Collect. Czech. Chem. Commun. 1995, 60, 2147-2155
https://doi.org/10.1135/cccc19952147

Synthesis of a Scaffold for the Creation of Non-Peptide Libraries

Alexander Kasal, Ladislav Kohout and Michal Lebl

Institute of Organic Chemistry and Biochemistry, Academy of Sciences of the Czech Republic, 166 10 Prague 6, Czech Republic

Individual author index pages


Other CCCC articles of these authors

  • Michal Lebl, David L. Heiner, Aaron C. Jones, Steven P. Fambro, Mark J. Nibbe, Steven R. Burgett and Brett M. Ellman
    Automatic oligonucleotide synthesizer utilizing the concept of parallel processing
    Symposium Series 2011, Vol. 12, pp. 264–267 [Abstract]
    Published online 2015-08-20 10:10:52
  • Miloš Buděšínský, Jan Fajkoš, Jaroslav Günter and Alexander Kasal*
    Synthesis, Reactions, Conformation Analysis, and NMR Spectra of 5,10-Epoxy-5ξ,10ξ-estrane-3,17-diones
    2005, Vol. 70, Issue 4, pp. 507–518 [Abstract]
  • Libor Matyáš, Alexander Kasal*, Zoila Babot Riera and Cristina E. Sunol
    Effects of 3α-Amino-5α-pregnan-20-one on GABAA Receptor: Synthesis, Activity and Cytotoxicity
    2004, Vol. 69, Issue 7, pp. 1506–1516 [Abstract]
  • František Franěk*, Tomáš Eckschlager and Ladislav Kohout
    24-Epibrassinolide at Subnanomolar Concentrations Modulates Growth and Production Characteristics of a Mouse Hybridoma
    2003, Vol. 68, Issue 11, pp. 2190–2200 [Abstract]
  • Miroslav Šíša, Miloš Buděšínský and Ladislav Kohout*
    Synthesis and Biological Activity of 7a-Homo- and 7a,7b-Dihomo-5α-cholestane Analogues of Brassinolide
    2003, Vol. 68, Issue 11, pp. 2171–2189 [Abstract]
  • Barbora Slavíková*, Alexander Kasal, Hana Chodounská and Zdena Krištofíková
    3α-Fluoro Analogues of "Allopregnanolone" and Their Binding to GABAA Receptors
    2002, Vol. 67, Issue 1, pp. 30–46 [Abstract]
  • Hana Chodounská, Miloš Buděšínský, Romana Šídová, Miroslav Šíša, Alexander Kasal and Ladislav Kohout*
    Simple NMR Determination of 5α/5β Configuration of 3-Oxosteroids
    2001, Vol. 66, Issue 10, pp. 1529–1544 [Abstract]
  • Michal Lebl*, Christine Burger, Brett Ellman, David Heiner, Georges Ibrahim, Aaron Jones, Mark Nibbe, Jaylynn Thompson, Petr Mudra, Vít Pokorný, Pavel Poncar and Karel Ženíšek
    Fully Automated Parallel Oligonucleotide Synthesizer
    2001, Vol. 66, Issue 8, pp. 1299–1314 [Abstract]
  • Ladislav Kohout*, Hana Chodounská, Tomáš Macek and Miroslav Strnad
    Synthesis of (20S)-2α,3α-Dihydroxy-6-oxo-7-oxa-7a-homo-5α-pregnane-20-carboxylic Acid as a Brassinosteroid Part of Ligands for Binding to Affinity Chromatography Carriers
    2000, Vol. 65, Issue 11, pp. 1754–1761 [Abstract]
  • Hana Chodounská* and Alexander Kasal
    Allopregnanolone Derivatives: Synthesis of 3α-Hydroxy-7a-homo-5α-pregnan-20-one
    2000, Vol. 65, Issue 7, pp. 1156–1162 [Abstract]
  • Jaroslava Hniličková* and Ladislav Kohout
    Synthesis of 21-Hydroxy-6β,19-epoxypregn-4-ene-3,20-dione
    2000, Vol. 65, Issue 3, pp. 380–384 [Abstract]
  • Alexander Kasal*, Miloš Buděšínský, Jan Pelnař, Michael A. Bruck* and Michael F. Brown
    Structures and Synthesis of 4a-Homo-7,19-dinorsteroids, X-Ray Crystallography and NMR Spectroscopy
    1999, Vol. 64, Issue 12, pp. 2019–2034 [Abstract]
  • Barbora Slavíková* and Alexander Kasal
    Epalons: Synthesis of New 16α-Carboxymethyl Derivatives
    1999, Vol. 64, Issue 9, pp. 1479–1484 [Abstract]
  • Alexander Kasal
