f]thiepins: Synthesis and pharmacology
1984, Vol. 49, Issue 8, pp. 1810–1815 [Abstract]
Václav Bártl, Antonín Dlabač, Martin Valchář and Miroslav Protiva
11-(4-Piperidylidene)-6,11-dihydrodibenzo[b,e]thiepins as potential antipsychotic agents; Synthesis and pharmacology
1984, Vol. 49, Issue 8, pp. 1800–1809 [Abstract]
Vojtěch Kmoníček, Václav Bártl and Miroslav Protiva
Thioxanthene derivatives with neurotropic activity; synthesis of 9-(3-dimethylaminopropylidene)-2-(methylthiomethyl)thioxanthene and of some related compounds
1984, Vol. 49, Issue 7, pp. 1722–1730 [Abstract]
Miloš Buděšínský, Miroslav Holub, David Šaman, Zdenka Smítalová, Ayhan Ulubelen and Sevil Öksüz
Structure of istanbulin A and istanbulin B - two sesquiterpenic lactones from Smyrnium olusatrum L.
1984, Vol. 49, Issue 5, pp. 1311–1317 [Abstract]
Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Antonín Dlabač, Martin Valchář and Miroslav Protiva
Analogues of the neuroleptic agent isobutaclamol: Stereoisomeric 3b,4,5,6,7,9,9a,10-octahydro-[1]benzothiepino[2,3,4-ed]pyrido[2,1-a]isoquinolin-5-ols and some related compounds
1984, Vol. 49, Issue 4, pp. 1021–1038 [Abstract]
Irena Červená and Miroslav Protiva
1-[2-(2-Hydroxymethylphenylthio)benzyl]-4-methylpiperzine and related compounds as potential antidepressants: Synthesis and pharmacological acreening
1984, Vol. 49, Issue 4, pp. 1009–1020 [Abstract]
Vladimír Valenta, Antonín Dlabač, Martin Valchář and Miroslav Protiva
α-Benzyldopamine and some related compounds: Synthesis and pharmacological screening
1984, Vol. 49, Issue 4, pp. 1002–1008 [Abstract]
Jiří Urban, Antonín Dlabač, Martin Valchář and Miroslav Protiva
Potential noncataleptic neuroleptic agents: 2,3-Dichloro-10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrobenzo[b,f]thiepin
1984, Vol. 49, Issue 4, pp. 992–1001 [Abstract]
Ivan Černý, Vladimír Pouzar, Pavel Drašar, Miloš Buděšínský and Miroslav Havel
Glucosylation of 5-androsten-3β-ol derivatives containing butenolide, furan or unsaturated ester moieties in the side chain
1984, Vol. 49, Issue 4, pp. 881–891 [Abstract]
Zdenka Smítalová, Miloš Buděšínský, David Šaman, Soňa Vašíčková and Miroslav Holub
Components of the extract from the underground parts of Laserpitium siler L. of slovenian origin, mainly sesquiterpenic lactones
1984, Vol. 49, Issue 4, pp. 852–870 [Abstract]
Karel Bláha, Ahmed M. Farag, Dick VAN DER Helm, M. Bilayet Hossain, Miloš Buděšínský, Petr Maloň, Jorga Smolíková and Miloš Tichý
Stereoisomeric chiral 2,9-diazabicyclo[4.4.0.]decane-3,10-diones as models of dipeptide grouping: Synthesis, X-ray, IR, NMR and cd studies
1984, Vol. 49, Issue 3, pp. 712–742 [Abstract]
Zdenko Procházka, Michal Lebl, Tomislav Barth, Jan Hlaváček, Antonín Trka, Miloš Buděšínský and Karel Jošt
Synthesis and properties of oxytocin analogues modified in the tripeptide side chain
1984, Vol. 49, Issue 3, pp. 642–652 [Abstract]
Miloš Buděšínský, David Šaman, Gerard Nowak, Bohdan Drożdż and Miroslav Holub
9α-Hydroxyparthenolide from Zoegea baldschuanica C. WINKL. and its absolute configuration
1984, Vol. 49, Issue 3, pp. 637–641 [Abstract]
Zdeněk Polívka, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
Potential hypnotics and anxiolytics: Synthesis of 2-bromo-4-(2-chlorophenyl)-9-[4-(2-methoxyethyl)piperazino]-6H-thieno[3,2,4-triazolo[4,3-a]-1,4-diazepine and of some related compounds
1984, Vol. 49, Issue 3, pp. 621–636 [Abstract]
Jiří Jílek, Josef Pomykáček, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiří Protiva and Miroslav Protiva
Reactions of 4,4'-disubstituted diphenyl sulfides with chloroacetyl chloride and aluminium chloride
1984, Vol. 49, Issue 3, pp. 603–620 [Abstract]
Miloš Tichý, Ahmed Farag, Miloš Buděšínský, Ludmila P. Otroshchenko, Tatjana A. Shibanova and Karel Bláha
Isomeric oxatricyclodecanones with non-planar lactone groups: Synthesis, absolute configuration, NMR and X-ray study
1984, Vol. 49, Issue 2, pp. 513–532 [Abstract]
Miloš Buděšínský, Miloslav Černý, Jitka Doležalová, Miloš Kulhánek, Josef Pacák and Milan Tadra
4-Deoxy-4-fluoro-D-fructose: Preparation and structure
1984, Vol. 49, Issue 1, pp. 267–274 [Abstract]
Jaroslav Zajíček, Miloš Buděšínský and Jiří Farkaš
Conformational study of blocked pentofuranoses and their 1,5-anhydro derivatives by ¹H NMR spectroscopy
1984, Vol. 49, Issue 1, pp. 235–243 [Abstract]
