Collect. Czech. Chem. Commun. 2004, 69, 1491-1498
https://doi.org/10.1135/cccc20041491

Synthesis and Leukemia Cell Growth Inhibition of a Series of 1,3-Dithiazolylbenzene Derivatives

Irene M. Lagojaa, Koen Nauwelaertsa, Christine Bal-Mahieub, Michela Pasqualinia, Christian Baillyb and Piet Herdewijna,*

a Laboratory of Medicinal Chemistry, Rega Institute for Medical Research, Katholieke Universiteit Leuven, Minderbroedersstraat 10, B-3000 Leuven, Belgium
b INSERM U-524 et Laboratoire de Pharmacologie Antitumorale du Centre Oscar Lambret, IRCL, 59045 Lille, France

Individual author index pages


Other CCCC articles of these authors

  • Dominiquer Askin, Inge Smits, Guy Schepers, Arthur Van Aerschot, Patrick Augustijns and Piet Herdewijn
    Synthesis of 3'- and 5'-cholesterol conjugates of oligonucleotides for improving cellular uptake
    Symposium Series 1999, Vol. 2, pp. 310–312 [Abstract]
    Published online 2016-05-08 23:33:35
  • Serge Van Calenbergh, Andreas Link, Shelly Fujikawa, Veerle Vanheusden, Denis De Keukeleire, Adriaan P. Ijzerman and Piet Herdewijn
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    Published online 2016-05-08 23:32:32
  • Karen Vastmans, Luk Kerremans, Chris Hendrix, Arthur Van Aerschot, Sylvie Pochet, Philippe Marlière and Piet Herdewijn
    Recognition of 1,5-anhydrohexitol adenine triphosphate by a DNA polymerase
    Symposium Series 1999, Vol. 2, pp. 156–160 [Abstract]
    Published online 2016-05-08 20:43:00
  • Arthur Van Aerschot, Mark Vandermeeren, Johan Geysen, Walter Luyten, Marc Miller, David Atkins, Sonia Preveral, Ester Saison-Behmoaras and Piet Herdewijn
    In vitro evaluation of hexitol nucleic acid antisense oligonucleotides
    Symposium Series 1999, Vol. 2, pp. 151–155 [Abstract]
    Published online 2016-05-08 20:42:54
  • Sergei N. Mikhailov, Boris S. Ermolinsky, Ekaterina V. Efimtseva, G. P. Moiseyev, V. L. Tunitskaya, E. E. Rusakova, S. N. Kochetkov, Oksana M. Gritsenko, Elezaveta S. Gromova, Arthur Van Aerschot and Piet Herdewijn
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    Symposium Series 1999, Vol. 2, pp. 141–144 [Abstract]
    Published online 2016-05-08 20:42:42
  • Arthur Van Aerschot, Yuris Maurinsh, Brigitte Allart, Valerie Boudou and Piet Herdewijn
    Analogues of hexitol nucleic acids: Structure function relationship of a new steric blocking agent
    Symposium Series 1999, Vol. 2, pp. 100–104 [Abstract]
    Published online 2016-05-08 20:41:57
  • Ekaterina V. Efimtseva, Andrei A. Rodionov, Georgii V. Bobkov, Boris S. Ermolinsky, Marina V. Fomitcheva, Sergey N. Mikhailov and Piet Herdewijn
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    Symposium Series 1999, Vol. 2, pp. 22–26 [Abstract]
    Published online 2016-05-08 20:40:11
  • Philippe Van Rompaey, Vanheusden Veerle, Sylvie Pochet, Hélene Munier-Lehmann, Matheus Froeyen, Piet Herdewijn and Serge Van Calenbergh
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  • Philippe Van Rompaey, Kenneth A. Jacobson, Zhan-Guo Gao, Aishe Chen, Dov Barak, Soon-Ai Kim, Kyeong Lee, Andreas Link, Bruce T. Liang, Piet Herdewijn and Serge Van Calenbergh
