Collection Symposium Series 1999, 3, 79-81
https://doi.org/10.1135/css199903079
Published online 2016-03-16 22:55:09

Synthesis of library of HIV proteases inhibitors

Martin Hradilek, Markéta Rinnová, Cyril Bařinka, Milan Souček and Jan Konvalinka

Individual author index pages


Other CCCC articles of these authors

  • Bohumír Koutek, Lubomír Musil, Libuše Pavlíčková, Soňa Vašíčková and Milan Souček
    IR spectra of some quinone methides. Transmission of electronic effects in cross-conjugated systems
    1979, Vol. 44, Issue 10, pp. 2970–2981 [Abstract]
  • Markéta Rinnová and Ivan Rosenberg
    3'-N-phosphonomethyl derivatives of pyrrolidine nucleosides related to L-nucleotides
    Symposium Series 1999, Vol. 2, pp. 60–62 [Abstract]
    Published online 2016-05-08 20:41:05
  • Markéta Rinnová, Michaela Nováková, Václav Kašička and Jiří Jiráček
    Side reactions during photochemical cleavage of α-methyl-6-nitroveratryl-based photolabile linker
    Symposium Series 1999, Vol. 3, pp. 97–99 [Abstract]
    Published online 2016-03-16 22:55:38
  • Václav Vaněk, Miloš Buděšínský, Ivana Kavenová, Markéta Rinnová and Ivan Rosenberg
    Isosteric phosphonate-pyrrolidine-based dinucleoside monophosphate analogues
    Symposium Series 2002, Vol. 5, pp. 391–392 [Abstract]
    Published online 2016-01-25 20:52:06
  • Petr Kočalka, Markéta Rinnová, Václav Vaněk, Dominik Rejman, Ivan Votruba, Ivana Tomečková, Šárka Králíková, Magdalena Petrová, Ondřej Páv, Radek Pohl, Miloš Buděšínský, Radek Liboska, Zdeněk Točík and Ivan Rosenberg
    Novel nucleoside phosphonic acids-based inhibitors of thymidine phosphorylase
    Symposium Series 2005, Vol. 7, pp. 415–416 [Abstract]
    Published online 2015-11-08 11:56:57
  • Dušan Koval, Jana Jirásková, Kvido Stříšovský, Jan Konvalinka and Václav Kašička
    Capillary electrophoresis assay for D-serine
    Symposium Series 2005, Vol. 8, pp. 50–53 [Abstract]
    Published online 2015-11-06 12:01:51
  • Hillary E. Hoffman, Jana Jirásková, Marketa Zvelebil and Jan Konvalinka*
    Random mutagenesis of human serine racemase reveals residues important for the enzymatic activity
    2010, Vol. 75, Issue 1, pp. 59–79 [Abstract] [Full text pdf]
  • Milan Kožíšek, Jana Prejdová, Milan Souček, Ladislav Machala, Marie Staňková, Marek Linka, Marie Brůčková and Jan Konvalinka*
    Characterisation of Mutated Proteinases Derived from HIV-Positive Patients: Enzyme Activity, Vitality and Inhibition
    2004, Vol. 69, Issue 3, pp. 703–714 [Abstract]
  • Zbyněk Matušina, Radomíra Olbřímková, Hana Votavová, Josef Neumann, Martin Hradilek, Milan Souček, Petr Maloň, Milan Kodíček and Ivan Stibor*
    Linear Heptapeptides Containing DNA-Intercalators. Synthesis and Interaction with DNA
    1999, Vol. 64, Issue 9, pp. 1419–1432 [Abstract]
  • Kateřina Brožková, Ivana Křížová, Libuše Pavlíčková, Martin Hradilek, Martin Fusek, Tomáš Ruml, Milan Souček and Iva Pichová*
    Peptidomimetic Inhibitors of Extracellular Aspartic Proteinases of Candida albicans and Candida tropicalis
    1999, Vol. 64, Issue 1, pp. 130–137 [Abstract]
  • Jaroslav Litera, Jan Weber, Ivana Křížová, Iva Pichová, Jan Konvalinka, Martin Fusek and Milan Souček
    Peptide Inhibitors of Aspartic Proteinases with Hydroxyethylene Isostere Replacement of Peptide Bond. II. Preparation of Pseudotetrapeptides Derived from Diastereoisomeric 5-Amino-2-benzyl-4-hydroxy-6-phenylhexanoic Acids
    1998, Vol. 63, Issue 4, pp. 541–548 [Abstract]