Miroslav Kuchař, Bohumila Brunová, Václav Rejholc, Magda Jelínková, Jiří Holubek and Oldřich Němeček
Quantitative relations between structure and activation of fibrinolysis in selected series of arylaliphatic acids
1984, Vol. 49, Issue 1, pp. 122–136 [Abstract]
Zdeněk Polívka, Jiří Jílek, Jiří Holubek, Emil Svátek, Antonín Dlabač, Martin Valchář and Miroslav Protiva
Noncataleptic neuroleptic agents: 2-Halogeno-8-isopropyl-10-piperazino-10,11-dihydrodibenzo[b,f,]thiepins
1984, Vol. 49, Issue 1, pp. 86–109 [Abstract]
Zdeněk Polívka, Jiří Holubek, Jan Metyš, Zdeněk Šedivý and Miroslav Protiva
Potential hypnotics and anxiolytics: 8-Chloro-6-(2-chlorophenyl)-1-[4-(2-methoxyethyl)piperazino]-methyl-4H-s-triazolo[4,3-a]-1,4-benzodiazepine and related compounds
1983, Vol. 48, Issue 12, pp. 3433–3443 [Abstract]
Zdeněk Vejdělek and Miroslav Protiva
Potential antitussives: Synthesis and pharmacology of a series of 1-[2-amino-2-(4-fluorophenyl)ethyl]-4-(2-benzoylpropyl)piperazines
1983, Vol. 48, Issue 10, pp. 2977–2988 [Abstract]
Zdeněk Polívka, Martin Valchář and Miroslav Protiva
Potential noncataleptic neuroleptic agents: Synthesis and pharmacology of 7-chloro-4-[4-(2-hydroxyethyl)piperazino]-4,5-dihydrothieno[2,3-b]-1-benzothiepin
1983, Vol. 48, Issue 10, pp. 2970–2976 [Abstract]
Petr Maloň, Petr Pančoška, Miloš Buděšínský, Jan Hlaváček, Jan Pospíšek and Karel Bláha
Chiroptical properties and conformation of N-acetyl-L-amino acids N'-methylamides with aliphatic side chains
1983, Vol. 48, Issue 10, pp. 2844–2861 [Abstract]
Miloslav Černý, Jitka Doležalová, Jindra Mácová, Josef Pacák, Tomáš Trnka and Miloš Buděšínský
Preparation of 3-deoxy-3-fluoro-D-mannose and corresponding hexitol
1983, Vol. 48, Issue 9, pp. 2693–2700 [Abstract]
Zdeněk Polívka, Miroslav Ryska, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
Potential hypnotics and anxiolytics in the 4H-s-triazolo[4,3-a]-1,4-benzodiazepine series: 8-Chloro-6-(2-chlorophenyl)-1-[4-(2-methoxyethyl)piperazino]-4H-s-triazolo[4,3-a]-1,4-benzodiazepine and some related compounds
1983, Vol. 48, Issue 8, pp. 2395–2410 [Abstract]
Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Jiří Urban and Miroslav Protiva
11-(Dimethylaminoalkyl)-6,11-dihydrodibenzo[b,e]thiepin-11-carbonitriles and some related compounds
1983, Vol. 48, Issue 7, pp. 1898–1909 [Abstract]
Alois Vystrčil, Václav Křeček and Miloš Buděšínský
Elimination reaction of angular hydroxymethyl groups of 20(29)-lupene derivatives
1983, Vol. 48, Issue 5, pp. 1499–1507 [Abstract]
Antonín Černý, Viktor Zikán, Drahuše Vlčková, Jan Beneš, Jiří Holubek, Karel Řežábek, Marie Aušková and Jiří Křepelka
(5R,8S,10R)-6-Alkyl-8-ergolinecarboxylic acids and some of their derivatives
1983, Vol. 48, Issue 5, pp. 1483–1488 [Abstract]
Zdeněk Vejdělek and Miroslav Protiva
Synthesis of two 1-substituted 8-bromo-6-(2-chlorophenyl)-4H-s-triazolo[4,3-a]-1,4-benzodiazepines
1983, Vol. 48, Issue 5, pp. 1477–1482 [Abstract]
Zdeněk Polívka, Jiří Holubek, Emil Svátek, Antonín Dlabač, Dušan Půček, Zdeněk Šedivý and Miroslav Protiva
3-(4-Methylpiperazino)dibenzo[b,f]-1,2,4-triazolo[4,3-d]-1,4-thiazepine and its 6-chloro and 12-chloro derivatives; Synthesis and pharmacology
1983, Vol. 48, Issue 5, pp. 1465–1476 [Abstract]
Vladimír Valenta, Jiří Holubek, Emil Svátek, Antonín Dlabač, Marie Bartošová and Miroslav Protiva
α-(4-Tolyl)dopamine, derivatives and analogues; Synthesis and pharmacological screening
1983, Vol. 48, Issue 5, pp. 1447–1464 [Abstract]
Jiří Křepelka, Vladimír Pouzar, Jiří Schlanger, Jiří Holubek, Jiří Körbl, Fedir Jančik and Rudolf Kotva
Oxidative transformations of some pyrimidine derivatives into oxazolidine derivatives
1983, Vol. 48, Issue 4, pp. 1212–1223 [Abstract]
Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Jiří Urban, Jaroslava Grimová, Irena Červená, Marta Hrubantová and Miroslav Protiva
Dibenzo[b,f]thiepin-10-carbonitrile, its 10,11-dihydro derivative, some transformation products and related compounds
1983, Vol. 48, Issue 4, pp. 1187–1211 [Abstract]
Václav Bártl, Jiří Holubek, Emil Svátek, Marie Bartošová and Miroslav Protiva
Potential anticonvulsants: Substituted N-benzylidene derivatives of 10-(4-aminopiperazino)-10,11-dihydrodibenzo[b,f]thiepins
1983, Vol. 48, Issue 4, pp. 1173–1186 [Abstract]
Vladimír Valenta, Jiří Němec and Miroslav Protiva
