Collection Symposium Series 2008, 10, 87-93
https://doi.org/10.1135/css200810087
Published online 2015-10-30 18:35:35

From M. tuberculosis thymidine monophosphate kinase (TMPKmt) inhibitors towards mitochondrial thymidine kinase (TK-2) inhibitors

Serge Van Calenbergh, Ineke Van Daele, Sara Van Poecke, Matheus Froeyen, Hélene Munier Lehmann and Jan Balzarini

Individual author index pages


Other CCCC articles of these authors

  • Serge Van Calenbergh, Andreas Link, Shelly Fujikawa, Veerle Vanheusden, Denis De Keukeleire, Adriaan P. Ijzerman and Piet Herdewijn
    5'-Deoxy congeners of 9-(3-amido-3-deoxy-β-D-xylofuranosyl)-N6-cyclopentyladenine: New adenosine A1 receptor antagonists
    Symposium Series 1999, Vol. 2, pp. 273–276 [Abstract]
    Published online 2016-05-08 23:32:32
  • Philippe Van Rompaey, Vanheusden Veerle, Sylvie Pochet, Hélene Munier-Lehmann, Matheus Froeyen, Piet Herdewijn and Serge Van Calenbergh
    Thymidine (monophosphate) analogues as Mycobacterium tuberculosis thymidylate kinase inhibitors
    Symposium Series 2002, Vol. 5, pp. 393–395 [Abstract]
    Published online 2016-01-25 20:52:11
  • Philippe Van Rompaey, Kenneth A. Jacobson, Zhan-Guo Gao, Aishe Chen, Dov Barak, Soon-Ai Kim, Kyeong Lee, Andreas Link, Bruce T. Liang, Piet Herdewijn and Serge Van Calenbergh
    Amine-modified nucleosides as adenosine A3 neoceptor ligands
    Symposium Series 2002, Vol. 5, pp. 267–271 [Abstract]
    Published online 2016-01-25 20:41:17
  • Liesbet Cosyn, Kenneth A. Jacobson and Serge Van Calenbergh
    2-(1,2,3-Triazol-1-yl) N6-CH3-substituted adenosine derivatives: Highly potent and selective A3 receptor ligands
    Symposium Series 2005, Vol. 7, pp. 393–394 [Abstract]
    Published online 2015-11-08 11:56:11
  • Ineke Van Daele, Hélene Munier-Lehmann and Serge Van Calenbergh
    Exploring high affinity inhibitors of M. tuberculosis thymidiylate kinase
    Symposium Series 2005, Vol. 7, pp. 313–314 [Abstract]
    Published online 2015-11-08 11:54:32
  • Chris Meier, Christian Ducho, Henning Jessen and Jan Balzarini
    Esterase-cleavable cycloSal-pronucleotides – the trapping concept
    Symposium Series 2005, Vol. 7, pp. 105–113 [Abstract]
    Published online 2015-11-08 11:50:56
  • Tatjana Gazivoda, Silvana Raić-Malić, Sandra Kraljević-Pavelić, Krešimir Pavelić, Jan Balzarini and Mladen Mintas
    The new unsaturated acyclic C-5 pyrimidine nucleoside analogues: synthesis, cytostatic and anti-HIV evaluations
    Symposium Series 2008, Vol. 10, pp. 439–441 [Abstract]
    Published online 2015-10-30 18:44:36
  • Marcela Krečmerová, Antonín Holý, Alois Pískala, Graciela Andrei, Robert Snoeck, Jan Balzarini and Erik De Clercq
    New antiviral agent, 1-(S)-[3-hydroxy-2-(phosphonomethoxy)propyl]-5-azacytosine: esters and base-modified derivatives
    Symposium Series 2008, Vol. 10, pp. 196–200 [Abstract]
    Published online 2015-10-30 18:37:33
  • Sara Van Poecke, Matt Barrett, Kenneth A. Jacobson, T. Kendall Harden and Serge Van Calenbergh
    Synthesis of base-substituted uridine 5'-phosphonate analogues as potential P2Y2 receptor ligands
    Symposium Series 2011, Vol. 12, pp. 485–486 [Abstract]
    Published online 2015-08-20 10:25:20
  • Kiran Toti, Jan Balzarini and Serge Van Calenbergh
    Dideoxyapiose nucleosides revisited: syntheses and protide derivatives