    Epalons: Synthesis of 7-Norallopregnanolone
    1999, Vol. 64, Issue 9, pp. 1471–1478 [Abstract]
  • Barbora Slavíková, Alexander Kasal* and Miloš Buděšínský
    Autoxidation vs Hydrolysis in 16α-Acyloxy Steroids
    1999, Vol. 64, Issue 7, pp. 1125–1134 [Abstract]
  • Carme Brosa, Ismael Zamora, Emma Terricabras and Ladislav Kohout
    The Effect of Electrostatic Properties and Abibility to Form Hydrogen-Bonds on the Activity of Brassinosteroid Side-Chain Analogs
    1998, Vol. 63, Issue 10, pp. 1635–1645 [Abstract]
  • Alexander Kasal, Jiří Polman and Miloš Buděšínský
    Hydrogenation of a Tetrasubstituted Double Bond: Synthesis of 5-Methyl-19-nor-5β-pregnanes
    1998, Vol. 63, Issue 10, pp. 1549–1563 [Abstract]
  • Hana Chodounská and Alexander Kasal
    Epalons: Synthesis of 3α,7α-Dihydroxy-5α-pregnan-20-one
    1998, Vol. 63, Issue 10, pp. 1543–1548 [Abstract]
  • Romana Šídová, Karel Stránský, Alexander Kasal, Barbora Slavíková and Ladislav Kohout
    Long-Range Effect of 17-Substituents in 3-Oxo Steroids on 4,5-Double Bond Hydrogenation
    1998, Vol. 63, Issue 10, pp. 1528–1542 [Abstract]
  • Barbora Slavíková, Alexander Kasal and Ladislav Kohout
    N-Benzoyl-N-methylandrostan-17β-amines; 20-Aza Analogues of Brassinolide
    1998, Vol. 63, Issue 5, pp. 655–661 [Abstract]
  • Ladislav Kohout, Barbora Slavíková and Miroslav Strnad
    17a-Oxa-17a-homobrassinosteroid Analogues
    1998, Vol. 63, Issue 5, pp. 646–654 [Abstract]
  • Lucie Dalibová and Ladislav Kohout
    Preparation of Steroid Olefins from Heptafluorobutyrates
    1998, Vol. 63, Issue 4, pp. 549–556 [Abstract]
  • Alexander Kasal, Barbora Slavíková, Ladislav Kohout and Miloš Buděšínský
    The Synthesis of A-Homo-B-norandrostanes: The Effect of a Hydroxyl on the Course of Hydrogenation of the ∆9-Double Bond
    1997, Vol. 62, Issue 10, pp. 1631–1641 [Abstract]
  • Barbora Slavíková, Alexander Kasal and Miloš Buděšínský
    Dihydrotestosterone with an Ammonium Centre in the Position 16β
    1997, Vol. 62, Issue 4, pp. 656–664 [Abstract]
  • Josef Vágner, Viktor Krchňák, Michal Lebl and George Barany
    Solid-Phase Organic Synthesis: Creation of Carbon-Carbon Double Bonds Under Mild Conditions by Wittig-Type Reactions
    1996, Vol. 61, Issue 12, pp. 1697–1702 [Abstract]
  • Alexander Kasal, Hana Chodounská and Wojciech J. Szczepek
    trans-Hydrindanes by Reduction: Synthesis of Dihydro-B-nortestosterone
    1996, Vol. 61, Issue 9, pp. 1386–1395 [Abstract]
  • Hana Chodounská, Alexander Kasal, David Šaman and Karel Ubik
    One-Pot Deuteration and Reduction of Ketones in the Synthesis of [16,16,17-2H3]-Epitestosterone
    1996, Vol. 61, Issue 7, pp. 1037–1046 [Abstract]
  • Ladislav Kohout, Alexander Kasal and Miroslav Strnad
    Pregnane-Type Brassinosteroids with a Four-Carbon Ester Functionality in Position 20
    1996, Vol. 61, Issue 6, pp. 930–940 [Abstract]
  • Oldřich Lapčík, Richard Hampl, Martin Hill, Luboslav Stárka, Alexander Kasal, Vladimír Pouzar and Zdeněk Putz
    Radioimmunological and Chromatographic Properties of Tyrosine Methyl Ester Conjugates with Stereoisomeric Steroid Carboxy Derivatives
    1996, Vol. 61, Issue 5, pp. 799–807 [Abstract]
  • Alexander Kasal and Miloš Buděšínský
    Partial Modifications of Hydroxy Groups in 5-Methyl-5β-estr-9-ene Derivatives
    1996, Vol. 61, Issue 2, pp. 276–287 [Abstract]
  • Markéta Rinnová and Michal Lebl
    Molecular Diversity and Libraries of Structures: Synthesis and Screening