Basic amides of 2,4,5-trichlorophenoxyacetic, 2,4,6-trimethylphenoxyacetic and 4-bromo-3,5-dimethylphenoxyacetic acid and some related compounds; Synthesis and pharmacological screening
1983, Vol. 48, Issue 4, pp. 1089–1096 [Abstract]
Miroslav Kuchař, Václav Rejholec, Zdeněk Roubal and Oluše Matoušová
The effects of lipophilicity on the inhibition of denaturation of serum albumin and on the activation of fibrinolysis observed with a series of benzyloxyarylaliphatic acids
1983, Vol. 48, Issue 4, pp. 1077–1088 [Abstract]
Jiří Jílek, Josef Pomykáček, Zdeněk Prošek, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Antonín Dlabač and Miroslav Protiva
8-Chloro and 8-methylthio derivatives of 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins; New compounds and new procedures
1983, Vol. 48, Issue 3, pp. 906–927 [Abstract]
Zdeněk Vejdělek and Miroslav Protiva
N-substituted aminomethyl 4-cyclopentylphenyl ketones and 2-amino-1-(4-cyclopentylphenyl)ethanol: Synthesis and pharmacological screening
1983, Vol. 48, Issue 2, pp. 642–648 [Abstract]
Zdeněk Polívka, Miroslav Rajšner, Jan Metyš, Jiří Holubek, Emil Svátek, Miroslav Ryska and Miroslav Protiva
Antiaminic agents derived from thieno[2,3-c]-2-benzothiepin: 4-(1-Methyl-4-piperidylidene)-4,9-dihydrothieno[2,3-c]-2-benzothiepin and some related compounds
1983, Vol. 48, Issue 2, pp. 623–641 [Abstract]
Jiří Křepelka, Drahuše Vlčková, Jiří Holubek and Jiří Roubík
8-Substitution derivatives of D-6-methylergoline-I
1983, Vol. 48, Issue 1, pp. 312–318 [Abstract]
Jiří Křepelka, Jan Beneš, Vladimír Pouzar, Jaroslav Vachek and Jiří Holubek
Some 2-substitution derivatives of 5-(4-oxo-6-hydroxy-3,4-dihydro-5-pyrimidinyl)pentanoic acid
1983, Vol. 48, Issue 1, pp. 304–311 [Abstract]
Miroslav Rajšner, Jan Metyš, Jiří Holubek and Miroslav Protiva
Potential antidepressants: Some N-substituted derivatives of (E)-11-(3-methylaminopropylidene)-6,11-dihydrodibenzo[b,e]thiepin
1983, Vol. 48, Issue 1, pp. 163–172 [Abstract]
Zdeněk Vejdělek, Marie Bartošová and Miroslav Protiva
N-(Aminoacyl) and N-(aminoalkyl) derivatives of 4-cyclopentylaniline and N-ethyl-4-cyclopentylaniline; Synthesis and pharmacological screening
1983, Vol. 48, Issue 1, pp. 156–162 [Abstract]
Karel Šindelář, Jiřina Metyšová, Jiří Holubek, Emil Svátek, Miroslav Ryska and Miroslav Protiva
Fluorinated tricyclic neuroleptics with prolonged action: 3-Fluoro-10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepins with less common substituents in position 8
1983, Vol. 48, Issue 1, pp. 144–155 [Abstract]
Zdeněk J. Vejdělek, Jan Metyš and Miroslav Protiva
S-Substituted derivatives of 8-chloro-6-(2-chlorophenyl)-1-mercaptomethyl-4H-s-triazolo[4,3-a]-1,4-benzodiazepine; Synthesis and pharmacology
1983, Vol. 48, Issue 1, pp. 123–136 [Abstract]
Zdeněk Vejdělek, Jiří Holubek, Marie Bartošová and Miroslav Protiva
4-(Aminoacylamido)-s-hydrindacenes and related compounds: Synthesis and pharmacological screening
1982, Vol. 47, Issue 12, pp. 3297–3305 [Abstract]
Miroslav Protiva, Zdeněk Šedivý, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Marie Bartošová
Potential psychotropic and antihistamine agents: 1- and 3-alkyl-9-(3-dimethylaminopropylidene)-thioxanthenes and 3-alkyl-11-piperazino-10,11-dihydrodibenzo[b,f]thiepins
1982, Vol. 47, Issue 11, pp. 3134–3147 [Abstract]
Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Antonín Dlabač, Jiřina Metyšová and Miroslav Protiva
Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: 2-Fluoro-8-substituted 6-(4-piperidyl)-6H-dibenz[b,e]-1,4-oxathiepins
1982, Vol. 47, Issue 11, pp. 3114–3133 [Abstract]
Miroslav Protiva, Karel Šindelář, Vladimír Valenta, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiří Schlanger, Jiří Urban and Marta Hrubantová
Reactions of 11-chloro-11-phenyl-6,11-dihydrodibenzo[b,e]-thiepin with piperidine and some further nucleophiles
1982, Vol. 47, Issue 11, pp. 3094–3113 [Abstract]
Karel Šindelář, Jiřina Metyšová, Jiří Holubek, Emil Svátek, Jiří Protiva and Miroslav Protiva
Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: 8-Substituted 6-(4-piperidyl)-6H-dibenz[b,e]-1,4-oxathiepins
1982, Vol. 47, Issue 11, pp. 3077–3093 [Abstract]
Miroslav Holub, Zdeněk Samek, Miloš Buděšínský, David Šaman, Ełżbieta Błoszyk and Bohdan Drożdż
8α-Hydroxybalchanin - A new sesquiterpenic lactone from Leucanthemella serotina (L.) TZVEL.
