Collect. Czech. Chem. Commun.
1993, 58, S44-S46
https://doi.org/10.1135/cccc1993s044
Synthesis, conformation and anti-HIV activity of 3'-substituted 2',3'-dideoxy-5-hydroxymethyluridines
Tadeusz Kulikowski, Jaroslaw Poznanski, Jan Balzarini, Arthur Van Aerschot and Erik De Clercq
Individual author index pages
Other CCCC articles of these authors
- Dominiquer Askin, Inge Smits, Guy Schepers, Arthur Van Aerschot, Patrick Augustijns and Piet Herdewijn
Synthesis of 3'- and 5'-cholesterol conjugates of oligonucleotides for improving cellular uptake
Symposium Series 1999, Vol. 2, pp. 310–312 [Abstract]
Published online 2016-05-08 23:33:35 - Krzysztof Felczak, Agnieszka Miazga and Tadeusz Kulikowski
Synthesis of novel acyclo 6-phenylselenenyluracils – potential selective anti-HIV agents
Symposium Series 1999, Vol. 2, pp. 245–247 [Abstract]
Published online 2016-05-08 23:31:18 - Karen Vastmans, Luk Kerremans, Chris Hendrix, Arthur Van Aerschot, Sylvie Pochet, Philippe Marlière and Piet Herdewijn
Recognition of 1,5-anhydrohexitol adenine triphosphate by a DNA polymerase
Symposium Series 1999, Vol. 2, pp. 156–160 [Abstract]
Published online 2016-05-08 20:43:00 - Arthur Van Aerschot, Mark Vandermeeren, Johan Geysen, Walter Luyten, Marc Miller, David Atkins, Sonia Preveral, Ester Saison-Behmoaras and Piet Herdewijn
In vitro evaluation of hexitol nucleic acid antisense oligonucleotides
Symposium Series 1999, Vol. 2, pp. 151–155 [Abstract]
Published online 2016-05-08 20:42:54 - Sergei N. Mikhailov, Boris S. Ermolinsky, Ekaterina V. Efimtseva, G. P. Moiseyev, V. L. Tunitskaya, E. E. Rusakova, S. N. Kochetkov, Oksana M. Gritsenko, Elezaveta S. Gromova, Arthur Van Aerschot and Piet Herdewijn
Oligonucleotides containing hexapyranosyl nucleosides and disaccharide nucleosides: Synthesis, incorporation of dialdehyde groups and use as affinity reagents
Symposium Series 1999, Vol. 2, pp. 141–144 [Abstract]
Published online 2016-05-08 20:42:42 - Arthur Van Aerschot, Yuris Maurinsh, Brigitte Allart, Valerie Boudou and Piet Herdewijn
Analogues of hexitol nucleic acids: Structure function relationship of a new steric blocking agent
Symposium Series 1999, Vol. 2, pp. 100–104 [Abstract]
Published online 2016-05-08 20:41:57 - Ekaterina V. Efimtseva, Sergey N. Mikhailov, Jef Rozenski, Roger Busson, Arthur Van Aerschot and Piet Herdewijn
Protection of 1-methyladenosine and its chemical incorporation into oligonucleotides
Symposium Series 2002, Vol. 5, pp. 195–199 [Abstract]
Published online 2016-01-25 20:40:02 - Sergey N. Mikhailov, Ekaterina V. Efimtseva, Alexandra A. Shelkunova, Jef Rozenski, Gert Emmerechts, Arthur Van Aerschot and Piet Herdewijn
Chemical incorporation of minor tRNA component O-β-D-ribofuranosyl-(1''-2')-adenosine-5''-phosphate into oligoribonucleotides
Symposium Series 2005, Vol. 7, pp. 333–337 [Abstract]
Published online 2015-11-08 11:54:55 - Chris Meier, Christian Ducho, Henning Jessen and Jan Balzarini
Esterase-cleavable cycloSal-pronucleotides – the trapping concept
Symposium Series 2005, Vol. 7, pp. 105–113 [Abstract]