  • Jaroslav Litera, Miloš Buděšínský, Ján Urban and Milan Souček
    Peptide Inhibitors of Aspartic Proteinases with Hydroxyethylene Isostere Replacement of Peptide Bond. I. Preparation of Four Diastereoisomeric (2R or 2S,4R or 4S,5S)-2-Benzyl-5-[(tert-butoxycarbonyl)amino]-4-hydroxy-6-phenylhexanoic Acids
    1998, Vol. 63, Issue 2, pp. 231–244 [Abstract]
  • Markéta Rinnová and Michal Lebl
    Molecular Diversity and Libraries of Structures: Synthesis and Screening
    1996, Vol. 61, Issue 2, pp. 171–231 [Abstract]
  • Milan Souček and Ján Urban
    An Efficient Method for Preparation of Optically Active N-Protected α-Amino Aldehydes from N-Protected α-Amino Alcohols
    1995, Vol. 60, Issue 4, pp. 693–696 [Abstract]
  • Stanislav Böhm, Richard Kubík, Martin Hradilek, Jan Němeček, Michal Hušák, Bohumil Kratochvíl and Josef Kuthan
    Sterically Crowded Heterocycles. II. Conformational Structure of 2-Phenyl-3-[(Z)-1,3-diphenyl-3-oxopropenyl]imidazo[1,2-a]pyridine and Related Compounds
    1995, Vol. 60, Issue 1, pp. 115–126 [Abstract]
  • Stanislav Böhm, Richard Kubík, Martin Hradilek, Jan Němeček, Michal Hušák, Svetlana Pakhomova, Jan Ondráček, Bohumil Kratochvíl and Josef Kuthan
    Sterically Crowded Heterocycles. I. Molecular Structure of 3-Chain Substituted 2-Phenylimidazo[1,2-a]pyridinium Salts
    1994, Vol. 59, Issue 12, pp. 2677–2690 [Abstract]
  • Milan Souček, Ján Urban and David Šaman
    Preparation of N-protected α-amino alcohols by acetoxyborohydride reduction of N-protected α-amino acid esters
    1990, Vol. 55, Issue 3, pp. 761–765 [Abstract]
  • Ján Urban, Petr Kuzmič, David Šaman and Milan Souček
    Regioselectivity of nucleophilic aromatic photosubstitution in the biphenyl series. Photohydrolysis of some dimethoxynitrobiphenyls
    1987, Vol. 52, Issue 10, pp. 2482–2491 [Abstract]
  • Petr Kuzmič, Libuše Pavlíčková and Milan Souček
    Photoreaction of N-butyl 3,4-dimethoxy-6-nitrobenzamide with butylamine. A model study for lysine-directed photoaffinity labelling
    1987, Vol. 52, Issue 7, pp. 1780–1785 [Abstract]
  • Petr Kuzmič and Milan Souček
    Substituent effects in aromatic photochemistry. UV irradiation of 3,4-dimethoxybenzonitrile and 3,4-dimethoxyacetophenone in the presence of inorganic anions
    1987, Vol. 52, Issue 4, pp. 980–988 [Abstract]
  • Petr Kuzmič, Libuše Pavlíčková, Jiří Velek and Milan Souček
    Photoreaction of 3,4-dimethoxy-1-nitrobenzene with butylamine. A pH dependence of regioselectivity
    1986, Vol. 51, Issue 8, pp. 1665–1670 [Abstract]
  • Petr Kuzmič, Libuše Pavlíčková and Milan Souček
    Photochemical hydrolysis of some nitrophenyl acetates
    1986, Vol. 51, Issue 6, pp. 1293–1300 [Abstract]
  • Libuše Pavlíčková, Petr Kuzmič and Milan Souček
    Chemical actinometry in the UV range based on the photohydrolysis of 3,4-dimethoxynitrobenzene
    1986, Vol. 51, Issue 2, pp. 368–374 [Abstract]
  • Petr Kuzmič and Milan Souček
    Photocyanation of 3,4-dimethoxy-1-nitrobenzene. A quantitative study
    1986, Vol. 51, Issue 2, pp. 358–367 [Abstract]
  • Bohumír Koutek, Lubomír Musil, Jiří Velek and Milan Souček
    Fluorescence behaviour of some 4-substituted halobenzenes
    1985, Vol. 50, Issue 8, pp. 1753–1763 [Abstract]
  • Lubomír Musil, Bohumír Koutek, Jiří Velek and Milan Souček
    Substitution effect in electronic absorption spectra of 2- and 2,6-substituted 4-benzhydrylidene-2,5-cyclohexadien-1-ones
    1984, Vol. 49, Issue 9, pp. 1949–1964 [Abstract]
  • Lubomír Musil, Bohumír Koutek, Jiří Velek, Josef Krupička and Milan Souček