    1996, Vol. 61, Issue 2, pp. 171–231 [Abstract]
  • Ladislav Kohout
    7-Oxo-7a-oxa-brassinosteroids with Cholestane Side-Chain
    1994, Vol. 59, Issue 5, pp. 1219–1225 [Abstract]
  • Ladislav Kohout and Alexander Kasal
    7a-Keto-B-homotestosterone and 7a-Keto-B-homoepitestosterone
    1994, Vol. 59, Issue 3, pp. 649–657 [Abstract]
  • Ladislav Kohout
    New Method of Preparation of Brassinosteroids
    1994, Vol. 59, Issue 2, pp. 457–460 [Abstract]
  • Hana Chodounská, Barbora Slavíková and Alexander Kasal
    Synthesis of Some Epitestosterone Analogues
    1994, Vol. 59, Issue 2, pp. 435–443 [Abstract]
  • Zdenko Procházka, Jiřina Slaninová, Per Melin, Carl-Johan Aurell and Michal Lebl
    The Deamino-Carba Analogs of Vasotocin. Synthesis and Some Biological Properties
    1994, Vol. 59, Issue 2, pp. 421–428 [Abstract]
  • Miroslava Žertová, Zdenko Procházka, Jiřina Slaninová, Tomislav Barth, Pavel Majer and Michal Lebl
    The Analogs of [D-Har8]Vasopressin with Di- and Trisubstituted Phenylalanine in Position 2; Synthesis and Some Biological Properties
    1993, Vol. 58, Issue 11, pp. 2751–2760 [Abstract]
  • Alexander Kasal
    Synthesis of 17α-Hydroxy Steroids: B-Norepitestosterone
    1993, Vol. 58, Issue 9, pp. 2202–2210 [Abstract]
  • Alexander Kasal and Světlana Pásztorová
    Synthesis of RIA Haptens: 3α,11α-Dihydroxy-5α-pregnan-20-one 11-Hemisuccinate
    1993, Vol. 58, Issue 3, pp. 619–628 [Abstract]
  • Alexander Kasal, Květa Fuksová and Vladimír Pouzar
    Preparation of Unlabelled and [3H]-Labelled Epitestosterone and Its Metabolites
    1993, Vol. 58, Issue 3, pp. 600–611 [Abstract]
  • Alexander Kasal, Richard Hampl, Zdeněk Putz, Ladislav Kohout and Luboslav Stárka
    Preparation and Properties of Three Immunogens with a Spacer on the β-Side of the Steroid Skeleton and the Effect of Immunogen Structure on Specificity of the Obtained Antisera
    1992, Vol. 57, Issue 10, pp. 2166–2173 [Abstract]
  • Ladislav Kohout and Miroslav Strnad
    Brassinosteroids with Ester Function with Five Carbon Atoms at the 20 Position
    1992, Vol. 57, Issue 8, pp. 1731–1738 [Abstract]
  • B. C. Pal, Jiřina Slaninová, Tomislav Barth, Jerzy Trojnar and Michal Lebl
    Synthesis and Properties of "Hormonogene" and "Inhibitorogene" Type Oxytocin Analogs
    1992, Vol. 57, Issue 6, pp. 1345–1351 [Abstract]
  • Zdenko Procházka, Jiřina Slaninová, Tomislav Barth, Alena Stierandová, Jerzy Trojnar, Per Melin and Michal Lebl
    Analogs of Deamino Carba Oxytocin with Inhibitory Properties; Synthesis and Biological Activities
    1992, Vol. 57, Issue 6, pp. 1335–1344 [Abstract]
  • Miroslava Žertová, Zdenko Procházka, Jiřina Slaninová, Tomislav Barth, Pavel Majer and Michal Lebl
    The Analogs of 8-D-Homoarginin-vasopressin with O-Substituted Phenylalanine in Position 2: Synthesis and Some Biological Properties
    1992, Vol. 57, Issue 5, pp. 1103–1110 [Abstract]
  • Rudolf Ježek, Jan Franc, Jiřina Slaninová and Michal Lebl
    Sequence Modification in Neurohypophyseal Hormones
    1992, Vol. 57, Issue 3, pp. 621–624 [Abstract]
  • Ivo Frič, Michal Lebl and Victor J. Hruby
    Melanin Concentrating Hormone Analogs: Contraction of the Cyclic Structure. III. CD Spectroscopic Study
    1992, Vol. 57, Issue 3, pp. 614–620 [Abstract]
  • Miroslava Žertová, Zdenko Procházka, Jiřina Slaninová, Jana Škopková, Tomislav Barth and Michal Lebl