1982, Vol. 47, Issue 11, pp. 2927–2931 [Abstract]
Patricia Sierra, Ladislav Novotný, Zdeněk Samek, Miloš Buděšínský, Ladislav Dolejš and Karel Bláha
Alkaloids of Rauvolfia salicifolia GRISEB species
1982, Vol. 47, Issue 11, pp. 2912–2921 [Abstract]
Miloš Buděšínský, David Šaman and Zdeněk Wimmer
Conformation studies of isomeric 1-acyloxy-2-(4-methoxybenzyl)-cyclohexanes by ¹H NMR spectroscopy
1982, Vol. 47, Issue 10, pp. 2763–2767 [Abstract]
Josef Hájíček, Jiří Holubek and Jan Trojánek
Synthesis of 4,4- and 5,5-disubstituted 4,5-dihydro-6H-canthin-6-ones
1982, Vol. 47, Issue 10, pp. 2749–2762 [Abstract]
Miroslav Kuchař, Václav Rejholec, Bohumila Brunová, Jaroslava Grimová, Oluše Matoušová, Oldřich Němeček and Hana Čepeláková
Benzyloxyarylaliphatic acids: Synthesis and quantitative relations between structure and antiinflammatory activity
1982, Vol. 47, Issue 9, pp. 2514–2524 [Abstract]
Zdenko Procházka, Miloš Buděšínský, Jorga Smolíková, Petr Trška and Karel Jošt
1-Aminocyclopropanecarboxylic acid and its derivatives
1982, Vol. 47, Issue 8, pp. 2291–2305 [Abstract]
Zdeněk Buděšínský, František Šmejkal and Miloš Buděšínský
Some 1-β-D-ribofuranosyl-5-phenylcytosines and -5-(2-chlorophenyl)-2-thiocytosine
1982, Vol. 47, Issue 8, pp. 2145–2149 [Abstract]
Ivan Beneš, Tomáš Vaněk and Miloš Buděšínský
Nardiin, a new ent-kaurane diterpenoid from the liverwort Nardia scalaris
1982, Vol. 47, Issue 7, pp. 1873–1877 [Abstract]
Jiří Křepelka, Iva Vančurová, Jiří Holubek, Milan Mělka and Karel Řežábek
Derivatives of benzo(c)fluorene: II. Synthesis and biological effect of basic ethers of 7-oxo-7H-benzo(c)fluorene
1982, Vol. 47, Issue 7, pp. 1856–1866 [Abstract]
Jan Beneš and Jiří Holubek
1,2-Fused derivatives of ergoline
1982, Vol. 47, Issue 6, pp. 1641–1644 [Abstract]
Jan Beneš and Jiří Holubek
Wittig type reactions of 2-formylated derivatives of 6-methylergoline - I
1982, Vol. 47, Issue 6, pp. 1636–1640 [Abstract]
Jiří Jílek, Josef Pomykáček, Jiřina Metyšová and Miroslav Protiva
Fluorinated tricyclic neuroleptics with prolonged action: 8-Methoxy, 8-ethoxy, 8-ethylthio and 8-hydroxy derivatives of 3-fluoro-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1982, Vol. 47, Issue 5, pp. 1382–1391 [Abstract]
Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Antonín Dlabač and Miroslav Protiva
Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: Synthesis of 6-(aminoalkyl) derivatives of 6H-dibenz[b,e]-1,4-oxathiepin
1982, Vol. 47, Issue 5, pp. 1367–1381 [Abstract]
Jiří Křepelka, Jiří Roubík, Jiří Holubek and Iva Vančurová
5-, 6- And 7-substitution derivatives of 7-oxo-7H-benzo(c)fluorene
1982, Vol. 47, Issue 4, pp. 1258–1266 [Abstract]
Jiří Křepelka, Iva Vančurová and Jiří Holubek
Reactions of 4-aryl-1-methoxynaphtalene-2,3-dicarboxylic acid anhydrides and naphtho(2,3-c)furan-1-(3H)-one derivatives with hydrazines
1982, Vol. 47, Issue 4, pp. 1252–1257 [Abstract]
Karel Bláha, Miloš Buděšínský, Zdena Koblicová, Petr Maloň, Miloš Tichý, J. R. Baker, M. B. Hossain and Dick Van der Helm
Optically active tricyclic dilactams with non-planar cis-amide groups: Synthesis, X-ray, NMR and CD studies
1982, Vol. 47, Issue 3, pp. 1000–1019 [Abstract]
Vladimír Valenta, Jan Metyš and Miroslav Protiva
(6,11-Dihydrodibenzo[b,e]thiepin-11-yl)methylamine, (4-methoxy-6,11-dihydrodibenzo[b,e]thiepin-11-yl)-methylamine and derivatives; Synthesis and pharmacological screening
1982, Vol. 47, Issue 3, pp. 984–993 [Abstract]
Karel Šindelář, Jiří Holubek, Miroslav Ryska, Antonín Dlabač, Jiřina Metyšová, Emil Svátek, Marta Hrubantová, Jiří Protiva and Miroslav Protiva
Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: Derivatives of 11H-dibenz[b,f]-1,4-oxathiepin
1982, Vol. 47, Issue 3, pp. 967–983 [Abstract]
Miroslav Holub, Miloš Buděšínský, Zdeněk Samek, Bohdan Drożdż, Halina Grabarczyk, Ayhan Ulubelen, Sevil Öksüz and Urszula Rychłewska
Absolute configuration of xerantholide, a sesquiterpenic lactone from Anthemis austriaca JACQ.