    Symposium Series 2011, Vol. 12, pp. 480–482 [Abstract]
    Published online 2015-08-20 10:25:10
  • Tomáš Tichý, Graciela Andrei, Martin Dračínský, Antonín Holý, Jan Balzarini, Robert Snoeck and Marcela Krečmerová
    New amphiphilic prodrugs of adefovir and cidofovir
    Symposium Series 2011, Vol. 12, pp. 477–479 [Abstract]
    Published online 2015-08-20 10:25:04
  • Irina D. Konstantinova, Olga M. Selezneva, Ilja V. Fateev, Tamara A. Balashova, Svetlana K. Kotovskaya, Zoya M. Baskakova, Valery N. Charushin, Alexander V. Baranovsky, Anatoly I. Miroshnikov, Jan Balzarini and Igor A. Mikhailopulo
    Chemo-enzymatic syntheses and biological evaluation of 5,6-disubstituted benzimidazole ribo- and 2'-deoxyribo-nucleosides
    Symposium Series 2011, Vol. 12, pp. 400–402 [Abstract]
    Published online 2015-08-20 10:20:32
  • Chris Meier, Edwuin Hander Rios Morales, Cristina Arbelo Román and Jan Balzarini
    Stereoselective synthesis of 3-methyl-cycloSal-nucleotides
    Symposium Series 2011, Vol. 12, pp. 33–41 [Abstract]
    Published online 2015-08-20 09:58:11
  • Anastasia Parchina, Matheus Froeyen, Lia Margamuljana, Jef Rozenski, Steven de Jonghe, Yves Briers, Rob Lavigne, Piet Herdewijn and Eveline Lescrinier
    Discovery of an acyclic nucleoside phosphonate that inhibits Mycobacterium Tuberculosis ThyX based on the binding mode of a 5-alkynyl substrate analogue
    Symposium Series 2014, Vol. 14, pp. 342–343 [Abstract]
    Published online 2015-07-06 23:07:34
  • Craig Sergeant, Jan Balzarini and Roman Dembinski
    Antiviral activity of 5-halofuropyrimidine nucleosides
    Symposium Series 2014, Vol. 14, pp. 209–212 [Abstract]
    Published online 2015-07-06 23:01:50
  • Matheus Froeyen, Hans De Winter and Piet Herdewijn*
    Conformational Analysis, Solvent-Accessible Surface and Geometric Extent of Inhibitors and Substrates
    2006, Vol. 71, Issue 6, pp. 842–858 [Abstract]
  • Hubert Hřebabecký, Jan Balzarini and Antonín Holý
    Preparation of Chloro and Sulfanyl Derivatives of 1-(2-Deoxy-4-C-hydroxymethyl-α-L-threo-Pentofuranosyl)uracil
    1997, Vol. 62, Issue 7, pp. 1114–1127 [Abstract]
  • Michal Hocek, Milena Masojídková, Antonín Holý, Graciela Andrei, Robert Snoeck, Jan Balzarini and Erik De Clercq
    Synthesis and Antiviral Activity of Acyclic Nucleotide Analogues Derived from 6-(Aminomethyl)purines and Purine-6-carboxamidines
    1996, Vol. 61, Issue 10, pp. 1525–1537 [Abstract]
  • Serge Van Calenbergh, Christophe Verlinde, André De Bruyn, Mia Callens, Elfride Van Den Eeckhout, Arthur Van Aerschot, Paul Michels, Fred Opperdoes, Wim Hol and Piet Herdewijn
    2'-Substituted adenosine analogues as trypanosomal glyceraldehyde phosphate dehydrogenase (GAPDH) inhibitors
    1993, Vol. 58, Special Issue, pp. S52–S55 [Abstract]
  • Tadeusz Kulikowski, Jaroslaw Poznanski, Jan Balzarini, Arthur Van Aerschot and Erik De Clercq
    Synthesis, conformation and anti-HIV activity of 3'-substituted 2',3'-dideoxy-5-hydroxymethyluridines
    1993, Vol. 58, Special Issue, pp. S44–S46 [Abstract]
  • Arthur Van Aerschot, Liu Jie, Jan Balzarini, Erik De Clercq and Piet Herdewijn
    5'-O-Phosphonomethyl-2',3'-dideoxynucleosides: Synthesis and anti-HIV activity
    1990, Vol. 55, Special Issue, pp. S129–S132 [Abstract]