    Amino and Deamino Analogs of 8-D-Homoarginin-vasopressin with Modified Tyrosine in Position 2: Synthesis and Some Biological Properties
    1992, Vol. 57, Issue 3, pp. 604–613 [Abstract]
  • Marcel Pátek and Michal Lebl
    "Safety-Catch" Protecting Groups in Peptide Synthesis
    1992, Vol. 57, Issue 3, pp. 508–524 [Abstract]
  • Jiří Polman and Alexander Kasal
    The synthesis of 5-methyl-19-nor-5β-pregna-9,16-diene-3,20-dione, 5-methyl-19-nor-5β-pregna-9,10-diene-3,6,20-trione and their analogues with annellated E ring
    1991, Vol. 56, Issue 12, pp. 2892–2905 [Abstract]
  • Miroslava Žertová, Zdenko Procházka, Tomislav Barth, Jiřina Slaninová, Jana Škopková, Ivo Bláha and Michal Lebl
    Strong uterotonic inhibitors – analogs of 1-deamino-8-D-homoarginine-vasopressin with p-substituted phenylalanine in position 2
    1991, Vol. 56, Issue 8, pp. 1761–1767 [Abstract]
  • Miloš Buděšínský, Alexander Kasal, Želimír Procházka, Huynh Kim Thoa, Soňa Vašíčková and Pavel Kočovský
    Revision of the structure of 3-methoxy-14α-hydroxy-D-homo-1,3,5-(10)-estratrien-17a-one. A simple 1H NMR method for the determination of configuration of hydroxy group in position 5 and/or 14 of the D-homo-steroid skeleton
    1991, Vol. 56, Issue 7, pp. 1512–1524 [Abstract]
  • Alexander Kasal, Jenny Pokorná and Jaroslav Zajíček
    3β,11α,17-Trihydroxy-5-pregnen-20-one 11-hemisuccinate as a haptene for RIA of "17α-hydroxypregnenolone"
    1991, Vol. 56, Issue 6, pp. 1340–1347 [Abstract]
  • Alexander Kasal, Jaroslav Podlaha and Jaroslav Zajíček
    A-homo-B,19-dinorandrostanes from 6β-methanesulfonyloxy-5-methyl-19-nor-5β-androst-9-ene derivatives
    1991, Vol. 56, Issue 5, pp. 1070–1086 [Abstract]
  • Miroslava Žertová, Zdenko Procházka, Ivo Bláha, Tomislav Barth, Jiřina Slaninová, Lenka Maletínská and Michal Lebl
    The analogs of 8-D-homoarginine-vasopressin with p-substituted phenylalanine in position 2; Synthesis and some biological properties
    1990, Vol. 55, Issue 12, pp. 3000–3007 [Abstract]
  • Jiří Polman and Alexander Kasal
    Synthesis of 5-methyl-19-nor-5β-pregn-9-ene derivatives
    1990, Vol. 55, Issue 7, pp. 1783–1791 [Abstract]
  • Zdenko Procházka, Juris E. Ancans, Jiřina Slaninová, Alena Machová, Tomislav Barth and Michal Lebl
    Synthesis and biological properties of vasopressin analogues containing 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
    1990, Vol. 55, Issue 4, pp. 1099–1105 [Abstract]
  • Ladislav Kohout
    Syntheis of brassino steroids with a five carbon atom ester functionality in position 17
    1989, Vol. 54, Issue 12, pp. 3348–3359 [Abstract]
  • Alexander Kasal
    Antiandrogenic A-homo-B,19-dinorandrostanes from 5β-methyl-19-norandrost-9-enes with different substituents in positions 3 and 17
    1989, Vol. 54, Issue 8, pp. 2218–2228 [Abstract]
  • Alexander Kasal and Jaroslav Zajíček
    Spontaneous transannular reaction in Δ9-unsaturated A-homo-B,19-dinorsteroids
    1989, Vol. 54, Issue 5, pp. 1327–1335 [Abstract]
  • Alexander Kasal
    Antiandrogenic A-homo-B,19-dinor-analogues of androgens from 6β-chloro-5-methyl-19-nor-5β-androst-9-enes
    1989, Vol. 54, Issue 5, pp. 1318–1326 [Abstract]
  • Ladislav Kohout
    7-Methanesulfonyloxy-3α,5-cyclo-5α-cholestanes
    1989, Vol. 54, Issue 4, pp. 1028–1035 [Abstract]
  • Ladislav Kohout and Miroslav Strnad
    Brassinolide analogues without side chain
    1989, Vol. 54, Issue 4, pp. 1019–1027 [Abstract]