1982, Vol. 47, Issue 2, pp. 670–675 [Abstract]
Josef Jizba, Miloš Buděšínský, Tomáš Vaněk, A. Boeva, Kalinka Dimitrova, František Šantavý and Ladislav Novotný
Components of Senecio pancicii DEGEN var. arnautorum (VELEN.) STOJ., STEF. et KIT. and S. Pancicii DEGEN var. pancicii
1982, Vol. 47, Issue 2, pp. 664–669 [Abstract]
Juraj Harmatha, Miloš Buděšínský and Antonín Trka
The structure of yatein. Determination of the positions, and configurations of benzyl groups in lignans of the 2,3-dibenzylbutyrolactone type
1982, Vol. 47, Issue 2, pp. 644–663 [Abstract]
Miroslav Protiva, Zdeňka Kopicová and Jaroslava Grimová
Synthesis of several 1-(aminoacyl)-4-cinnamylpiperazines as potential analgetics
1982, Vol. 47, Issue 2, pp. 636–643 [Abstract]
Jiří Křepelka, Iva Vančurová, Jiří Holubek, Jiří Roubík and Drahuše Vlčková
Syntheses and antineoplastic effects of some N-substituted imides of 1-substituted 4-aryl-naphthalene-2,3-dicarboxylic acids
1982, Vol. 47, Issue 1, pp. 304–314 [Abstract]
Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Antonín Dlabač, Marta Hrubantová and Miroslav Protiva
Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: Synthesis of 11-(dimethylaminoalkyl) derivatives of 11H-dibenzo[b,e]-1,4-dioxepin and 11H-dibenzo[b,e]-1,4-dithiepin
1982, Vol. 47, Issue 1, pp. 72–87 [Abstract]
Miroslav Rajšner, Emil Svátek, Jan Metyš and Miroslav Protiva
Antidepressant fluorinated prothiadene derivatives: 9-Fluoro and 2,9-difluoro derivative of 11-(3-dimethylaminopropylidene)-6,11-dihydrodibenzo[b,e]thiepin
1982, Vol. 47, Issue 1, pp. 65–71 [Abstract]
Bohumír Koutek, Libuše Pavlíčková, Miloš Buděšínský and Milan Souček
Synthesis and properties of benzoannelated 6-(1,3-dithiolan-2-yliden)-2,4-cyclohexadien-1-ones
1982, Vol. 47, Issue 1, pp. 59–64 [Abstract]
Jiří Jílek, Josef Pomykáček, Jiří Němec and Miroslav Protiva
1-(3-Dimethylamino-1-phenylpropyl)piperazines and related compounds: Synthesis and pharmacological screening
1981, Vol. 46, Issue 11, pp. 2729–2733 [Abstract]
Zdeněk Buděšínský, Miloš Buděšínský and Alois Šváb
Addition of 2-methylthio-5-pyrimidinol and 5-methoxy-2-pyrimidinethiol to the acetylene triple bond
1981, Vol. 46, Issue 9, pp. 2254–2262 [Abstract]
Miroslav Protiva, Zdeněk Šedivý, Josef Pomykáček, Václav Bártl, Jiří Holubek and Emil Svátek
Potential metabolites of the noncataleptic neuroleptics: Synthesis of 2-chloro-6-hydroxy(and methoxy)-10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
1981, Vol. 46, Issue 9, pp. 2245–2253 [Abstract]
Zdeněk Vejdělek, Jiří Holubek, Marie Bartošová and Miroslav Protiva
1-(4-Cyclopentylphenyl)ethylamine and derivatives: Synthesis and pharmacological screening
1981, Vol. 46, Issue 9, pp. 2234–2244 [Abstract]
Zdeněk Polívka, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
Fluorinated tricyclic neuroleptics: Synthesis and pharmacology of 2-chloro-8-fluoro-4-(4-methylpiperazino)-4,5-dihydrothieno[2,3-b]-1-benzothiepin
1981, Vol. 46, Issue 9, pp. 2222–2233 [Abstract]
Jiří Křepelka, Iva Vančurová, Jiří Holubek and Jiří Roubík
Hydrolytic products of 4-aryl-2,3-dicyano-1-naphthol derivatives
1981, Vol. 46, Issue 9, pp. 2207–2216 [Abstract]
Jiří Křepelka and Jiří Holubek
The synthesis of model lactones of cyclolignan type
1981, Vol. 46, Issue 9, pp. 2123–2128 [Abstract]
Jiří Křepelka, Jiří Roubík and Jiří Holubek
1-Substitution derivatives of 4-aryl-2,3-dibromo-1-naphthol
1981, Vol. 46, Issue 9, pp. 2116–2122 [Abstract]
Miroslav Protiva, Karel Šindelář, Zdeněk Šedivý, Jiří Holubek and Marie Bartošová
Potential metabolites of tricyclic neuroleptics: 3,7-Dimethoxy and 7,8-dimethoxy derivatives of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1981, Vol. 46, Issue 8, pp. 1808–1817 [Abstract]
Zdeněk Vejdělek, Marie Bartošová and Miroslav Protiva
3-(s-Hydrindacen-4-yl)propylamines and 4-(s-hydrindacen-4-yl)butylamines; Synthesis and pharmacological screening
1981, Vol. 46, Issue 8, pp. 1800–1807 [Abstract]
Miroslav Protiva, Karel Šindelář, Jiřina Metyšová, Jiří Holubek, Miroslav Ryska, Emil Svátek, Zdeněk Šedivý and Josef Pomykáček
Fluorinated tricyclic neuroleptics with prolonged action: 3-Fluoro-8-halogeno derivatives of 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
1981, Vol. 46, Issue 8, pp. 1788–1799 [Abstract]
Jiří Jílek, Josef Pomykáček, Jiřina Metyšová and Miroslav Protiva
Neuroleptic agents derived from perathiepin: 6,7-Dichloro derivative of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin and related compounds
1981, Vol. 46, Issue 7, pp. 1607–1613 [Abstract]
Miroslav Rajšner, Antonín Dlabač and Miroslav Protiva
Esters of 1-[4,4-bis(4-fluorophenyl)butyl]-4-(4-chloro-3-trifluoromethylphenyl)-4-piperidinol
1981, Vol. 46, Issue 6, pp. 1530–1533 [Abstract]
Jiří Křepelka, Iva Vančurová and Jiří Holubek
Some derivatives of 4-aryl-2,3-dicyano-1-naphthol
1981, Vol. 46, Issue 6, pp. 1523–1529 [Abstract]
Vladimír Valenta, Marie Bartošová and Miroslav Protiva