Published online 2015-11-08 11:50:56 - Tatjana Gazivoda, Silvana Raić-Malić, Sandra Kraljević-Pavelić, Krešimir Pavelić, Jan Balzarini and Mladen Mintas
The new unsaturated acyclic C-5 pyrimidine nucleoside analogues: synthesis, cytostatic and anti-HIV evaluations
Symposium Series 2008, Vol. 10, pp. 439–441 [Abstract]
Published online 2015-10-30 18:44:36 - Mikhail Abramov, Michael Fisher, Arthur Van Aerschot, Dong Xu, Rudolph L. Juliano and Piet Herdewijn
Inhibition of gene expression with altritol- and hexitol-modified siRNAs
Symposium Series 2008, Vol. 10, pp. 300–301 [Abstract]
Published online 2015-10-30 18:39:42 - Marcela Krečmerová, Antonín Holý, Alois Pískala, Graciela Andrei, Robert Snoeck, Jan Balzarini and Erik De Clercq
New antiviral agent, 1-(S)-[3-hydroxy-2-(phosphonomethoxy)propyl]-5-azacytosine: esters and base-modified derivatives
Symposium Series 2008, Vol. 10, pp. 196–200 [Abstract]
Published online 2015-10-30 18:37:33 - Serge Van Calenbergh, Ineke Van Daele, Sara Van Poecke, Matheus Froeyen, Hélene Munier Lehmann and Jan Balzarini
From M. tuberculosis thymidine monophosphate kinase (TMPKmt) inhibitors towards mitochondrial thymidine kinase (TK-2) inhibitors
Symposium Series 2008, Vol. 10, pp. 87–93 [Abstract]
Published online 2015-10-30 18:35:35 - Kiran Toti, Jan Balzarini and Serge Van Calenbergh
Dideoxyapiose nucleosides revisited: syntheses and protide derivatives
Symposium Series 2011, Vol. 12, pp. 480–482 [Abstract]
Published online 2015-08-20 10:25:10 - Tomáš Tichý, Graciela Andrei, Martin Dračínský, Antonín Holý, Jan Balzarini, Robert Snoeck and Marcela Krečmerová
New amphiphilic prodrugs of adefovir and cidofovir
Symposium Series 2011, Vol. 12, pp. 477–479 [Abstract]
Published online 2015-08-20 10:25:04 - Irina D. Konstantinova, Olga M. Selezneva, Ilja V. Fateev, Tamara A. Balashova, Svetlana K. Kotovskaya, Zoya M. Baskakova, Valery N. Charushin, Alexander V. Baranovsky, Anatoly I. Miroshnikov, Jan Balzarini and Igor A. Mikhailopulo
Chemo-enzymatic syntheses and biological evaluation of 5,6-disubstituted benzimidazole ribo- and 2'-deoxyribo-nucleosides
Symposium Series 2011, Vol. 12, pp. 400–402 [Abstract]
Published online 2015-08-20 10:20:32 - Chris Meier, Edwuin Hander Rios Morales, Cristina Arbelo Román and Jan Balzarini
Stereoselective synthesis of 3-methyl-cycloSal-nucleotides
Symposium Series 2011, Vol. 12, pp. 33–41 [Abstract]
Published online 2015-08-20 09:58:11 - Craig Sergeant, Jan Balzarini and Roman Dembinski
Antiviral activity of 5-halofuropyrimidine nucleosides
Symposium Series 2014, Vol. 14, pp. 209–212 [Abstract]
Published online 2015-07-06 23:01:50 - Erik De Clercq
Acyclic nucleoside phosphonates: An unfinished story
2011, Vol. 76, Issue 7, pp. 829–842 [Abstract] - Georgii V. Bobkov, Kirill V. Brilliantov, Sergey N. Mikhailov*, Jef Rozenski, Arthur Van Aerschot and Piet Herdewijn
Synthesis of Oligoribonucleotides Containing Pyrimidine 2'-O-[(Hydroxyalkoxy)methyl]ribonucleosides
2006, Vol. 71, Issue 6, pp. 804–819 [Abstract] - Ding Zhou, Irene M. Lagoja, Arthur Van Aerschot and Piet Herdewijn*