    CNDO/S MO study of the fuchsone derivatives with sterically crowded exocyclic double bond
    1983, Vol. 48, Issue 10, pp. 2825–2839 [Abstract]
  • Libuše Pavlíčková, Bohumír Koutek, Václav Jehlička and Milan Souček
    Solvatochromic study of internal charge transfer in 7,7-disubstituted quinone methides
    1983, Vol. 48, Issue 8, pp. 2376–2385 [Abstract]
  • Milena Píšová and Milan Souček
    Oxidative rearrangement of o-fuchsone to 2,2-diphenyl-1,3-benzodioxol
    1982, Vol. 47, Issue 12, pp. 3318–3327 [Abstract]
  • Bohumír Koutek, Milena Píšová, Josef Krupička, Antonín Lyčka, Dobroslav Šnobl and Milan Souček
    Benzoannelated quinone methides
    1982, Vol. 47, Issue 6, pp. 1645–1653 [Abstract]
  • Milena Píšová and Milan Souček
    Intermolecular cyclization of o-fuchsones
    1982, Vol. 47, Issue 3, pp. 838–842 [Abstract]
  • Bohumír Koutek, Libuše Pavlíčková, Miloš Buděšínský and Milan Souček
    Synthesis and properties of benzoannelated 6-(1,3-dithiolan-2-yliden)-2,4-cyclohexadien-1-ones
    1982, Vol. 47, Issue 1, pp. 59–64 [Abstract]
  • Bohumír Koutek, Lubomír Musil, Jiří Velek, Antonín Lyčka, Dobroslav Šnobl, Miroslava Synáčková and Milan Souček
    Perturbation of the fuchsone chromophore by 3,5-methyl substitution. Sterically crowded exocyclic double bond
    1981, Vol. 46, Issue 10, pp. 2540–2556 [Abstract]
  • Antonín Lyčka, Dobroslav Šnobl, Bohumír Koutek, Libuše Pavlíčková and Milan Souček
    13C NMR study of 7,7-disubstituted quinone methides
    1981, Vol. 46, Issue 9, pp. 2083–2090 [Abstract]
  • Jiří Velek, Bohumír Koutek, Lubomír Musil, Soňa Vašíčková and Milan Souček
    Basicity of fuchsones. Infrared study of the ν(OH) stretching vibration in phenol-fuchsone complexes
    1981, Vol. 46, Issue 8, pp. 1818–1827 [Abstract]
  • Antonín Lyčka, Dobroslav Šnobl, Bohumír Koutek, Libuše Pavlíčková and Milan Souček
    13C NMR study of substituted quinone methides. 2- and 2,6-substituted fuchsones
    1981, Vol. 46, Issue 8, pp. 1775–1787 [Abstract]
  • Lubomír Musil, Bohumír Koutek, Milena Píšová and Milan Souček
    Delocalization and stability of o- and p-quinone methides: A HMO study
    1981, Vol. 46, Issue 5, pp. 1148–1159 [Abstract]
  • Jiří Velek, Bohumír Koutek, Lubomír Musil, Soňa Vašíčková and Milan Souček
    IR spectra of some quinone methides. A study of the ortho-effect
    1981, Vol. 46, Issue 4, pp. 873–882 [Abstract]
  • Josef Krupička, Bohumír Koutek, Lubomír Musil, Libuše Pavlíčková and Milan Souček
    Half-wave potentials of quinone methides in dimethylformamide: Substituent effects
    1981, Vol. 46, Issue 4, pp. 861–872 [Abstract]
  • Libuše Pavlíčková, Soňa Vašíčková and Milan Souček
    Synthesis and properties of 7,7-diaminoquinone methides
    1980, Vol. 45, Issue 10, pp. 2675–2683 [Abstract]
  • Miroslav Havel, Jiří Velek, Jan Pospíšek and Milan Souček
    Selective acylation of hydroxy steroids with acyl cyanides
    1979, Vol. 44, Issue 8, pp. 2443–2446 [Abstract]
  • Libuše Pavlíčková and Milan Souček
    Preparation and reactions of 5,7-ditert-butyl-1,2-diphenylspiro[2,5]octa-1,4,7-trien-6-one: A revision of the literature
    1979, Vol. 44, Issue 6, pp. 1810–1818 [Abstract]
  • Jiří Velek, Bohumír Koutek and Milan Souček
    Mechanism of hydration and isomerisation of 4-ethylidene-2,6-di-tert-butyl-2,5-cyclohexadien-1-one. Kinetics, acid-base catalysis and solvent deuterium isotope effects
    1979, Vol. 44, Issue 1, pp. 110–122 [Abstract]