1-[3-(2-Alkoxyphenoxy)-3-phenylpropyl]piperazines and some related compounds
1981, Vol. 46, Issue 5, pp. 1280–1287 [Abstract]
Miroslav Protiva, Zdeněk Šedivý, Josef Pomykáček, Emil Svátek and Jiří Holubek
Potential metabolites of the neuroleptic agent octoclothepin; Synthesis of 8-chloro-2,6-dihydroxy and 8-chloro-3,6-dihydroxy derivatives of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1981, Vol. 46, Issue 5, pp. 1199–1209 [Abstract]
Irena Červená, Marta Hrubantová, Marie Bartošová and Miroslav Protiva
Synthesis of arylthioacetamidoximes as potential antidepressants
1981, Vol. 46, Issue 5, pp. 1188–1198 [Abstract]
Vladimír Valenta, Antonín Dlabač and Miroslav Protiva
Potential noncataleptic neuroleptic agents: 2,4-Dichloro- and 2,4,8-trichloro-10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
1981, Vol. 46, Issue 3, pp. 781–791 [Abstract]
Ladislav Kniežo, Pavol Kristian, Miloš Buděšínský and Katarína Havrilová
Stereochemical course of the reaction of 2-haloethyl isothiocyanates with nucleophiles. Stereospecific route to 4,5-disubstituted Δ²-thiazolines and thiazolidine-2-thiones
1981, Vol. 46, Issue 3, pp. 717–728 [Abstract]
Karel Šindelář, Jiří Holubek, Jan Metyš, Marie Bartošová and Miroslav Protiva
Synthesis of 3-(2-alkoxyphenoxy)-2-methyl (or phenyl)propylamines as potential antidepressants
1981, Vol. 46, Issue 3, pp. 597–606 [Abstract]
Zdeněk Vejdělek, Emil Svátek, Jiří Holubek, Jan Metyš, Marie Bartošová and Miroslav Protiva
Synthesis and pharmacological screening of 1-[2-tert-aminoethyl]-8-fluoro-5-[4-fluorophenyl]-2,3,4,5-tetrahydro-1H-1-benzazepines, their 1-[aminoacetyl] analogues and 1-substituted 9-fluoro-6-[4-fluorophenyl]-5,6-dihydro-4H-s-triazolo[4,3-a]-1-benzazepines
1981, Vol. 46, Issue 1, pp. 148–160 [Abstract]
Václav Bártl, Jiřina Metyšová and Miroslav Protiva
2-Chloro-7-fluoro- and 2-chloro-3,7-difluoro-11-[4-(4-fluoroaralkyl)piperazino]-10,11-dihydrodibenzo-[b,f]thiepins and related compounds; Long acting tranquillizers
1981, Vol. 46, Issue 1, pp. 141–147 [Abstract]
Karel Šindelář, Miroslav Ryska, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Jiří Protiva and Miroslav Protiva
Fluorinated tricyclic neuroleptics with prolonged action: 3-Fluoro-8-trifluoromethyl derivatives of 10-(4-methylpiperazino)- and 10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo-[b,f]thiepin
1981, Vol. 46, Issue 1, pp. 118–140 [Abstract]
Zdeněk Vejdělek, Miroslav Rajšner, Antonín Dlabač, Miroslav Ryska, Jiří Holubek, Emil Svátek and Miroslav Protiva
Psychotropic derivatives of 5-phenyl-7-chloro-1,3-dihydro-1,4-benzodiazepin-2-one and contribution to the synthesis of its 5-(2-chlorophenyl) analogue
1980, Vol. 45, Issue 12, pp. 3593–3615 [Abstract]
Miroslav Semonský, Antonín Černý, Jiří Křepelka, Rudolf Kotva, Bohumil Kakáč, Jiří Holubek and Jaroslav Vachek
Some ω-(2-amino-6-hydroxy-4-oxo-3,4-dihydro-5-pyrimidinyl) alkanoic acids, their derivatives and analogues
1980, Vol. 45, Issue 12, pp. 3583–3592 [Abstract]
Václav Bártl, Antonín Dlabač and Miroslav Protiva
Tricyclic potential neuroleptics: 2-chloro-11-[4-(4-fluoroaralkyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepins and related compounds
1980, Vol. 45, Issue 11, pp. 3182–3189 [Abstract]
Karel Šindelář, Jiří Jílek, Jiří Körbl, Fedir Jančik, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
Potential metabolites of the neuroleptic agent chlorprothixene; synthesis and pharmacology of the 3-, 4-, 6- and 7-hydroxy and methoxy derivatives of 2-chloro-9-(3-dimethylaminopropylidene)-thioxanthenes
1980, Vol. 45, Issue 11, pp. 3166–3181 [Abstract]
Miloš Buděšínský, Zdeněk Samek and Miloš Tichý
In situ reactions of amines and amino alcohols and their application to structural assignment by ¹H NMR spectroscopy
1980, Vol. 45, Issue 10, pp. 2784–2803 [Abstract]
Jiří Křepelka, Viktor Zikán, Jiří Holubek and Miroslav Semonský
Derivatives of 4-aryl-2,3-dihalogeno-1-naphthol
1980, Vol. 45, Issue 10, pp. 2700–2705 [Abstract]
Jiří Křepelka, Jiří Holubek and Miroslav Semonský
Esters of 4,4-bis(4-ethylphenyl)-2,3-dibromo-2-butenoic acid and 7-ethyl-4-(4-ethylphenyl)-2,3-dibromo-1-naphthol
1980, Vol. 45, Issue 10, pp. 2695–2699 [Abstract]
Irena Červená, Marta Hrubantová, Emil Svátek, Jiří Holubek, Miroslav Ryska, Jiřina Metyšová and Miroslav Protiva
Fluorinated analogues of tricyclic neuroleptics: 6,9-difluoro derivative of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1980, Vol. 45, Issue 10, pp. 2688–2694 [Abstract]
Karel Šindelář, Emil Svátek, Jiří Holubek, Miroslav Ryska, Jiřina Metyšová, Zdeněk Šedivý and Miroslav Protiva
Fluorinated analogues of the tricyclic neuroleptics; 7-Fluoro and 7-trifluoromethyl derivative of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1980, Vol. 45, Issue 4, pp. 1086–1098 [Abstract]
Jiří Křepelka, Jiří Holubek and Miroslav Semonský
Some condensation products of ergoline - I Derivatives with ketones