    Amine-modified nucleosides as adenosine A3 neoceptor ligands
    Symposium Series 2002, Vol. 5, pp. 267–271 [Abstract]
    Published online 2016-01-25 20:41:17
  • Ekaterina V. Efimtseva, Sergey N. Mikhailov, Jef Rozenski, Roger Busson, Arthur Van Aerschot and Piet Herdewijn
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    Symposium Series 2002, Vol. 5, pp. 195–199 [Abstract]
    Published online 2016-01-25 20:40:02
  • Sergey N. Mikhailov, Ekaterina V. Efimtseva, Alexandra A. Shelkunova, Jef Rozenski, Gert Emmerechts, Arthur Van Aerschot and Piet Herdewijn
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    Symposium Series 2005, Vol. 7, pp. 333–337 [Abstract]
    Published online 2015-11-08 11:54:55
  • Irene M. Lagoja
    "Split-nucleosides" – a novel class of purine bioisosters
    Symposium Series 2005, Vol. 7, pp. 173–175 [Abstract]
    Published online 2015-11-08 11:51:59
  • Piet Herdewijn
    The Diels–Alder cyclo addition as key reaction for the synthesis of cyclohexenyl nucleosides
    Symposium Series 2005, Vol. 7, pp. 29–37 [Abstract]
    Published online 2015-11-08 11:50:03
  • Mikhail Abramov, Michael Fisher, Arthur Van Aerschot, Dong Xu, Rudolph L. Juliano and Piet Herdewijn
    Inhibition of gene expression with altritol- and hexitol-modified siRNAs
    Symposium Series 2008, Vol. 10, pp. 300–301 [Abstract]
    Published online 2015-10-30 18:39:42
  • Martin Kögler, Bart Vanderhoydonck, Steven de Jonghe, Jean Herman, Thierry Louat, Kristien van Belle, Jef Rozenski and Piet Herdewijn
    Synthesis and evaluation of 5-substituted-2'-deoxyuridine monophosphate analogues as inhibitors of flavin-dependent thymidylate synthase in Mycobacterium tuberculosis
    Symposium Series 2011, Vol. 12, pp. 364–366 [Abstract]
    Published online 2015-08-20 10:19:12
  • Anastasia Parchina, Matheus Froeyen, Lia Margamuljana, Jef Rozenski, Steven de Jonghe, Yves Briers, Rob Lavigne, Piet Herdewijn and Eveline Lescrinier
    Discovery of an acyclic nucleoside phosphonate that inhibits Mycobacterium Tuberculosis ThyX based on the binding mode of a 5-alkynyl substrate analogue
    Symposium Series 2014, Vol. 14, pp. 342–343 [Abstract]
    Published online 2015-07-06 23:07:34
  • Matheus Froeyen, Hans De Winter and Piet Herdewijn*
    Conformational Analysis, Solvent-Accessible Surface and Geometric Extent of Inhibitors and Substrates
    2006, Vol. 71, Issue 6, pp. 842–858 [Abstract]
  • Georgii V. Bobkov, Kirill V. Brilliantov, Sergey N. Mikhailov*, Jef Rozenski, Arthur Van Aerschot and Piet Herdewijn
    Synthesis of Oligoribonucleotides Containing Pyrimidine 2'-O-[(Hydroxyalkoxy)methyl]ribonucleosides
    2006, Vol. 71, Issue 6, pp. 804–819 [Abstract]
  • Ding Zhou, Irene M. Lagoja, Arthur Van Aerschot and Piet Herdewijn*
    Synthesis of Aminopropyl Phosphonate Nucleosides with Purine and Pyrimidine Bases
    2006, Vol. 71, Issue 1, pp. 15–34 [Abstract]
