Collect. Czech. Chem. Commun.
2006, 71, 804-819
https://doi.org/10.1135/cccc20060804
Synthesis of Oligoribonucleotides Containing Pyrimidine 2'-O-[(Hydroxyalkoxy)methyl]ribonucleosides
Georgii V. Bobkova, Kirill V. Brilliantova, Sergey N. Mikhailova,*, Jef Rozenskib, Arthur Van Aerschotb and Piet Herdewijnb
a Engelhardt Institute of Molecular Biology, Russian Academy of Sciences, Vavilov str. 32, Moscow 119991, Russia
b Rega Institute, Katholieke Universiteit Leuven, Minderbroedersstraat 10, B-3000 Leuven, Belgium
Individual author index pages
- Georgii V. Bobkov
- Kirill V. Brilliantov
- Sergey N. Mikhailov
- Jef Rozenski
- Arthur Van Aerschot
- Piet Herdewijn
Other CCCC articles of these authors
- Dominiquer Askin, Inge Smits, Guy Schepers, Arthur Van Aerschot, Patrick Augustijns and Piet Herdewijn
Synthesis of 3'- and 5'-cholesterol conjugates of oligonucleotides for improving cellular uptake
Symposium Series 1999, Vol. 2, pp. 310–312 [Abstract]
Published online 2016-05-08 23:33:35 - Serge Van Calenbergh, Andreas Link, Shelly Fujikawa, Veerle Vanheusden, Denis De Keukeleire, Adriaan P. Ijzerman and Piet Herdewijn
5'-Deoxy congeners of 9-(3-amido-3-deoxy-β-D-xylofuranosyl)-N6-cyclopentyladenine: New adenosine A1 receptor antagonists
Symposium Series 1999, Vol. 2, pp. 273–276 [Abstract]
Published online 2016-05-08 23:32:32 - Karen Vastmans, Luk Kerremans, Chris Hendrix, Arthur Van Aerschot, Sylvie Pochet, Philippe Marlière and Piet Herdewijn
Recognition of 1,5-anhydrohexitol adenine triphosphate by a DNA polymerase
Symposium Series 1999, Vol. 2, pp. 156–160 [Abstract]
Published online 2016-05-08 20:43:00 - Arthur Van Aerschot, Mark Vandermeeren, Johan Geysen, Walter Luyten, Marc Miller, David Atkins, Sonia Preveral, Ester Saison-Behmoaras and Piet Herdewijn
In vitro evaluation of hexitol nucleic acid antisense oligonucleotides
Symposium Series 1999, Vol. 2, pp. 151–155 [Abstract]
Published online 2016-05-08 20:42:54 - Sergei N. Mikhailov, Boris S. Ermolinsky, Ekaterina V. Efimtseva, G. P. Moiseyev, V. L. Tunitskaya, E. E. Rusakova, S. N. Kochetkov, Oksana M. Gritsenko, Elezaveta S. Gromova, Arthur Van Aerschot and Piet Herdewijn
Oligonucleotides containing hexapyranosyl nucleosides and disaccharide nucleosides: Synthesis, incorporation of dialdehyde groups and use as affinity reagents
Symposium Series 1999, Vol. 2, pp. 141–144 [Abstract]
Published online 2016-05-08 20:42:42 - Arthur Van Aerschot, Yuris Maurinsh, Brigitte Allart, Valerie Boudou and Piet Herdewijn
Analogues of hexitol nucleic acids: Structure function relationship of a new steric blocking agent
Symposium Series 1999, Vol. 2, pp. 100–104 [Abstract]
Published online 2016-05-08 20:41:57 - Ekaterina V. Efimtseva, Andrei A. Rodionov, Georgii V. Bobkov, Boris S. Ermolinsky, Marina V. Fomitcheva, Sergey N. Mikhailov and Piet Herdewijn
Studies on disaccharide nucleoside synthesis
Symposium Series 1999, Vol. 2, pp. 22–26 [Abstract]
Published online 2016-05-08 20:40:11 - Philippe Van Rompaey, Vanheusden Veerle, Sylvie Pochet, Hélene Munier-Lehmann, Matheus Froeyen, Piet Herdewijn and Serge Van Calenbergh
Thymidine (monophosphate) analogues as Mycobacterium tuberculosis thymidylate kinase inhibitors
Symposium Series 2002, Vol. 5, pp. 393–395 [Abstract]
Published online 2016-01-25 20:52:11 - Irina V. Gulyaeva, Ekaterina V. Efimtseva, Andrei A. Rodionov, Boris S. Ermolinsky and Sergey N. Mikhailov