1980, Vol. 45, Issue 3, pp. 755–760 [Abstract]
Zdeněk Buděšínský, Josef Vavřina, Leon Langšádl and Jiří Holubek
On the synthesis of 4- and 5-pyrimidinyl-diphenyl-(1-imidazolyl)methanes and their antifungal activity
1980, Vol. 45, Issue 2, pp. 539–547 [Abstract]
Vladimír Valenta, Antonín Dlabač, Marie Bartošová, Emil Svátek and Miroslav Protiva
10-[4-(3-Hydroxypropyl)piperazino]-8-methylsulfonyl-10,11-dihydrodibenzo[b,f]thiepin and some related potential metabolites of the neuroleptic agents oxyprothepin and methiothepin
1980, Vol. 45, Issue 2, pp. 529–538 [Abstract]
Vladimír Valenta, Marie Bartošová and Miroslav Protiva
Carbamates and ureas derived from 11-amino-6,11-dihydrodibenzo[b,e]thiepin; Synthesis and pharmacological screening
1980, Vol. 45, Issue 2, pp. 517–528 [Abstract]
Jiří Jílek, Josef Pomykáček, Antonín Dlabač, Marie Bartošová and Miroslav Protiva
Neuroleptics of the 8-methylthio-10-piperazino-10,11-dihydrodibenzo[b,f]thiepin series: New compounds and new procedures
1980, Vol. 45, Issue 2, pp. 504–516 [Abstract]
Karel Šindelář, Jiří Holubek, Emil Svátek and Miroslav Protiva
Synthesis of 3-chloro-5-(4-methylpiperazino)-6,7-dihydro-5H-dibenzo[b,g]thiocin, an eight-membered ring homologue of the neuroleptic agent octoclothepin
1980, Vol. 45, Issue 2, pp. 491–503 [Abstract]
Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiřina Metyšová, Zdeněk Šedivý and Miroslav Protiva
Potential metabolites of the neuroleptic agents noroxyclothepin and oxyclothepin; Synthesis of 8-chloro-3-hydroxy-10-[4-(2-hydroxyethyl)piperazino]- and -10-[4-(3-hydroxypropyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
1979, Vol. 44, Issue 12, pp. 3617–3626 [Abstract]
Zdeněk Vejdělek, Miroslav Rajšner, Emil Svátek, Jiří Holubek and Miroslav Protiva
Synthesis of 7-chloro-5-(6,7,8,9-tetrahydro-5H-benzocyclohepten-2-yl)-2-methylamino-3H-1,4-benzodiazepine 4-oxide and of some related compounds
1979, Vol. 44, Issue 12, pp. 3604–3616 [Abstract]
Vladimír Valenta, Emil Svátek, Antonín Dlabač, Marie Bartošová and Miroslav Protiva
Noncataleptic neuroleptics: Potential metabolites of 2-chloro-10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo[b,fthiepin
1979, Vol. 44, Issue 10, pp. 3008–3018 [Abstract]
Miroslav Rajšner, František Mikšík, Jiřina Metyšová and Miroslav Protiva
Fluorinated tricyclic neuroleptics: Synthesis and pharmacology of 8-fluoro-4-(4-methylpiperazino)-4,5-dihydrothieno[2,3-b]-1-benzothiepin
1979, Vol. 44, Issue 10, pp. 2997–3007 [Abstract]
Miroslav Protiva, Karel Šindelář, Zdeněk Šedivý and Josef Pomykáček
Potential metabolites of tricyclic neuroleptics: 2,8-Dihydroxy and 3,8-dihydroxy derivatives of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1979, Vol. 44, Issue 10, pp. 2987–2996 [Abstract]
Vladimír Valenta, František Kvis, Jiří Němec and Miroslav Protiva
6,11-Dihydrodibenzo[b,e]thiepin-11-thiol and 11-acetic acid derivatives; Some 2-methyl-6,11-dihydrodibenzo[b,e]thiepins; Synthesis and pharmacological screening
1979, Vol. 44, Issue 9, pp. 2689–2701 [Abstract]
Vladimír Valenta, Jiří Jílek, Josef Pomykáček, Antonín Dlabač, Martin Valchář, Jan Metyš and Miroslav Protiva
Noncataleptic potential neuroleptics: 2-Methyl-10-(4-methylpiperazino)- and -10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
1979, Vol. 44, Issue 9, pp. 2677–2688 [Abstract]
Miroslav Rajšner, Václav Bártl, Karel Šindelář, Emil Svátek, Jiří Holubek, Jan Metyš and Miroslav Protiva
Synthesis of new dibenzo[b,e]thiepin derivatives related to the antidepressant agent prothiadene
1979, Vol. 44, Issue 8, pp. 2536–2549 [Abstract]
Irena Červená, Jiřina Metyšová, Václav Bártl and Miroslav Protiva
Fluorinated neuroleptics of the 10-piperazino-10,11-dihydrodibenzo[b,f]thiepin series; 6-Fluoro derivatives of perathiepin, octoclothepin, doclothepin and some related compounds
1979, Vol. 44, Issue 7, pp. 2139–2155 [Abstract]
Jiří O. Jílek, Jiří Holubek, Emil Svátek, Miroslav Ryska, Josef Pomykáček and Miroslav Protiva
Reaction of some 3-(phenylthioaryl)propionic acids with polyphosphoric acid; Formation of 2H-cyclopenta[k,l]thioxanthenes
1979, Vol. 44, Issue 7, pp. 2124–2138 [Abstract]
Miroslav Protiva, Karel Šindelář, Zdeněk Šedivý and Jiřina Metyšová
Potential metabolites of tricyclic neuroleptics and their fluorinated analogues; 3-Hydroxy-, 3-methoxy- and 3-fluoro-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
1979, Vol. 44, Issue 7, pp. 2108–2123 [Abstract]
Miloš Buděšínský, Miloslav Černý, Tomáš Trnka and Soňa Vašíčková
¹H NMR spectra and the conformation of 1,6 : 2,3- and 1,6 : 3,4-dianhydro-β-D-hexopyranoses and their derivatives
1979, Vol. 44, Issue 6, pp. 1965–1983 [Abstract]
Miloš Buděšínský, Tomáš Trnka and Miloslav Černý
The ¹H NMR spectra and the conformation of 1,6-anhydro-β-D-hexopyranoses and their triacetates
1979, Vol. 44, Issue 6, pp. 1949–1964 [Abstract]
Emil Svátek, Viktor Zikán and Miroslav Semonský