  • Běla Bendlová, Michal Lebl, Pavel Štolba and Luboslav Stárka
    Synthesis of modified human C-peptide and its fragments
    1988, Vol. 53, Issue 11, pp. 2637–2644 [Abstract]
  • Giorgio Fassina, Michal Lebl and Irwin M. Chaiken
    Screening the recognition properties of peptide hormone sequence mutants by analytical high performance liquid affinity chromatography on immobilized neurophysin
    1988, Vol. 53, Issue 11, pp. 2627–2636 [Abstract]
  • Zdenko Procházka, Juris E. Ancans, Jiřina Slaninová, Alena Machová, Tomislav Barth, Jana Škopková, Miloš Buděšínský, Františka Pavlíková and Michal Lebl
    Synthesis and properties of analogues of vasopressin with 1-aminocyclopropane-1-carboxylic acid in position 9
    1988, Vol. 53, Issue 11, pp. 2604–2616 [Abstract]
  • Viktor Krchňák, Josef Vágner, Pavel Šafář and Michal Lebl
    Noninvasive continuous monitoring of solid-phase peptide synthesis by acid-base indicator
    1988, Vol. 53, Issue 11, pp. 2542–2548 [Abstract]
  • Pavel Mader, Věra Veselá, Michael Heyrovský, Michal Lebl and Milena Braunsteinová
    Polarography of the oxytocin and vasopressin synthetic analogs
    1988, Vol. 53, Issue 7, pp. 1579–1605 [Abstract]
  • Ladislav Kohout, Václav Černý and Miroslav Strnad
    Alternative syntheses of 2α,3α,17β-trihydroxy-7-oxa-B-homo-5α-androstan-6-one and some androstane brassinolide analogs
    1987, Vol. 52, Issue 4, pp. 1026–1042 [Abstract]
  • Ladislav Kohout, Helena Velgová, Miroslav Strnad and Miroslav Kamínek
    Brassino steroids with androstane and pregnane skeleton
    1987, Vol. 52, Issue 2, pp. 476–486 [Abstract]
  • Ladislav Kohout
    Solvolytic reactions of epimeric 3-methanesulfonyloxy-7-benzoyloxy-5α,6α-cyclopropanocholestanes
    1986, Vol. 51, Issue 10, pp. 2222–2231 [Abstract]
  • Alexander Kasal and Jaroslav Zajíček
    Solvolysis of Westphalen-type compounds
    1986, Vol. 51, Issue 7, pp. 1462–1475 [Abstract]
  • Ladislav Kohout and Miroslav Strnad
    Brassinosteroids with a cholestane side chain
    1986, Vol. 51, Issue 2, pp. 447–458 [Abstract]
  • Ladislav Kohout, Vijay Kumar Sethi, Jaroslav Zajíček and Alexander Kasal
    Solvolytic reactions of empiric 3-methanesulfonyloxy-7-benzoyloxy-5β,6β-cyclopropanocholestanes
    1986, Vol. 51, Issue 2, pp. 436–446 [Abstract]
  • Ladislav Kohout
    The synthesis of 5,6-cyclopropanocholestanes with oxygen functions in positions 3 and 7
    1986, Vol. 51, Issue 2, pp. 429–435 [Abstract]
  • Alexander Kasal, Ladislav Kohout and Jiří Filip
    4,5-Secoandrostanes by Eschenmoser's reaction
    1985, Vol. 50, Issue 6, pp. 1402–1414 [Abstract]
  • Helena Velgová and Ladislav Kohout
    6,7-Secoandrostane derivatives
    1985, Vol. 50, Issue 4, pp. 962–972 [Abstract]
  • Michal Lebl, Victor J. Hruby, Jiřina Slaninová and Tomislav Barth
    Solid phase synthesis and biological activities of oxytocin carba analogues containing threonine in position 4
    1985, Vol. 50, Issue 2, pp. 418–427 [Abstract]
  • Michal Lebl, Tomislav Barth, Linda Servítová, Jiřina Slaninová and Karel Jošt
    Oxytocin analogues with inhibitory properties, containing in position 2 a hydrophobic amino acid of D-configuration
    1985, Vol. 50, Issue 1, pp. 132–145 [Abstract]
  • Luboslav Stárka, Alexander Kasal, Marie Bičíková and Richard Hampl
    Preparation and synandrogenic activity of 17β-hydroxy-4,5-seco-5-androsten-3-one
    1984, Vol. 49, Issue 12, pp. 2942–2947 [Abstract]