Direct synthesis of 5'-nucleotides using glycosylation reaction
Symposium Series 2002, Vol. 5, pp. 312–315 [Abstract]
Published online 2016-01-25 20:42:07 - Philippe Van Rompaey, Kenneth A. Jacobson, Zhan-Guo Gao, Aishe Chen, Dov Barak, Soon-Ai Kim, Kyeong Lee, Andreas Link, Bruce T. Liang, Piet Herdewijn and Serge Van Calenbergh
Amine-modified nucleosides as adenosine A3 neoceptor ligands
Symposium Series 2002, Vol. 5, pp. 267–271 [Abstract]
Published online 2016-01-25 20:41:17 - Ekaterina V. Efimtseva, Sergey N. Mikhailov, Jef Rozenski, Roger Busson, Arthur Van Aerschot and Piet Herdewijn
Protection of 1-methyladenosine and its chemical incorporation into oligonucleotides
Symposium Series 2002, Vol. 5, pp. 195–199 [Abstract]
Published online 2016-01-25 20:40:02 - Sergey N. Mikhailov and Ekaterina V. Efimtseva
Disaccharide nucleosides and oligonucleotides on their basis
Symposium Series 2002, Vol. 5, pp. 181–194 [Abstract]
Published online 2016-01-25 20:39:56 - Irina V. Kulikova, Ivan S. Varizhuk, Georgii V. Bobkov, Ekaterina V. Efimtseva and Sergey N. Mikhailov
Effective anomerisation of 2'-deoxyadenosine and thymidine derivatives
Symposium Series 2005, Vol. 7, pp. 425–427 [Abstract]
Published online 2015-11-08 11:57:16 - Sergey N. Mikhailov, Ekaterina V. Efimtseva, Alexandra A. Shelkunova, Jef Rozenski, Gert Emmerechts, Arthur Van Aerschot and Piet Herdewijn
Chemical incorporation of minor tRNA component O-β-D-ribofuranosyl-(1''-2')-adenosine-5''-phosphate into oligoribonucleotides
Symposium Series 2005, Vol. 7, pp. 333–337 [Abstract]
Published online 2015-11-08 11:54:55 - Piet Herdewijn
The Diels–Alder cyclo addition as key reaction for the synthesis of cyclohexenyl nucleosides
Symposium Series 2005, Vol. 7, pp. 29–37 [Abstract]
Published online 2015-11-08 11:50:03 - Natalia R. Kildeeva, Vasilii V. Nikonorov, Petr A. Perminov, Alexandra N. Zakharova and Sergey N. Mikhailov
Periodate oxidized derivatives of nucleosides and nucleotides as novel crosslinking reagents
Symposium Series 2008, Vol. 10, pp. 407–409 [Abstract]
Published online 2015-10-30 18:43:37 - Mikhail Abramov, Michael Fisher, Arthur Van Aerschot, Dong Xu, Rudolph L. Juliano and Piet Herdewijn
Inhibition of gene expression with altritol- and hexitol-modified siRNAs
Symposium Series 2008, Vol. 10, pp. 300–301 [Abstract]
Published online 2015-10-30 18:39:42 - Irina V. Kulikova, Daria A. Muradova, Ivan S. Varizhuk and Sergey N. Mikhailov
Stereospecific synthesis of 2'-O-α-D-ribofuranosylnucleosides
Symposium Series 2008, Vol. 10, pp. 155–158 [Abstract]
Published online 2015-10-30 18:36:41 - Svetlana V. Kolyachkina, Vitali I. Tararov, Cyril S. Alexeev and Sergey N. Mikhailov
Synthesis of N6-substituted adenosines
Symposium Series 2011, Vol. 12, pp. 405–407 [Abstract]
Published online 2015-08-20 10:20:43 - Mikhail S. Drenichev, Georgii V. Bobkov, Vitali I. Tararov and Sergey N. Mikhailov
Selective cleavage of acyl protecting groups in 3',5'-O-(tetraisopropyldisiloxane-1,3-diyl)ribonucleosides
Symposium Series 2011, Vol. 12, pp. 403–404 [Abstract]
Published online 2015-08-20 10:20:37 - Martin Kögler, Bart Vanderhoydonck, Steven de Jonghe, Jean Herman, Thierry Louat, Kristien van Belle, Jef Rozenski and Piet Herdewijn
Synthesis and evaluation of 5-substituted-2'-deoxyuridine monophosphate analogues as inhibitors of flavin-dependent thymidylate synthase in Mycobacterium tuberculosis
