Collect. Czech. Chem. Commun. 2008, 73, 1-18
https://doi.org/10.1135/cccc20080001

New Hydrophobicity Constants of Substituents in Pyrazine Rings Derived from RP-HPLC Study

Marta Kučerová-Chlupáčováa, Veronika Opletalováa,*, Josef Jampílekb, Jan Doležela, Jiří Dohnalb, Milan Pourc, Jiří Kunešc and Viktor Voříšekd

a Department of Pharmaceutical Chemistry and Drug Control, Faculty of Pharmacy, Charles University, Heyrovského 1203, CZ-500 05 Hradec Králové, Czech Republic
b Zentiva a.s., U kabelovny 130, CZ-102 37 Prague 10, Czech Republic
c Department of Inorganic and Organic Chemistry, Faculty of Pharmacy, Charles University, Heyrovského 1203, CZ-500 05 Hradec Králové, Czech Republic
d Institute of Clinical Biochemistry and Diagnostics, University Hospital, Sokolská 581, CZ-500 05 Hradec Králové, Czech Republic

Individual author index pages


Other CCCC articles of these authors

  • Vojtěch Balšánek, Lucie Tichotová, Jiří Kuneš, Marcel Špulák, Milan Pour*, Ivan Votruba and Vladimír Buchta
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  • Ivan Šnajdr, Jan Pavlík, Radan Schiller, Jiří Kuneš and Milan Pour*
    Pentenolide Analogues of Antifungal Butenolides: Strategies Towards 3,6-Disubstituted Pyranones and Unexpected Loss of Biological Effect
    2007, Vol. 72, Issue 11, pp. 1472–1498 [Abstract]
  • Veronika Opletalová*, Milan Pour, Jiří Kuneš, Vladimír Buchta, Luís Silva, Katarína Kráľová, Marta Chlupáčová, Dana Meltrová, Milan Peterka and Martina Posledníková
    Synthesis and Biological Evaluation of (E)-3-(Nitrophenyl)-1-(pyrazin-2-yl)prop-2-en-1-ones
    2006, Vol. 71, Issue 1, pp. 44–58 [Abstract]
  • Jiří Kuneš, Vojtěch Balšánek, Milan Pour* and Vladimír Buchta
    Synthesis and Antifungal Activity Evaluation of 3-Hetaryl-2,5-dihydrofuran-2-ones. An Unusual Fragmentation of the Oxazole Ring via 2,3-Selenoxide Shift
    2001, Vol. 66, Issue 12, pp. 1809–1830 [Abstract]
  • Karel Waisser*, Miloš Macháček, Hynek Dostál, Jiří Gregor, Lenka Kubicová, Věra Klimešová, Jiří Kuneš, Karel Palát, Jr., Jana Hladůvková, Jarmila Kaustová and Ute Möllmann
    Relationships Between the Chemical Structure of Substances and Their Antimycobacterial Activity Against Atypical Strains. Part 18. 3-Phenyl-2H-1,3-benzoxazine-2,4(3H)-diones and Isosteric 3-Phenylquinazoline-2,4(1H,3H)-diones
    1999, Vol. 64, Issue 11, pp. 1902–1924 [Abstract]
  • Věra Klimešová*, Martin Svoboda, Karel Waisser, Milan Pour and Jarmila Kaustová
    Synthesis and Antimicrobial Activity of New 4-(Benzylsulfanyl)pyridine Derivatives
    1999, Vol. 64, Issue 2, pp. 417–434 [Abstract]
  • Jiří Kuneš, Jiří Jáchym, Petr Jirásko, Želmíra Odlerová and Karel Waisser
    Combination of the Topliss Approach with the Free-Wilson Analysis in the Study of Antimycobacterial Activityof 4-Alkylthiobenzanilides
    1997, Vol. 62, Issue 9, pp. 1503–1510 [Abstract]
  • Veronika Opletalová, Asmita Patel, Michael Boulton, Alice Dundrová, Eva Lacinová, Marta Převorová, Martina Appeltauerová and Milada Coufalová
    5-Alkyl-2-pyrazinecarboxamides, 5-Alkyl-2-pyrazinecarbonitriles and 5-Alkyl-2-acetylpyrazines as Synthetic Intermediates for Antiinflammatory Agents
    1996, Vol. 61, Issue 7, pp. 1093–1101 [Abstract]
  • Karel Waisser, Jiří Kuneš, Alexandr Hrabálek, Miloš Macháček and Želmíra Odlerová
    New Groups of Potential Antituberculotics: 5-Alkylthio-1-aryltetrazoles
    1996, Vol. 61, Issue 5, pp. 791–798 [Abstract]
  • Veronika Opletalová, Jiří Hartl, Asmita Patel and Michael Boulton
    Homolytic Acetylation of 2,5-Dimethylpyrazine
    1995, Vol. 60, Issue 9, pp. 1551–1554 [Abstract]
  • Karel Waisser, Jiří Kuneš, Alexandr Hrabálek and Želmíra Odlerová
    New Groups of Potential Antituberculotics: Bis(1-aryltetrazol-5-yl) Disulfides. Structure Activity Relationship
    1994, Vol. 59, Issue 1, pp. 234–238 [Abstract]
  • Karel Waisser, Jiří Kuneš, Jiří Klimeš, Miroslav Polášek and Želmíra Odlerová
    Relations between Structure and Antituberculotic Activity of 4-Alkoxybenzoic Acids
    1993, Vol. 58, Issue 1, pp. 191–196 [Abstract]
  • Karel Waisser, Jiří Kuneš and Želmíra Odlerová
    Correlation of structural parameters with antituberculotic activity in a group of 2-benzamidobenzothiazoles
    1991, Vol. 56, Issue 12, pp. 2978–2985 [Abstract]
  • Pavel Seichter, Jiří Dohnal and František Rieger
    Process characteristics of screw impellers with a draught tube for Newtonian liquids. The power input
    1981, Vol. 46, Issue 9, pp. 2007–2020 [Abstract]