  • Alexander Kasal and Jorga Smolíková
    Photochemical 6β-hydroxylation of 11β-hydroxy-4-androstene-3,17-dione
    1984, Vol. 49, Issue 12, pp. 2932–2941 [Abstract]
  • Michal Lebl, Wayne L. Cody, Brian C. Wilkes, Victor J. Hruby, Anna M. de L. Castrucci and Mac E. Hadley
    Modification of the disulfide bridge in cyclic melanotropins
    1984, Vol. 49, Issue 11, pp. 2680–2688 [Abstract]
  • Michal Lebl, Tomislav Barth, Linda Servítová, Jiřina Slaninová and Pavel Hrbas
    Synthesis and properties of carba-6-analogues of oxytocin containing a deaminopenicillamine residue in position 1
    1984, Vol. 49, Issue 9, pp. 2012–2023 [Abstract]
  • Michal Lebl, Tomislav Barth, Denis J. Crankshaw, Bohuslav Černý, Edwin E. Daniel, A. K. Grover and Karel Jošt
    Synthesis and properties of [2-[3,5-3H2]-tyrosine,4-glutamic acid]deamino-1-carba-oxytocin
    1984, Vol. 49, Issue 8, pp. 1921–1926 [Abstract]
  • Alexander Kasal
    A new type of A-homo-B-norcholestane derivatives
    1984, Vol. 49, Issue 4, pp. 892–902 [Abstract]
  • Zdenko Procházka, Michal Lebl, Tomislav Barth, Jan Hlaváček, Antonín Trka, Miloš Buděšínský and Karel Jošt
    Synthesis and properties of oxytocin analogues modified in the tripeptide side chain
    1984, Vol. 49, Issue 3, pp. 642–652 [Abstract]
  • Ladislav Kohout and Jaroslav Zajíček
    Lead tetraacetate oxidation of 3β-acetoxy-B-homo-5α-cholestan-7aβ-ol
    1984, Vol. 49, Issue 1, pp. 301–305 [Abstract]
  • Daniel Butlen, Tomislav Barth, Bernard Cantau, Gilles Guillon, Serge Jard, Michal Lebl, František Brtník and Karel Jošt
    The structural requirements of oxytocin and vassopressin analogues for the activation of adenylate cyclase in the rat kidney medullary membrane system
    1983, Vol. 48, Issue 11, pp. 3166–3176 [Abstract]
  • Ladislav Kohout and Alexander Kasal
    Electrophilic addition to the 5,6-double bond in A-nor-3,5-secosteroids
    1983, Vol. 48, Issue 7, pp. 2051–2063 [Abstract]
  • Alexander Kasal, Luboš Stárka, Richard Hampl and Ladislav Kohout
    Preparation and pharmacological properties of 4,5-secopregnane-3,20-dione and its derivatives
    1983, Vol. 48, Issue 7, pp. 2040–2050 [Abstract]
  • Tomislav Barth, Bernard Cantau, Daniel Butlen, Gilles Guillon, Serge Jard, Michal Lebl and Karel Jošt
    Oxytocin and vasopressin analogues capable of competition with vasopressin binding to rat liver membranes
    1983, Vol. 48, Issue 6, pp. 1788–1795 [Abstract]
  • Alexander Kasal
    4-Thia-5-cholesten-3-one and some further steroidal δ-thioenol lactones
    1983, Vol. 48, Issue 5, pp. 1489–1498 [Abstract]
  • Ladislav Kohout, Alexander Kasal, Vlastimil Šanda and Helena Velgová
    Rearrangement of the 16,17-cyclopropano derivatives
    1983, Vol. 48, Issue 1, pp. 173–183 [Abstract]
  • Alexander Kasal
    Desulfuration of steroidal thians
    1982, Vol. 47, Issue 11, pp. 3148–3159 [Abstract]
  • Antonín Trka and Alexander Kasal
    Inductive effect in EI-mass spectra of some 5,6-dihalogenides and 5,6-halohydrins of 5α-cholestan-3β-ol and 3β-acetoxy-5α-cholestane
    1982, Vol. 47, Issue 11, pp. 2946–2960 [Abstract]
  • Michal Lebl, Pavel Hrbas, Jana Škopková, Jiřina Slaninová, Alena Machová, Tomislav Barth and Karel Jošt
    Synthesis and properties of oxytocin analogues with high and selective natriuretic activity
    1982, Vol. 47, Issue 9, pp. 2540–2560 [Abstract]
  • Ladislav Kohout, Vlastimil Šanda and Jan Fajkoš