Symposium Series 2011, Vol. 12, pp. 364–366 [Abstract]
Published online 2015-08-20 10:19:12 - Alexandra N. Zakharova, Valentin V. Novikov, Petr A. Perminov, Natalia R. Kildeeva and Sergey N. Mikhailov
Dialdehyde derivatives of nucleosides and nucleotides as novel crosslinking reagents and their comparison with glutaraldehyde
Symposium Series 2011, Vol. 12, pp. 254–258 [Abstract]
Published online 2015-08-20 10:10:40 - Anastasia Parchina, Matheus Froeyen, Lia Margamuljana, Jef Rozenski, Steven de Jonghe, Yves Briers, Rob Lavigne, Piet Herdewijn and Eveline Lescrinier
Discovery of an acyclic nucleoside phosphonate that inhibits Mycobacterium Tuberculosis ThyX based on the binding mode of a 5-alkynyl substrate analogue
Symposium Series 2014, Vol. 14, pp. 342–343 [Abstract]
Published online 2015-07-06 23:07:34 - Mikhail S. Drenichev, Vladimir E. Oslovsky and Sergey N. Mikhailov
Synthesis of 1-N and N6-substituted adenosines
Symposium Series 2014, Vol. 14, pp. 257–258 [Abstract]
Published online 2015-07-06 23:03:52 - Mikhail S. Drenichev, Vladimir E. Oslovsky and Sergey N. Mikhailov
Further improvements in disaccharide synthesis: synthesis of 2’-O-α-D-ribofuranosyladenosine and its derivatives
Symposium Series 2014, Vol. 14, pp. 255–256 [Abstract]
Published online 2015-07-06 23:03:46 - Svetlana V. Kolyachkina, Vitali I. Tararov, Cyril S. Alexeev, Dmitry M. Krivosheev, Georgy A. Romanov, Evgenia V. Stepanova, Eliso S. Solomko, Andrey N. Inshakov and Sergey N. Mikhailov*
N6-substituted adenosines. Cytokinin and antitumor activities
2011, Vol. 76, Issue 11, pp. 1361–1378 [Abstract] - Matheus Froeyen, Hans De Winter and Piet Herdewijn*
Conformational Analysis, Solvent-Accessible Surface and Geometric Extent of Inhibitors and Substrates
2006, Vol. 71, Issue 6, pp. 842–858 [Abstract] - Ding Zhou, Irene M. Lagoja, Arthur Van Aerschot and Piet Herdewijn*
Synthesis of Aminopropyl Phosphonate Nucleosides with Purine and Pyrimidine Bases
2006, Vol. 71, Issue 1, pp. 15–34 [Abstract] - Thierry Lioux, Roger Busson, Jef Rozenski, Martine Nguyen-Distèche, Jean-Marie Frère and Piet Herdewijn*
Synthesis of Peptidoglycan Units with UDP at the Anomeric Position
2005, Vol. 70, Issue 10, pp. 1615–1641 [Abstract] - Irene M. Lagoja, Koen Nauwelaerts, Christine Bal-Mahieu, Michela Pasqualini, Christian Bailly and Piet Herdewijn*
Synthesis and Leukemia Cell Growth Inhibition of a Series of 1,3-Dithiazolylbenzene Derivatives
2004, Vol. 69, Issue 7, pp. 1491–1498 [Abstract] - Zhenyu Zhang, Arthur Van Aerschot, Patrick Chaltin, Roger Busson and Piet Herdewijn*
Epimerization During Coupling to the Unnatural Amino Acid in Solid Phase Peptide Synthesis
2001, Vol. 66, Issue 6, pp. 923–932 [Abstract] - Irene M. Lagoja, Arthur Van Aerschot, Chris Hendrix and Piet Herdewijn*
Glycosylation of 1-Aminoimidazole-2(3H)-thiones
2000, Vol. 65, Issue 7, pp. 1145–1155 [Abstract] - Boris S. Ermolinsky, Marina V. Fomitcheva, Ekaterina V. Efimtseva, Sergey V. Meshkov, Sergey N. Mikhailov, Dmitriy S. Esipov, Elena F. Boldyreva and Vyacheslav G. Korobko
Oligodeoxyribonucleosides containing 1-(β-D-glucopyranosyl)thymine: Synthesis and substrate properties
1996, Vol. 61, Special Issue, pp. S222–S225 [Abstract] - Sergey N. Mikhailov, Ekaterina V. Efimtseva, Boris S. Ermolinsky, Marina V. Fomitcheva, Oxana M. Gritsenko, Maxim G. Brevnov, Elizaveta S. Gromova, Guy Schepers, Arthur Van Aerschot and Piet Herdewijn