Spectral manifestations of strong hydrogen bonds in seven-membered rings of pyrazolecarboxylic acid derivatives
1979, Vol. 44, Issue 3, pp. 781–787 [Abstract]
Zdeněk Samek and Miloš Buděšínský
In situ reactions with trichloroacetyl isocyanate and their application to structural assignment of hydroxy compounds by ¹H NMR spectroscopy. A general comment
1979, Vol. 44, Issue 2, pp. 558–588 [Abstract]
Jiří Klinot, Jarmil Světlý, Dagmar Kudláčková, Miloš Buděšínský and Alois Vystrčil
Preparation of 2-methyl-3-oxo triterpenoids of 18α-oleanane series and the conformation of ring A
1979, Vol. 44, Issue 1, pp. 211–225 [Abstract]
Jiří Jílek, Jiří Holubek, Emil Svátek, Marie Bartošová, Jiřina Metyšová, Josef Pomykáček and Miroslav Protiva
8-Chloro-3-hydroxy-10-piperazino-10,11-dihydrodibenzo[b,f]thiepins, their O-methyl derivatives and further potential metabolites of the neuroleptic agent octoclothepin
1978, Vol. 43, Issue 11, pp. 3092–3102 [Abstract]
Miroslav Protiva, Irena Červená, Miroslav Rajšner, Jiřina Metyšová and Marta Hrubantová
Fluorinated tricyclic neuroleptics: 3-Fluoro and 3,6-difluoro derivatives of chlorprothixene and 6-fluoro-2-isopropyl derivative of prothixene
1978, Vol. 43, Issue 10, pp. 2656–2663 [Abstract]
Jan Vrkoč, Miloš Buděšínský and Petr Sedmera
Structure of 2α,3α-dihydroxy- and 2α,3β-dihydroxy-1(15),8(19)-trinervitadines from Nasututermes costalis (HOLMGREN)
1978, Vol. 43, Issue 9, pp. 2478–2485 [Abstract]
Václav Bártl, Jiří Holubek, Jiří Němec, Marie Bartošová and Miroslav Protiva
Derivatives of 8-chloro-10,11-dihydrodibenzo[b,f]thiepin-10-amine, -10-ol and -10-thiol; Synthesis and pharmacological screening
1978, Vol. 43, Issue 9, pp. 2427–2443 [Abstract]
Huynh Kim Thoa, Želimír Procházka, Miloš Buděšínský and Pavel Kočovský
Hydroxylation of 6β-methoxy-3α,5-cyclo-5α-androstan-17-one with Rhizopus nigricans
1978, Vol. 43, Issue 9, pp. 2305–2311 [Abstract]
Jan Kovář, Ladislav Skurský and Miroslav Protiva
Structural factors affecting interactions of tricyclic psychotropic drugs with alcohol dehydrogenase
1978, Vol. 43, Issue 8, pp. 2068–2081 [Abstract]
Miroslav Rajšner, Zdeňka Kopicová, Jiří Holubek, Emil Svátek, Jan Metyš, Marie Bartošová, František Mikšík and Miroslav Protiva
4,4-Bis(4-fluorophenyl)butylamines and their cyclic analogues; An efficient synthesis of the neuroleptic penfluridol
1978, Vol. 43, Issue 7, pp. 1760–1777 [Abstract]
Jiří O. Jílek, Josef Pomykáček, Jiřina Metyšová, Marie Bartošová and Miroslav Protiva
Potential metabolites of the neuroleptic agent octoclothepin; Synthesis and pharmacology of 8-chloro-6-hydroxy-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin and some related compounds
1978, Vol. 43, Issue 7, pp. 1747–1759 [Abstract]
Zdeněk J. Vejdělek, Marie Bartošová, Miroslav Ryska and Miroslav Protiva
2-(s-Hydrindacen-4-yl)ethylamines and their 1-methyl and 1,1-dimethyl derivatives; Synthesis and pharmacological screening
1978, Vol. 43, Issue 7, pp. 1732–1746 [Abstract]
Viktor Zikán, Miroslav Semonský, Bohumil Kakáč, Jiří Holubek and Karel Řežábek
Reactions of methyl esters of 3-bromo-4-(4-alkoxyphenyl)-4-oxo-2-butenoic acids with diethyl sodium malonate
1978, Vol. 43, Issue 7, pp. 1727–1731 [Abstract]
Miroslav Rajšner, František Mikšík and Miroslav Protiva
[5-Chloro-2-(phenylthio)phenyl]acetic acid, some derivatives and products of further transformations
1978, Vol. 43, Issue 5, pp. 1276–1284 [Abstract]
Jan Vrkoč, Miloš Buděšínský and Petr Sedmera
Structure of trinervitene diterpenoids from Nasutitermes rippertii (RAMBUR)
1978, Vol. 43, Issue 4, pp. 1125–1133 [Abstract]
Zdeněk J. Vejdělek, Marie Bartošová, Alois Čapek and Miroslav Protiva
4-(Aminoacetyl)-s-hydrindacenes and 2-amino-1-(s-hydrindacen-4-yl)-ethanols; Synthesis and pharmacological screening
1978, Vol. 43, Issue 4, pp. 970–980 [Abstract]
Karel Šindelář, Jiří O. Jílek, Josef Pomykáček, Zdeněk Šedivý and Miroslav Protiva
Synthesis of 2-acetyl and 3-acetyl derivatives of 8-chloro-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]-thiepin; 2-Acyl-7-substituted thioxanthenes
1978, Vol. 43, Issue 2, pp. 471–497 [Abstract]
Huynh Kim Thoa, Václav Šašek, Miloš Buděšínský, Ivan Jablonský, Ludmila Eignerová, Nguyen Gia Chan and Želimír Procházka
Biological transformation of 3β-hydroxy-5-androsten-17-one with the mushroom Pleurotus ostreatus (JACQ. ex FR.) KUMM.
1978, Vol. 43, Issue 1, pp. 336–343 [Abstract]
Karel Šindelář, Antonín Dlabač and Miroslav Protiva
Noncataleptic neuroleptics; 8-Chloro-2-hydroxy-11-(4-methylpiperazino)-5H-dibenzo[b,e]-1,4-diazepine as a potential metabolite of clozapine
1978, Vol. 43, Issue 1, pp. 309–315 [Abstract]

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Potentional anxiolytics and hypnotics: 1-(Alkanesulfonamidoalkyl)-6-aryl-8-halogeno-s-triazolo[4,3-a]-1,4-benzodiazepines and related compounds

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