Synthesis of Aminopropyl Phosphonate Nucleosides with Purine and Pyrimidine Bases
2006, Vol. 71, Issue 1, pp. 15–34 [Abstract] - Zhenyu Zhang, Arthur Van Aerschot, Patrick Chaltin, Roger Busson and Piet Herdewijn*
Epimerization During Coupling to the Unnatural Amino Acid in Solid Phase Peptide Synthesis
2001, Vol. 66, Issue 6, pp. 923–932 [Abstract] - Irene M. Lagoja, Arthur Van Aerschot, Chris Hendrix and Piet Herdewijn*
Glycosylation of 1-Aminoimidazole-2(3H)-thiones
2000, Vol. 65, Issue 7, pp. 1145–1155 [Abstract] - Erik De Clercq
Towards an Effective Chemotherapy of Virus Infections: Therapeutic Potential of Cidofovir [(S)-1-[3-Hydroxy-2-(phosphonomethoxy)propyl]cytosine, HPMPC] for the Treatment of DNA Virus Infections
1998, Vol. 63, Issue 4, pp. 480–506 [Abstract] - Erik De Clercq
New Perspectives for the Treatment of HIV Infections
1998, Vol. 63, Issue 4, pp. 449–479 [Abstract] - Hubert Hřebabecký, Jan Balzarini and Antonín Holý
Preparation of Chloro and Sulfanyl Derivatives of 1-(2-Deoxy-4-C-hydroxymethyl-α-L-threo-Pentofuranosyl)uracil
1997, Vol. 62, Issue 7, pp. 1114–1127 [Abstract] - Sergey N. Mikhailov, Ekaterina V. Efimtseva, Boris S. Ermolinsky, Marina V. Fomitcheva, Oxana M. Gritsenko, Maxim G. Brevnov, Elizaveta S. Gromova, Guy Schepers, Arthur Van Aerschot and Piet Herdewijn
Regioselective incorporation of reactive dialdehyde groups into synthetic oligonucleotides
1996, Vol. 61, Special Issue, pp. S210–S212 [Abstract] - Ekaterina V. Efimtseva, Boris S. Ermolinsky, Marina V. Fomitcheva, Sergey V. Meshkov, Nelly Sh. Padyukova, Sergey N. Mikhailov, Arthur Van Aerschot, Jef Rozenski and Piet Herdewijn
Synthesis of disaccharide nucleosides and their incorporation into oligonucleotides
1996, Vol. 61, Special Issue, pp. S206–S209 [Abstract] - Mirella Marangoni, Arthur Van Aerschot, Patrick Augustijns and Piet A. Herdewijn
Cyclopentylethyl nucleosides as "constrained" acyclic building blocks for oligonucleotides
1996, Vol. 61, Special Issue, pp. S203–S205 [Abstract] - Nicolai E. Poopeiko, Alicja K. Drabikowska, Jaroslav Poznanski, David Shugar and Tadeusz Kulikowski
Synthesis, conformation and biological properties of 2',3'-dideoxy-3'-fluoro-5-chloro-4-thiouridine, potential anti-HIV agent
1996, Vol. 61, Special Issue, pp. S16–S19 [Abstract] - Michal Hocek, Milena Masojídková, Antonín Holý, Graciela Andrei, Robert Snoeck, Jan Balzarini and Erik De Clercq
Synthesis and Antiviral Activity of Acyclic Nucleotide Analogues Derived from 6-(Aminomethyl)purines and Purine-6-carboxamidines
1996, Vol. 61, Issue 10, pp. 1525–1537 [Abstract] - C. Pannecouque, K. Van Poppel, Arthur Van Aerschot and Piet Herdewijn
Synthesis and physicochemical properties of oligonucleotides with an N-cyanoguanidine function instead of the natural phosphate internucleotide linkage
1993, Vol. 58, Special Issue, pp. S191–S194 [Abstract] - Arthur Van Aerschot, F. Vandendriessche, K. Augustyns and Piet Herdewijn
Acyclic nucleosides: Useful for antisense constructs or as universal analogues for degenerate positions?