Regioselective incorporation of reactive dialdehyde groups into synthetic oligonucleotides
1996, Vol. 61, Special Issue, pp. S210–S212 [Abstract] - Ekaterina V. Efimtseva, Boris S. Ermolinsky, Marina V. Fomitcheva, Sergey V. Meshkov, Nelly Sh. Padyukova, Sergey N. Mikhailov, Arthur Van Aerschot, Jef Rozenski and Piet Herdewijn
Synthesis of disaccharide nucleosides and their incorporation into oligonucleotides
1996, Vol. 61, Special Issue, pp. S206–S209 [Abstract] - Mirella Marangoni, Arthur Van Aerschot, Patrick Augustijns and Piet A. Herdewijn
Cyclopentylethyl nucleosides as "constrained" acyclic building blocks for oligonucleotides
1996, Vol. 61, Special Issue, pp. S203–S205 [Abstract] - C. Pannecouque, K. Van Poppel, Arthur Van Aerschot and Piet Herdewijn
Synthesis and physicochemical properties of oligonucleotides with an N-cyanoguanidine function instead of the natural phosphate internucleotide linkage
1993, Vol. 58, Special Issue, pp. S191–S194 [Abstract] - Arthur Van Aerschot, F. Vandendriessche, K. Augustyns and Piet Herdewijn
Acyclic nucleosides: Useful for antisense constructs or as universal analogues for degenerate positions?
1993, Vol. 58, Special Issue, pp. S98–S101 [Abstract] - Ilse Verheggen, Nathalie Pillet, Arthur Van Aerschot, Erik De Clercq and Piet Herdewijn
Synthesis and anti-herpesvirus activity of nucleosides with a 1,5-anhydrohexitol moiety
1993, Vol. 58, Special Issue, pp. S64–S67 [Abstract] - Serge Van Calenbergh, Christophe Verlinde, André De Bruyn, Mia Callens, Elfride Van Den Eeckhout, Arthur Van Aerschot, Paul Michels, Fred Opperdoes, Wim Hol and Piet Herdewijn
2'-Substituted adenosine analogues as trypanosomal glyceraldehyde phosphate dehydrogenase (GAPDH) inhibitors
1993, Vol. 58, Special Issue, pp. S52–S55 [Abstract] - Tadeusz Kulikowski, Jaroslaw Poznanski, Jan Balzarini, Arthur Van Aerschot and Erik De Clercq
Synthesis, conformation and anti-HIV activity of 3'-substituted 2',3'-dideoxy-5-hydroxymethyluridines
1993, Vol. 58, Special Issue, pp. S44–S46 [Abstract] - Arthur Van Aerschot, Liu Jie, Jan Balzarini, Erik De Clercq and Piet Herdewijn
5'-O-Phosphonomethyl-2',3'-dideoxynucleosides: Synthesis and anti-HIV activity
1990, Vol. 55, Special Issue, pp. S129–S132 [Abstract] - Sergey N. Mikhailov and Leon N. Beigelman
Transient protection in nucleoside synthesis using trityl groups: Is it necessary to block hydroxyl groups?
1990, Vol. 55, Special Issue, pp. S105–S108 [Abstract] - Ivan I. Fedorov, Yaroslav E. Bezchinsky, Nikolay A. Novikov, Emma M. Kazmina, Marina V. Fomitcheva and Sergey N. Mikhailov
Syntheses of 3'-C-methyl-2'-deoxypyrimidine nucleosides
1990, Vol. 55, Special Issue, pp. S25–S28 [Abstract] - Mikko Oivanen, Tuula Viinamäki, Sergei Zavgorodny, Michael Polianski, Alex Azhayev, Arthur Van Aerschot, Piet Herdewijn and Harri Lönnberg
Hydrolytic stability of potential antiviral nucleoside analogues: 3'-Substituted 2',3'-dideoxy- and 2',3'-didehydro-2',3'-dideoxyribonucleosides
1990, Vol. 55, Special Issue, pp. S17–S20 [Abstract] - Piet Wigerinck, Paul Claes, Arthur Van Aerschot and Piet Herdewijn
Heterocycles in the 5-position of 2'-deoxyuridine
1990, Vol. 55, Special Issue, pp. S5–S8 [Abstract] - Marat Yu. Karpeisky, Leon N. Beigelman, Sergey N. Mikhailov, Nelly Sh. Padyukova and Jiří Smrt
Synthesis of adenylyl-(2'→5')adenylyl-(2'→5')adenosine
1982, Vol. 47, Issue 1, pp. 156–166 [Abstract]