    Synthesis of two isomeric 16,17-cyclopropano derivatives of 5-pregnene
    1982, Vol. 47, Issue 5, pp. 1503–1513 [Abstract]
  • Michal Lebl, Jan Pospíšek, Jan Hlaváček, Tomislav Barth, Petr Maloň, Linda Servítová, Karel Hauzer and Karel Jošt
    Analogues of neurohypophysial hormones, containing tert-leucine: Synthesis and properties
    1982, Vol. 47, Issue 2, pp. 689–701 [Abstract]
  • Alexander Kasal and Ladislav Kohout
    4,5-Secoanalogues of dihydrotestosterone with a cyclopropane ring in the position 5(6)
    1982, Vol. 47, Issue 1, pp. 130–143 [Abstract]
  • Tomislav Barth, Jiřina Slaninová, Linda Servítová, Michal Lebl, Christine Kotsira-Engonopoulos, Chrysa Tzougraki, Iphigenia Photaki, Milan Krojidlo and Karel Jošt
    The effect of some structural modifications of the oxytocin molecule on the duration of the galactogogic response
    1981, Vol. 46, Issue 10, pp. 2441–2445 [Abstract]
  • Alexander Kasal
    Hydrogenation of 12-oxo-5β-chol-9(11)-enates on platinum
    1981, Vol. 46, Issue 8, pp. 1839–1849 [Abstract]
  • Ladislav Kohout
    Synthesis of 5,6-cyclopropanocholestane derivatives with an oxygen function in position 7
    1981, Vol. 46, Issue 8, pp. 1828–1838 [Abstract]
  • Jiřina Slaninová, Michal Lebl, Tomislav Barth and Karel Jošt
    The effect of magnesium ions on the uterotonic activity of carba analogues of oxytocin modified in position 4
    1981, Vol. 46, Issue 7, pp. 1689–1692 [Abstract]
  • Zdenko Procházka, Michal Lebl, Linda Servítová, Tomislav Barth and Karel Jošt
    Synthesis and pharmacological properties of [2-p-fluorophenylalanine]deamino-1-carba-oxytocin and its diastereoisomeric sulfoxides
    1981, Vol. 46, Issue 4, pp. 947–956 [Abstract]
  • Tomislav Barth, Jiřina Slaninová, Michal Lebl and Karel Jošt
    Biological activities and protracted action of carba-analogues of deamino-oxytocin with O-methyltyrosine in position 2
    1980, Vol. 45, Issue 11, pp. 3045–3050 [Abstract]
  • Alexander Kasal and Antonín Trka
    Splitting off of water from the molecular ions of steroidal cyclopropyl ketones
    1980, Vol. 45, Issue 11, pp. 2985–2997 [Abstract]
  • Michal Lebl
    High-performance liquid chromatography of carba-analogues of oxytocin; a method for the determination of sulfides and sulfoxides in peptides
    1980, Vol. 45, Issue 11, pp. 2927–2937 [Abstract]
  • Michal Lebl, Tomislav Barth, Jana Škopková and Karel Jošt
    Synthesis and some pharmacological properties of [7-glycine, 8-ornithine]vasopressin and two of its analogues
    1980, Vol. 45, Issue 10, pp. 2865–2871 [Abstract]
  • Michal Lebl, Tomislav Barth and Karel Jošt
    Synthesis and pharmacological properties of oxytocin analogues modified simultaneously in position 2 and in the disulfide bridge
    1980, Vol. 45, Issue 10, pp. 2855–2864 [Abstract]
  • Michal Lebl, Alena Machová, Pavel Hrbas, Tomislav Barth and Karel Jošt
    Analogues of deamino-1-carba-oxytocin with an aliphatic amino acid in position 4: chemical synthesis and biological activities
    1980, Vol. 45, Issue 10, pp. 2714–2723 [Abstract]
  • Alexander Kasal
    Analogues of androgens with the open ring A
    1980, Vol. 45, Issue 9, pp. 2541–2549 [Abstract]
  • František Tureček and Ladislav Kohout
    The stereospecific loss of water from B-homocholestanols under electron impact
    1980, Vol. 45, Issue 9, pp. 2433–2442 [Abstract]
  • Ladislav Kohout and Jan Fajkoš
    Analogues of androgens with a cyclopropane ring in 6α,7α-position