  • Thierry Lioux, Roger Busson, Jef Rozenski, Martine Nguyen-Distèche, Jean-Marie Frère and Piet Herdewijn*
    Synthesis of Peptidoglycan Units with UDP at the Anomeric Position
    2005, Vol. 70, Issue 10, pp. 1615–1641 [Abstract]
  • Zhenyu Zhang, Arthur Van Aerschot, Patrick Chaltin, Roger Busson and Piet Herdewijn*
    Epimerization During Coupling to the Unnatural Amino Acid in Solid Phase Peptide Synthesis
    2001, Vol. 66, Issue 6, pp. 923–932 [Abstract]
  • Irene M. Lagoja, Arthur Van Aerschot, Chris Hendrix and Piet Herdewijn*
    Glycosylation of 1-Aminoimidazole-2(3H)-thiones
    2000, Vol. 65, Issue 7, pp. 1145–1155 [Abstract]
  • Sergey N. Mikhailov, Ekaterina V. Efimtseva, Boris S. Ermolinsky, Marina V. Fomitcheva, Oxana M. Gritsenko, Maxim G. Brevnov, Elizaveta S. Gromova, Guy Schepers, Arthur Van Aerschot and Piet Herdewijn
    Regioselective incorporation of reactive dialdehyde groups into synthetic oligonucleotides
    1996, Vol. 61, Special Issue, pp. S210–S212 [Abstract]
  • Ekaterina V. Efimtseva, Boris S. Ermolinsky, Marina V. Fomitcheva, Sergey V. Meshkov, Nelly Sh. Padyukova, Sergey N. Mikhailov, Arthur Van Aerschot, Jef Rozenski and Piet Herdewijn
    Synthesis of disaccharide nucleosides and their incorporation into oligonucleotides
    1996, Vol. 61, Special Issue, pp. S206–S209 [Abstract]
  • C. Pannecouque, K. Van Poppel, Arthur Van Aerschot and Piet Herdewijn
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    1993, Vol. 58, Special Issue, pp. S191–S194 [Abstract]
  • Arthur Van Aerschot, F. Vandendriessche, K. Augustyns and Piet Herdewijn
    Acyclic nucleosides: Useful for antisense constructs or as universal analogues for degenerate positions?
    1993, Vol. 58, Special Issue, pp. S98–S101 [Abstract]
  • Ilse Verheggen, Nathalie Pillet, Arthur Van Aerschot, Erik De Clercq and Piet Herdewijn
    Synthesis and anti-herpesvirus activity of nucleosides with a 1,5-anhydrohexitol moiety
    1993, Vol. 58, Special Issue, pp. S64–S67 [Abstract]
  • Serge Van Calenbergh, Christophe Verlinde, André De Bruyn, Mia Callens, Elfride Van Den Eeckhout, Arthur Van Aerschot, Paul Michels, Fred Opperdoes, Wim Hol and Piet Herdewijn
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    1993, Vol. 58, Special Issue, pp. S52–S55 [Abstract]
  • Arthur Van Aerschot, Liu Jie, Jan Balzarini, Erik De Clercq and Piet Herdewijn
    5'-O-Phosphonomethyl-2',3'-dideoxynucleosides: Synthesis and anti-HIV activity
    1990, Vol. 55, Special Issue, pp. S129–S132 [Abstract]
  • Mikko Oivanen, Tuula Viinamäki, Sergei Zavgorodny, Michael Polianski, Alex Azhayev, Arthur Van Aerschot, Piet Herdewijn and Harri Lönnberg
    Hydrolytic stability of potential antiviral nucleoside analogues: 3'-Substituted 2',3'-dideoxy- and 2',3'-didehydro-2',3'-dideoxyribonucleosides
    1990, Vol. 55, Special Issue, pp. S17–S20 [Abstract]
  • Piet Wigerinck, Paul Claes, Arthur Van Aerschot and Piet Herdewijn
    Heterocycles in the 5-position of 2'-deoxyuridine
    1990, Vol. 55, Special Issue, pp. S5–S8 [Abstract]