1993, Vol. 58, Special Issue, pp. S98–S101 [Abstract] - Ilse Verheggen, Nathalie Pillet, Arthur Van Aerschot, Erik De Clercq and Piet Herdewijn
Synthesis and anti-herpesvirus activity of nucleosides with a 1,5-anhydrohexitol moiety
1993, Vol. 58, Special Issue, pp. S64–S67 [Abstract] - Serge Van Calenbergh, Christophe Verlinde, André De Bruyn, Mia Callens, Elfride Van Den Eeckhout, Arthur Van Aerschot, Paul Michels, Fred Opperdoes, Wim Hol and Piet Herdewijn
2'-Substituted adenosine analogues as trypanosomal glyceraldehyde phosphate dehydrogenase (GAPDH) inhibitors
1993, Vol. 58, Special Issue, pp. S52–S55 [Abstract] - Arthur Van Aerschot, Liu Jie, Jan Balzarini, Erik De Clercq and Piet Herdewijn
5'-O-Phosphonomethyl-2',3'-dideoxynucleosides: Synthesis and anti-HIV activity
1990, Vol. 55, Special Issue, pp. S129–S132 [Abstract] - Hiromichi Tanaka, Masanori Baba, Masaru Ubasawa, Hideaki Takashima, Kouichi Sekiya, Tadashi Miyasaka, Issei Nitta, Richard T. Walker and Erik De Clercq
The synthesis of novel 6-substituted acyclouridine derivatives which show specific inhibition of HIV-1
1990, Vol. 55, Special Issue, pp. S89–S92 [Abstract] - Mikko Oivanen, Tuula Viinamäki, Sergei Zavgorodny, Michael Polianski, Alex Azhayev, Arthur Van Aerschot, Piet Herdewijn and Harri Lönnberg
Hydrolytic stability of potential antiviral nucleoside analogues: 3'-Substituted 2',3'-dideoxy- and 2',3'-didehydro-2',3'-dideoxyribonucleosides
1990, Vol. 55, Special Issue, pp. S17–S20 [Abstract] - Piet Wigerinck, Paul Claes, Arthur Van Aerschot and Piet Herdewijn
Heterocycles in the 5-position of 2'-deoxyuridine
1990, Vol. 55, Special Issue, pp. S5–S8 [Abstract] - Antonín Holý, Joachim König, Jiří Veselý, Dieter Cech, Ivan Votruba and Erik De Clercq
5'-O-Alkyl-5-fluorouridines: Synthesis and biological activity
1987, Vol. 52, Issue 6, pp. 1589–1608 [Abstract] - Antonín Holý, Ivan Votruba and Erik De Clercq
Structure-activity studies on open-chain analogues of nucleosides: Inhibition of S-adenosyl-L-homocysteine hydrolase and antiviral activity 2. Acid open-chain analogues
1985, Vol. 50, Issue 1, pp. 262–279 [Abstract] - Antonín Holý, Ivan Votruba and Erik De Clercq
Structure-activity studies on open-chain analogues of nucleosides: Inhibition of S-adenosyl-L-homocysteine hydrolase and antiviral activity 1. Neutral open-chain analogues
1985, Vol. 50, Issue 1, pp. 245–261 [Abstract] - Antonín Holý, Ivan Votruba and Erik De Clercq
Synthesis and antiviral activity of stereoisomeric eritadenines
1982, Vol. 47, Issue 5, pp. 1392–1407 [Abstract] - Antonín Holý and Erik De Clercq
Preparation, spectral properties and biological activities of 5-bromo-6-methyl-2'-deoxyuridine and 5-iodo-6-methyl-2'-deoxyuridine
1980, Vol. 45, Issue 8, pp. 2364–2370 [Abstract]