    1980, Vol. 45, Issue 7, pp. 1974–1981 [Abstract]
  • Antonín Trka and Alexander Kasal
    Electron impact mass spectra of some vicinal trans-dihalo- and trans-hydroxyhalocholestanes
    1980, Vol. 45, Issue 6, pp. 1720–1733 [Abstract]
  • Pavel Kočovský, Ladislav Kohout and Václav Černý
    Participation of 19-substituents in electrophilic additions to 6,7-unsaturated 5α-cholestane and B-homo 5α-cholestane derivatives; A case of competition between the participation of an ambident neighboring group and external nucleophile attack
    1980, Vol. 45, Issue 2, pp. 559–583 [Abstract]
  • Vlastimil Šanda, Ladislav Kohout and Jan Fajkoš
    5,7-Cyclo-B-homopregnane derivatives with the corticoid ketol side chain
    1980, Vol. 45, Issue 1, pp. 269–273 [Abstract]
  • Ladislav Kohout and Jan Fajkoš
    Acetolysis of 4β-methanesulphonyloxy-6β,7aβ-cyclo-B-homo-5α-cholestane
    1979, Vol. 44, Issue 11, pp. 3308–3320 [Abstract]
  • Michal Lebl, Vera Bojanovska, Tomislav Barth and Karel Jošt
    Synthesis and properties of oxytocin analogues acting as irreversible inhibitors of the uterotonic response to oxytocin
    1979, Vol. 44, Issue 8, pp. 2573–2582 [Abstract]
  • Michal Lebl, Tomislav Barth and Karel Jošt
    Analogues of oxytocin with esters of glutamic acid instead of glutamine in position 4: Synthesis of a compound with high and specific galactogogic activity
    1979, Vol. 44, Issue 8, pp. 2563–2572 [Abstract]
  • Michal Lebl, Anastasia Dimeli, Vera Bojanovska, Jiřina Slaninová, Tomislav Barth and Karel Jošt
    Synthesis and some biological properties of amides derived from [4-glutamic acid]deamino-1-carba-oxytocin
    1979, Vol. 44, Issue 8, pp. 2556–2562 [Abstract]
  • Alexander Kasal
    Deoxygenation at the carbon C(5) of 3,6-cyclo-A-nor-3,5-secoandrostanes
    1979, Vol. 44, Issue 5, pp. 1619–1629 [Abstract]
  • Bruno Schönecker, Dieter Tresselt, Gerd Schubert, Ladislav Kohout and Jan Fajkoš
    1H-NMR investigations. Application of trichloroacetyl isocyanate to structure determination of 3-, 6-, 7-, 7a- and 17-hydroxy steroids
    1978, Vol. 43, Issue 10, pp. 2609–2618 [Abstract]
  • Alexander Kasal
    Synthesis of 3,6-cyclo-A-nor-3,5-secoandrostanes
    1978, Vol. 43, Issue 7, pp. 1778–1792 [Abstract]
  • Michal Lebl, Tomislav Barth and Karel Jošt
    Synthesis, reduction, and pharmacological properties of the sulfoxides of some carba-analogues of oxytocin
    1978, Vol. 43, Issue 6, pp. 1538–1556 [Abstract]
  • Michal Lebl, Tomislav Barth and Karel Jošt
    Nα-Glycyl-glycyl-glycyl-8-ornithine-vasopressin: A trypsin resistant vasopressin analog with a specific pressor effect
    1978, Vol. 43, Issue 5, pp. 1300–1305 [Abstract]
  • Ladislav Kohout and Jan Fajkoš
    Methylenation of 4,6-cholestadien-3-one
    1978, Vol. 43, Issue 4, pp. 1134–1141 [Abstract]
  • Ladislav Kohout
    2,3-Disubstituted derivatives of the 6β,7aβ-cyclo-B-homo-5α-cholestane series
    1978, Vol. 43, Issue 3, pp. 889–899 [Abstract]
  • Ladislav Kohout and Jan Fajkoš
    Fission of the epimeric 2,3-epoxides in the 5,7β-cyclo-B-homo-5β-cholestane series
    1978, Vol. 43, Issue 2, pp. 638–646 [Abstract]
  • Michal Lebl and Karel Jošt
    Synthesis of [4-glutamic acid]deamino-1-carba-oxytocin
    1978, Vol. 43, Issue 2, pp. 523–534 [Abstract]
  • Alexander Kasal
    Reduction of some 3,6-cyclo-A-nor-3,5-seco-6β-cholestanes
    1978, Vol. 43, Issue 2, pp. 498–510 [Abstract]